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ChemBioChem

Volumn 14, Issue 16, 2013, Pages 2119-2125

Allosteric lariat peptide inhibitors of abl kinase

(4) Bharathikumar, V M a Barreto, Kris a Decoteau, John F a Geyer, C Ronald a

a UNIVERSITY OF SASKATCHEWAN (Canada)

Author keywords

Abl kinase; Combinatorial chemistry; Enzyme inhibitors; Lariat peptides; Uncompetitive inhibition

Indexed keywords

ABELSON KINASE; DASATINIB; IMATINIB; LARIAT PEPTIDE INHIBITOR; NILOTINIB; PROTEIN TYROSINE KINASE INHIBITOR; TOZASERTIB; UNCLASSIFIED DRUG;

AMINO ACID SEQUENCE; AMINO ACID SUBSTITUTION; ARTICLE; BINDING AFFINITY; CHRONIC MYELOID LEUKEMIA; CRYSTAL STRUCTURE; CYCLIZATION; DRUG BINDING; DRUG SCREENING; DRUG TARGETING; HUMAN; IC 50; MOLECULAR DOCKING; NONHUMAN; POINT MUTATION; PRIORITY JOURNAL; PROTEIN ANALYSIS; TRANSCRIPTION INITIATION;

ABL KINASE; COMBINATORIAL CHEMISTRY; ENZYME INHIBITORS; LARIAT PEPTIDES; UNCOMPETITIVE INHIBITION;

ADENOSINE TRIPHOSPHATE; ALLOSTERIC REGULATION; AMINO ACID SEQUENCE; BINDING SITES; CATALYTIC DOMAIN; CELL LINE, TUMOR; ENZYME ACTIVATION; HUMANS; KINETICS; PEPTIDES; PROTEIN BINDING; PROTEIN KINASE INHIBITORS; PROTO-ONCOGENE PROTEINS C-ABL;

EID: 84889590153 PISSN: 14394227 EISSN: 14397633 Source Type: Journal
DOI: 10.1002/cbic.201300253 Document Type: Article

Times cited : (9)

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