Molecular analysis of the site for 2-arachidonylglycerol (2-AG) on the β2 subunit of GABAA receptors

Journal of Neurochemistry

Volumn 126, Issue 1, 2013, Pages 29-36

  Baur, Roland ^a   Kielar, Marie ^a   Richter, Lars ^c   Ernst, Margot ^b   Ecker, Gerhard F ^c   Sigel, Erwin ^a  

^a UNIVERSITY OF BERN   (Switzerland)

^b MEDICAL UNIVERSITY OF VIENNA   (Austria)

^c UNIVERSITY OF VIENNA   (Austria)

Author keywords

2 arachidonylglycerol (2 AG); endocannabinoids; GABA; GABAA receptors

Indexed keywords

2 ARACHIDONOYLGLYCEROL; 4 AMINOBUTYRIC ACID A RECEPTOR BETA2; CYSTEINE; MUTANT PROTEIN;

ALPHA HELIX; AMINO ACID SEQUENCE; ANIMAL CELL; ARTICLE; CONTROLLED STUDY; DRUG TARGETING; FEMALE; HYDROPHOBICITY; MOLECULAR DOCKING; MOLECULAR MODEL; NONHUMAN; PRIORITY JOURNAL; PROTEIN STRUCTURE;

ANIMALS; ARACHIDONIC ACIDS; BINDING SITES; CYSTEINE; DOSE-RESPONSE RELATIONSHIP, DRUG; ENDOCANNABINOIDS; ETHANOLAMINES; FATTY ACIDS, UNSATURATED; FEMALE; GLYCERIDES; HUMANS; KINETICS; MODELS, MOLECULAR; MUTATION; OOCYTES; POINT MUTATION; POLYUNSATURATED ALKAMIDES; RECEPTOR, CANNABINOID, CB1; RECEPTORS, GABA-A; XENOPUS LAEVIS;

EID: 84879411618     PISSN: 00223042     EISSN: 14714159     Source Type: Journal    
DOI: 10.1111/jnc.12270     Document Type: Article

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