Selective non-nucleoside inhibitors of human DNA methyltransferases active in cancer including in cancer stem cells

Journal of Medicinal Chemistry

Volumn 57, Issue 3, 2014, Pages 701-713

  Valente, Sergio ^a   Liu, Yiwei ^b   Schnekenburger, Michael ^c   Zwergel, Clemens ^a,d   Cosconati, Sandro ^e   Gros, Christina ^f   Tardugno, Maria ^a   Labella, Donatella ^a   Florean, Cristina ^c   Minden, Steven ^c   Hashimoto, Hideharu ^b   Chang, Yanqi ^b   Zhang, Xing ^b   Kirsch, Gilbert ^d   Novellino, Ettore ^g   Arimondo, Paola B ^f   Miele, Evelina ^a   Ferretti, Elisabetta ^a   Gulino, Alberto ^a   Diederich, Marc ^c,h   Cheng, Xiaodong ^b   Mai, Antonello ^a   more..

^a SAPIENZA UNIVERSITY OF ROME   (Italy)

^b EMORY UNIVERSITY SCHOOL OF MEDICINE   (United States)

^c LABORATOIRE DE BIOLOGIE MOLÉCULAIRE ET CELLULAIRE DU CANCER   (Luxembourg)

^d UNIVERSITÉ DE LORRAINE   (France)

^e SECOND UNIVERSITY OF NAPLES   (Italy)

^f INSTITUT DE RECHERCHE PIERRE FABRE   (France)

^g UNIVERSITY OF NAPLES FEDERICO II   (Italy)

^h Seoul National University   (South Korea)

Author keywords

[No Author keywords available]

Indexed keywords

AMINOQUINOLINES; ANIMALS; ANTINEOPLASTIC AGENTS; BENZAMIDES; CELL LINE, TUMOR; DNA (CYTOSINE-5-)-METHYLTRANSFERASE; DRUG SCREENING ASSAYS, ANTITUMOR; HUMANS; MICE; NEOPLASTIC STEM CELLS; PYRIMIDINES; QUINOLINES; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84894065301     PISSN: 00222623     EISSN: 15204804     Source Type: Journal    
DOI: 10.1021/jm4012627     Document Type: Article

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