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Bioorganic and Medicinal Chemistry Letters

Volumn 23, Issue 18, 2013, Pages 5213-5216

Optimization of diarylazines as anti-HIV agents with dramatically enhanced solubility

(5) Bollini, Mariela a Cisneros, José A a Spasov, Krasimir A b Anderson, Karen S b Jorgensen, William L a

a YALE UNIVERSITY (United States)

b YALE UNIVERSITY SCHOOL OF MEDICINE (United States)

Author keywords

Anti HIV agent; Drug solubility; NNRTI

Indexed keywords

ANTI HUMAN IMMUNODEFICIENCY VIRUS AGENT; ETRAVIRINE; NEVIRAPINE; RILPIVIRINE;

ARTICLE; BINDING SITE; CRYSTAL STRUCTURE; DRUG BIOAVAILABILITY; DRUG SOLUBILITY; MOLECULAR WEIGHT; PH;

HUMAN IMMUNODEFICIENCY VIRUS 1;

ANTI-HIV AGENT; DRUG SOLUBILITY; NNRTI;

ANTI-HIV AGENTS; CELL LINE, TRANSFORMED; CELL PROLIFERATION; DOSE-RESPONSE RELATIONSHIP, DRUG; HIV-1; HUMANS; HYDRAZINES; MICROBIAL SENSITIVITY TESTS; MODELS, MOLECULAR; MOLECULAR STRUCTURE; SOLUBILITY; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84882672782 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2013.06.091 Document Type: Article

Times cited : (33)

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