2-aminothiophene-3-carboxylic acid ester derivatives as novel highly selective cytostatic agents

Investigational New Drugs

Volumn 32, Issue 1, 2014, Pages 200-210

  Balzarini, J ^a   Thomas, J ^b   Liekens, S ^a   Noppen, S ^a   Dehaen, W ^b   Romagnoli, R ^c  

^a REGA INSTITUTE FOR MEDICAL RESEARCH   (Belgium)

^b UNIVERSITY OF LEUVEN   (Belgium)

^c UNIVERSITY OF FERRARA   (Italy)

Author keywords

2 aminothiophene 3 carboxylic acid esters; Cytostatic selectivity; Hepatoma and prostate carcinoma; Kidney carcinoma; T lymphoma

Indexed keywords

AMINO ACIDS; APOPTOSIS; CELL CYCLE; CELL LINE, TUMOR; CYTOSTATIC AGENTS; ESTERS; HUMANS; NEOPLASMS; STRUCTURE-ACTIVITY RELATIONSHIP; THIOPHENES;

EID: 84899061866     PISSN: 01676997     EISSN: 15730646     Source Type: Journal    
DOI: 10.1007/s10637-013-9981-4     Document Type: Article

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