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European Journal of Medicinal Chemistry

Volumn 69, Issue , 2013, Pages 182-190

Synthesis and cytotoxic activity of some novel steroidal C-17 pyrazolinyl derivatives

(6) Fan, Ning Juan a Tang, Jiang Jiang a Li, He a Li, Xiao Jun a Luo, Bo a Gao, Jin Ming a

a NORTHWEST A F UNIVERSITY (China)

Author keywords

Cytotoxicity; Progesterone; Pyrazoline; Steroid; Steroidal heterocycles

Indexed keywords

17 (4,5 DIHYDRO 1 ACETYL 5 (2' CHLOROPHENYL) 3 PYRAZOLINYL)ANDROST 1,4 DIEN 3 ONE; 17 (4,5 DIHYDRO 1 ACETYL 5 (2' METHOXYPHENYL) 3 PYRAZOLINYL)ANDROST 1,4 DIEN 3 ONE; 17 (4,5 DIHYDRO 1 ACETYL 5 (2' NITROPHENYL) 3 PYRAZOLINYL)ANDROST 1,4 DIEN 3 ONE; 17 (4,5 DIHYDRO 1 ACETYL 5 (4' CHLOROPHENYL) 3 PYRAZOLINYL)ANDROST 1,4 DIEN 3 ONE; 17 (4,5 DIHYDRO 1 ACETYL 5 (4' METHOXYPHENYL) 3 PYRAZOLINYL)ANDROST 1,4 DIEN 3 ONE; 17 (4,5 DIHYDRO 1 ACETYL 5 (4' NITROPHENYL) 3 PYRAZOLINYL)ANDROST 1,4 DIEN 3 ONE; 17 (4,5 DIHYDRO 1 ACETYL 5 PHENYL 3 PYRAZOLINYL) 4 CHLOROANDROST 1,4 DIEN 3 ONE; 17 (4,5 DIHYDRO 1 ACETYL 5 PHENYL 3 PYRAZOLINYL)ANDROST 1,4 DIEN 3 ONE; 17 [4,5 DIHYDRO 1 ACETYL 5 (2' CHLOROPHENYL) 3 PYRAZOLINYL] 4 CHLOROANDROST 1,4 DIEN 3 ONE; 17 [4,5 DIHYDRO 1 ACETYL 5 (2' METHOXYPHENYL) 3 PYRAZOLINYL] 4 CHLOROANDROST 1,4 DIEN 3 ONE; 17 [4,5 DIHYDRO 1 ACETYL 5 (2' NITROPHENYL) 3 PYRAZOLINYL] 4 CHLOROANDROST 1,4 DIEN 3 ONE; 17 [4,5 DIHYDRO 1 ACETYL 5 (4' CHLOROPHENYL) 3 PYRAZOLINYL] 4 CHLOROANDROST 1,4 DIEN 3 ONE; 17 [4,5 DIHYDRO 1 ACETYL 5 (4' METHOXYPHENYL) 3 PYRAZOLINYL] 4 CHLOROANDROST 1,4 DIEN 3 ONE; 17 [4,5 DIHYDRO 1 ACETYL 5 (4' NITROPHENYL) 3 PYRAZOLINYL] 4 CHLOROANDROST 1,4 DIEN 3 ONE; ANTINEOPLASTIC AGENT; PROGESTERONE; PYRAZOLINYL DERIVATIVE; UNCLASSIFIED DRUG;

ANTINEOPLASTIC ACTIVITY; ARTEMIA SALINA; ARTICLE; CELL POPULATION; CONTROLLED STUDY; DRUG CYTOTOXICITY; DRUG SYNTHESIS; HUMAN; HUMAN CELL; IN VITRO STUDY; NONHUMAN; S PHASE CELL CYCLE CHECKPOINT; STRUCTURE ACTIVITY RELATION;

CYTOTOXICITY; PROGESTERONE; PYRAZOLINE; STEROID; STEROIDAL HETEROCYCLES;

ANIMALS; ANTINEOPLASTIC AGENTS; ARTEMIA; CELL CYCLE; CELL LINE, TUMOR; CELL PROLIFERATION; DOSE-RESPONSE RELATIONSHIP, DRUG; DRUG SCREENING ASSAYS, ANTITUMOR; HELA CELLS; HEP G2 CELLS; HUMANS; MOLECULAR STRUCTURE; PYRAZOLES; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84883633682 PISSN: 02235234 EISSN: 17683254 Source Type: Journal
DOI: 10.1016/j.ejmech.2013.08.016 Document Type: Article

Times cited : (37)

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