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Volumn 28, Issue 2, 2001, Pages 177-185

New halogenated [11C]WAY analogues, [11C]6FPWAY and [11C]6BPWAY-Radiosynthesis and assessment as radioligands for the study of brain 5-HT1A receptors in living monkey

(11) Sandell, Johan a Halldin, Christer a Pike, Victor W b Chou, Yuan Hwa a Varnäs, Katarina a Hall, Håkan a Marchais, Sandrine c Nowick, Bartek c Wikström, Håkan V c Swahn, Carl Gunnar a Farde, Lars a

a KAROLINSKA UNIVERSITY HOSPITAL (Sweden)

b HAMMERSMITH HOSPITAL (United Kingdom)

c UNIVERSITY MEDICAL CENTER GRONINGEN (Netherlands)

Author keywords

5 HT1A receptor; Human brain autoradiography; Monkey brain; PET; Radioligand; 11C 6BPWAY; 11C 6FPWAY

Indexed keywords

AMINOPYRIDINE DERIVATIVE; CARBON; DIAGNOSTIC AGENT; N (2 (1 (4 (2 METHOXYPHENYL) PIPERAZINYL)ETHYL)) N (2 (6 FLUOROPYRIDINYL))CYCLOHEXANECARBOXAMIDE; N (2 (1 (4 (2 METHOXYPHENYL)PIPERAZINYL)ETHYL)) N (2 (6 BROMOPYRIDINYL))CYCLOHEXANECARBOXAMIDE; N [2 [4 (2 METHOXYPHENYL) 1 PIPERAZINYL]ETHYL] N (2 PYRIDYL)CYCLOHEXANECARBOXAMIDE; N-(2-(1-(4-(2-METHOXYPHENYL)-PIPERAZINYL)ETHYL))-N-(2-(6-FLUOROPYRIDINYL))CYCLOHEXANECARBOXAMIDE; N-(2-(1-(4-(2-METHOXYPHENYL)PIPERAZINYL)ETHYL))-N-(2-(6-BROMOPYRIDINYL))CYCLOHEXANECARBOXAMIDE; PIPERAZINE DERIVATIVE; PYRIDINE DERIVATIVE; RADIOPHARMACEUTICAL AGENT; SEROTONIN 1 RECEPTOR; SEROTONIN ANTAGONIST; SEROTONIN RECEPTOR; CYCLOHEXANECARBOXYLIC ACID DERIVATIVE; FLUORINE 18; HALOCARBON; IODINE 123; N [2 [1 [4 (2 METHOXYPHENYL)PIPERAZINYL]ETHYL] N [2 (6 BROMOPYRIDINYL)]CYCLOHEXANECARBOXAMIDE C 11; N [2 [1 [4 (2 METHOXYPHENYL)PIPERAZINYL]ETHYL] N [2 (6 FLUOROPYRIDINYL)]CYCLOHEXANECARBOXAMIDE C 11; N [2 [4 (2 METHOXYPHENYL) 1 PIPERAZINYL]ETHYL] N (2 PYRIDYL)CYCLOHEXANECARBOXAMIDE C 11; RADIOLIGAND; SEROTONIN 1A RECEPTOR; UNCLASSIFIED DRUG;

ANIMAL; ARTICLE; AUTORADIOGRAPHY; BRAIN; BRAIN CORTEX; COMPUTER ASSISTED EMISSION TOMOGRAPHY; HIPPOCAMPUS; HUMAN; KINETICS; MACACA; METABOLISM; METHODOLOGY; SCINTISCANNING; SYNTHESIS; TISSUE DISTRIBUTION; ACYLATION; ANIMAL EXPERIMENT; BIOACCUMULATION; BRAIN TISSUE; CEREBELLUM; CONTROLLED STUDY; FRONTAL CORTEX; HUMAN TISSUE; ISOTOPE LABELING; METABOLITE; MONKEY; NONHUMAN; POSITRON EMISSION TOMOGRAPHY; RADIOACTIVITY; RAPHE NUCLEUS; RECEPTOR BINDING; TEMPORAL CORTEX;

AMINOPYRIDINES; ANIMALS; AUTORADIOGRAPHY; BRAIN; CARBON RADIOISOTOPES; CEREBRAL CORTEX; HIPPOCAMPUS; HUMANS; KINETICS; MACACA FASCICULARIS; PIPERAZINES; PYRIDINES; RADIOPHARMACEUTICALS; RECEPTORS, SEROTONIN; RECEPTORS, SEROTONIN, 5-HT1; SEROTONIN ANTAGONISTS; TISSUE DISTRIBUTION; TOMOGRAPHY, EMISSION-COMPUTED;

EID: 0034744763 PISSN: 09698051 EISSN: None Source Type: Journal
DOI: 10.1016/S0969-8051(00)00181-5 Document Type: Article

Times cited : (27)

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