FDA-approved drugs and other compounds tested as inhibitors of human glutathione transferase P1-1

Chemico-Biological Interactions

Volumn 205, Issue 1, 2013, Pages 53-62

  Musdal, Yaman ^a,b   Hegazy, Usama M ^a,c   Aksoy, Yasemin ^b   Mannervik, Bengt ^a,d  

^a UPPSALA UNIVERSITY   (Sweden)

^b HACETTEPE UNIVERSITY   (Turkey)

^c NATIONAL RESEARCH CENTRE   (Egypt)

^d STOCKHOLM UNIVERSITY   (Sweden)

Author keywords

Adjuvant chemotherapeutics; Enzyme inhibition; Ethacrynic acid; FDA approved drugs; Glutathione transferase; P1 1

Indexed keywords

AMPHOTERICIN B; ATOVAQUONE; AVOBENZONE; BITHIONATE SODIUM; CHLORAMPHENICOL PALMITATE; CHLOROPHYLLIDE; CLOFAZIMINE; CLOTRIMAZOLE; DIIODOHYDROXYQUIN; DITHRANOL; ECONAZOLE; ENZYME INHIBITOR; ERGOTAMINE TARTRATE; ESTRADIOL ACETATE; ESTRADIOL VALERATE; ETACRYNIC ACID; FENBENDAZOLE; FLUFENAMIC ACID; GLUTATHIONE TRANSFERASE A3 3 INHIBITOR; GLUTATHIONE TRANSFERASE P1; GLUTATHIONE TRANSFERASE P1 1 INHIBITOR; HEXACHLOROPHENE; MECLOZINE; MERBROMIN; NISOLDIPINE; OXICONAZOLE; SANGUINARINE SULFATE; SULCONAZOLE; TEMEFOS; UNCLASSIFIED DRUG;

ARTICLE; CONCENTRATION RESPONSE; DRUG APPROVAL; DRUG EFFICACY; DRUG POTENCY; DRUG SCREENING; DRUG STRUCTURE; ENZYME ACTIVITY; ENZYME SPECIFICITY; FOOD AND DRUG ADMINISTRATION; IC 50; PROTEIN EXPRESSION;

ADJUVANT CHEMOTHERAPEUTICS; ENZYME INHIBITION; ETHACRYNIC ACID; FDA-APPROVED DRUGS; GLUTATHIONE TRANSFERASE P1-1;

ANTINEOPLASTIC AGENTS; CHLOROPHYLLIDES; DRUG APPROVAL; DRUG EVALUATION, PRECLINICAL; DRUG RESISTANCE, NEOPLASM; ENZYME INHIBITORS; ETHACRYNIC ACID; GLUTATHIONE S-TRANSFERASE PI; GLUTATHIONE TRANSFERASE; HEXACHLOROPHENE; HUMANS; KINETICS; MERBROMIN; NEOPLASMS; RECOMBINANT PROTEINS; UNITED STATES; UNITED STATES FOOD AND DRUG ADMINISTRATION;

EID: 84885107829     PISSN: 00092797     EISSN: 18727786     Source Type: Journal    
DOI: 10.1016/j.cbi.2013.06.003     Document Type: Article

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