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Bioorganic Chemistry

Volumn 49, Issue , 2013, Pages 49-58

The adenosine A2A antagonistic properties of selected C8-substituted xanthines

(5) Van Der Walt, Mietha M a Terre'Blanche, Gisella a Petzer, Anél a Lourens, Anna C U a Petzer, Jacobus P a

a NORTH WEST UNIVERSITY (South Africa)

Author keywords

Antagonism; Haloperidol induced catalepsy; Parkinson's disease; Xanthine

Indexed keywords

8 (3 CHLOROSTYRYL)CAFFEINE; ADENOSINE A2A RECEPTOR ANTAGONIST; CAFFEINE; HALOPERIDOL; HETEROCYCLIC COMPOUND; ISTRADEFYLLINE; XANTHINE; ADENOSINE A2 RECEPTOR ANTAGONIST; ADENOSINE A2A RECEPTOR; AMINE OXIDASE (FLAVIN CONTAINING); ENZYME INHIBITOR; RECOMBINANT PROTEIN; XANTHINE DERIVATIVE;

ARTICLE; BINDING AFFINITY; CATALEPSY; CONTROLLED STUDY; DRUG EFFECT; IN VITRO STUDY; IN VIVO STUDY; MALE; NONHUMAN; PRIORITY JOURNAL; RAT; STRUCTURE ACTIVITY RELATION; CHEMICAL STRUCTURE; CHEMISTRY; DOSE RESPONSE; HUMAN; METABOLISM; SYNTHESIS;

RATTUS;

ADENOSINE A2 RECEPTOR ANTAGONISTS; DOSE-RESPONSE RELATIONSHIP, DRUG; ENZYME INHIBITORS; HUMANS; MOLECULAR STRUCTURE; MONOAMINE OXIDASE; RECEPTOR, ADENOSINE A2A; RECOMBINANT PROTEINS; STRUCTURE-ACTIVITY RELATIONSHIP; XANTHINES;

EID: 84885142896 PISSN: 00452068 EISSN: 10902120 Source Type: Journal
DOI: 10.1016/j.bioorg.2013.06.006 Document Type: Article

Times cited : (28)

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