SCOPUS 정보 검색 플랫폼

Volumn 9, Issue 2, 2014, Pages 337-349

A new sif-dipropargyl glycerol scaffold as a versatile prosthetic group to design dimeric radioligands: Synthesis of the [18f]bmppsif tracer to image serotonin receptors

(8) Hazari, Puja Panwar a Schulz, Jurgen b Vimont, Delphine b Chadha, Nidhi a Allard, Michele b Szlosek Pinaud, Magali c Fouquet, Eric c Mishra, Anil Kumar a

a INMAS DRDO Division of Cyclotron and Radiopharmaceutical Sciences (India)

b UMR 5287 (France)

c INSTITUT DES SCIENCES MOLÉCULAIRES (France)

Author keywords

Click Chemistry; Fluorides; Ligand Design; Radiolabeling; Silicon

Indexed keywords

1 (2 AZIDOETHYL) 4 (2 METHOXYPHENYL)PIPERAZINE; 1 (2 HYDROXYETHYL) 4 (2 METHOXYPHENYL)PIPERAZINE; 3 [4 (DI TERT BUTYLSILYL]PHENOXY)PROPANE 1,2 DIOL; 4 (DI TERT BUTYLSILANYL)PHENOL; BMPPSIF F 18; DI TERT BUTYL[4 [(2,2 DIMETHYL 1,3 DIOXOLAN 4 YL)METHOXY]PHENYL] SILANE; GLYCEROL; RADIOLIGAND; SEROTONIN 1A RECEPTOR; UNCLASSIFIED DRUG; [4 [2,3 BIS(PROP 2 YNYLOXY)PROPOXY]PHENYL]DI TERT BUTYLSILANE;

ANIMAL EXPERIMENT; ARTICLE; BINDING AFFINITY; CHEMICAL STRUCTURE; CLICK CHEMISTRY; CYTOTOXICITY ASSAY; FLUORINATION; HIPPOCAMPUS; ISOTOPE LABELING; MEASUREMENT; MOLECULAR DOCKING; NONHUMAN; NUCLEAR MAGNETIC RESONANCE SPECTROSCOPY; POSITRON EMISSION TOMOGRAPHY; PRIMARY CULTURE; PRIORITY JOURNAL; RAT; SYNTHESIS;

CLICK CHEMISTRY; FLUORIDES; LIGAND DESIGN; RADIOLABELING; SILICON;

ANIMALS; BRAIN; BRAIN CHEMISTRY; DIMERIZATION; FLUORINE RADIOISOTOPES; GLYCEROL; LIGANDS; MOLECULAR DOCKING SIMULATION; ORGANOSILICON COMPOUNDS; POSITRON-EMISSION TOMOGRAPHY; RATS; RATS, SPRAGUE-DAWLEY; RECEPTOR, SEROTONIN, 5-HT1A;

EID: 84897022102 PISSN: 18607179 EISSN: 18607187 Source Type: Journal
DOI: 10.1002/cmdc.201300458 Document Type: Article

Times cited : (17)

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