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Bioorganic and Medicinal Chemistry Letters

Volumn 23, Issue 14, 2013, Pages 4253-4257

Design, synthesis and evaluation of inhibitor of apoptosis protein (IAP) antagonists that are highly selective for the BIR2 domain of XIAP

(12) Ardecky, Robert J a Welsh, Kate a Finlay, Darren a Lee, Pooi San a González López, Marcos a Ganji, Santhi Reddy a Ravanan, Palaniyandi a Mace, Peter D a Riedl, Stefan J a Vuori, Kristiina a Reed, John C a Cosford, Nicholas D P a

a BURNHAM INSTITUTE (United States)

Author keywords

Apoptosis; Monovalent Smac mimetics; Probe compounds; XIAP

Indexed keywords

APOPTOSIS INDUCING FACTOR; INHIBITOR OF APOPTOSIS PROTEIN ANTAGONIST; UNCLASSIFIED DRUG; X LINKED INHIBITOR OF APOPTOSIS;

APOPTOSIS; ARTICLE; CANCER CELL; CELL VIABILITY; DRUG DESIGN; DRUG SYNTHESIS; PROTEIN BINDING; PROTEIN DOMAIN; PROTEIN STRUCTURE;

BINDING SITES; BIOMIMETIC MATERIALS; CELL LINE, TUMOR; CELL SURVIVAL; DRUG DESIGN; DRUG RESISTANCE, NEOPLASM; HUMANS; MOLECULAR DOCKING SIMULATION; OLIGOPEPTIDES; PROTEIN BINDING; PROTEIN STRUCTURE, TERTIARY; STRUCTURE-ACTIVITY RELATIONSHIP; TNF-RELATED APOPTOSIS-INDUCING LIGAND; X-LINKED INHIBITOR OF APOPTOSIS PROTEIN;

EID: 84879411444 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2013.04.096 Document Type: Article

Times cited : (12)

References (24)

1
- 84894405292
- http://www.cancerresearchuk.org/cancer-info/cancerstats/world/ cancer-worldwide-the-global-picture.

2
- 0036176510
- M.M. Gottesman Annu. Rev. Med. 53 2002 615
- (2002) Annu. Rev. Med. , vol.53 , pp. 615
- Gottesman, M.M.¹

3
- 0034614637
- D. Hanahan, and R.A. Weinberg Cell 100 2000 57
- (2000) Cell , vol.100 , pp. 57
- Hanahan, D.¹ Weinberg, R.A.²

4
- 84856495152
- S. Fulda, and D. Vucic Nat. Rev. Drug Discov. 11 2012 109
- (2012) Nat. Rev. Drug Discov. , vol.11 , pp. 109
- Fulda, S.¹ Vucic, D.²

5
- 80054122612
- S. Condon Ann. Rep. Med. Chem. 46 2011 211
- (2011) Ann. Rep. Med. Chem. , vol.46 , pp. 211
- Condon, S.¹

6
- 69249100500
- C. Pop, and G.S. Salvesen J. Biol. Chem. 284 2009 21777
- (2009) J. Biol. Chem. , vol.284 , pp. 21777
- Pop, C.¹ Salvesen, G.S.²

7
- 30844457537
- A.D. Schimmer, S. Dalili, R.A. Batey, and S.J. Riedl Cell Death Differ. 13 2006 179
- (2006) Cell Death Differ. , vol.13 , pp. 179
- Schimmer, A.D.¹ Dalili, S.² Batey, R.A.³ Riedl, S.J.⁴

8
- 0035831019
- S.J. Riedl, M. Renatus, R. Schwarzenbacher, Q. Zhou, C. Sun, S.W. Fesik, R.C. Liddington, and G.S. Salvesen Cell 104 2001 791
- (2001) Cell , vol.104 , pp. 791
- Riedl, S.J.¹ Renatus, M.² Schwarzenbacher, R.³ Zhou, Q.⁴ Sun, C.⁵ Fesik, S.W.⁶ Liddington, R.C.⁷ Salvesen, G.S.⁸

9
- 4344691959
- E.N. Shiozaki, and Y. Shi Trends Biochem. Sci. 39 2004 486
- (2004) Trends Biochem. Sci. , vol.39 , pp. 486
- Shiozaki, E.N.¹ Shi, Y.²

10
- 57349147782
- H. Sun, Z. Nikolovska-Coleska, C.-Y. Yang, D. Qian, J. Lu, S. Qiu, L. Bai, Y. Peng, Q. Cai, and S. Wang Acc. Chem. Res. 41 2008 1264
- (2008) Acc. Chem. Res. , vol.41 , pp. 1264
- Sun, H.¹ Nikolovska-Coleska, Z.² Yang, C.-Y.³ Qian, D.⁴ Lu, J.⁵ Qiu, S.⁶ Bai, L.⁷ Peng, Y.⁸ Cai, Q.⁹ Wang, S.¹⁰

11
- 77649239222
- R. Mannhold, S. Fulda, and E. Carosati Drug Discov. Today 15 2010 210
- (2010) Drug Discov. Today , vol.15 , pp. 210
- Mannhold, R.¹ Fulda, S.² Carosati, E.³

12
- 76149118435
- J.A. Flygare, and W.J. Fairbrother Expert Opin. Ther. Pat. 20 2010 251
- (2010) Expert Opin. Ther. Pat. , vol.20 , pp. 251
- Flygare, J.A.¹ Fairbrother, W.J.²

13
- 84861034546
- J.A. Flygare, M. Beresini, N. Budha, H. Chan, I.T. Chan, S. Cheeti, F. Cohen, K. Deshayes, K. Doerner, S.G. Eckhardt, L.O. Elliott, B. Feng, M.C. Franklin, S.F. Reisner, L. Gazzard, J. Halladay, S.G. Hymowitz, H. La, P. LoRusso, B. Maurer, L. Murray, E. Plise, C. Quan, J.-P. Stephan, S.G. Young, J. Tom, V. Tsui, J. Um, E. Varfolomeev, D. Vucic, A.J. Wagner, H.J.A. Wallweber, L. Wang, J. Ware, Z. Wen, H. Wong, J.M. Wong, M. Wong, S. Wong, R. Yu, K. Zobel, and W.J. Fairbrother J. Med. Chem. 55 2012 4101
- (2012) J. Med. Chem. , vol.55 , pp. 4101
- Flygare, J.A.¹ Beresini, M.² Budha, N.³ Chan, H.⁴ Chan, I.T.⁵ Cheeti, S.⁶ Cohen, F.⁷ Deshayes, K.⁸ Doerner, K.⁹ Eckhardt, S.G.¹⁰ Elliott, L.O.¹¹ Feng, B.¹² Franklin, M.C.¹³ Reisner, S.F.¹⁴ Gazzard, L.¹⁵ Halladay, J.¹⁶ Hymowitz, S.G.¹⁷ La, H.¹⁸ Lorusso, P.¹⁹ Maurer, B.²⁰ more..

14
- 84872398313
- R.I. Erickson, J. Tarrant, G. Cain, S.C. Lewin-Koh, N. Dybdal, H. Wong, E. Blackwood, K. West, R. Steigerwalt, M. Mamounas, J.A. Flygare, K. Amemiya, D. Dambach, W.J. Fairbrother, and D. Diaz Toxicol. Sci. 131 2013 247
- (2013) Toxicol. Sci. , vol.131 , pp. 247
- Erickson, R.I.¹ Tarrant, J.² Cain, G.³ Lewin-Koh, S.C.⁴ Dybdal, N.⁵ Wong, H.⁶ Blackwood, E.⁷ West, K.⁸ Steigerwalt, R.⁹ Mamounas, M.¹⁰ Flygare, J.A.¹¹ Amemiya, K.¹² Dambach, D.¹³ Fairbrother, W.J.¹⁴ Diaz, D.¹⁵

15
- 79955876177
- H. Sun, L. Liu, J. Lu, L. Bai, X. Li, Z. Nikolovska-Coleska, D. McEachern, C.Y. Yang, S. Qiu, H. Yi, D. Sun, and S. Wang J. Med. Chem. 54 2011 3306
- (2011) J. Med. Chem. , vol.54 , pp. 3306
- Sun, H.¹ Liu, L.² Lu, J.³ Bai, L.⁴ Li, X.⁵ Nikolovska-Coleska, Z.⁶ McEachern, D.⁷ Yang, C.Y.⁸ Qiu, S.⁹ Yi, H.¹⁰ Sun, D.¹¹ Wang, S.¹²

16
- 77952099836
- H. Sun, L. Liu, J. Lu, S. Qiu, C.Y. Yang, H. Yi, and S. Wang Bioorg. Med. Chem. Lett. 20 2010 3043
- (2010) Bioorg. Med. Chem. Lett. , vol.20 , pp. 3043
- Sun, H.¹ Liu, L.² Lu, J.³ Qiu, S.⁴ Yang, C.Y.⁵ Yi, H.⁶ Wang, S.⁷

17
- 9144234685
- A.D. Schimmer, K. Welsh, C. Pinilla, Z. Wang, M. Krajewska, M.J. Bonneau, I.M. Pedersen, S. Kitada, F.L. Scott, B. Bailly-Maitre, G. Glinsky, D. Scudiero, E. Sausville, G. Salvesen, A. Nefzi, J.M. Ostresh, R.A. Houghten, and J.C. Reed Cancer Cell 5 2004 25
- (2004) Cancer Cell , vol.5 , pp. 25
- Schimmer, A.D.¹ Welsh, K.² Pinilla, C.³ Wang, Z.⁴ Krajewska, M.⁵ Bonneau, M.J.⁶ Pedersen, I.M.⁷ Kitada, S.⁸ Scott, F.L.⁹ Bailly-Maitre, B.¹⁰ Glinsky, G.¹¹ Scudiero, D.¹² Sausville, E.¹³ Salvesen, G.¹⁴ Nefzi, A.¹⁵ Ostresh, J.M.¹⁶ Houghten, R.A.¹⁷ Reed, J.C.¹⁸

18
- 79955813671
- M. Orzaez, A. Gortat, M. Sancho, R.J. Carbajo, A. Pineda-Lucena, Y. Palacios-Rodriguez, and E. Perez-Paya Apoptosis 16 2011 460
- (2011) Apoptosis , vol.16 , pp. 460
- Orzaez, M.¹ Gortat, A.² Sancho, M.³ Carbajo, R.J.⁴ Pineda-Lucena, A.⁵ Palacios-Rodriguez, Y.⁶ Perez-Paya, E.⁷

19
- 79959871720
- M. González-Lopez, K. Welsh, D. Finlay, R.J. Ardecky, S.R. Ganji, Y. Su, H. Yuan, P. Teriete, P.D. Mace, S.J. Riedl, K. Vuori, J.C. Reed, and N.D.P. Cosford Bioorg. Med. Chem. Lett. 21 2011 4332
- (2011) Bioorg. Med. Chem. Lett. , vol.21 , pp. 4332
- González-Lopez, M.¹ Welsh, K.² Finlay, D.³ Ardecky, R.J.⁴ Ganji, S.R.⁵ Su, Y.⁶ Yuan, H.⁷ Teriete, P.⁸ Mace, P.D.⁹ Riedl, S.J.¹⁰ Vuori, K.¹¹ Reed, J.C.¹² Cosford, N.D.P.¹³

20
- 7444262377
- Z. Nikolovska-Coleska, R. Wang, X. Fang, H. Pan, Y. Tomita, P. Li, P.P. Roller, K. Krajewski, N. Saito, J. Stuckey, and S. Wang Anal. Biochem. 332 2004 261
- (2004) Anal. Biochem. , vol.332 , pp. 261
- Nikolovska-Coleska, Z.¹ Wang, R.² Fang, X.³ Pan, H.⁴ Tomita, Y.⁵ Li, P.⁶ Roller, P.P.⁷ Krajewski, K.⁸ Saito, N.⁹ Stuckey, J.¹⁰ Wang, S.¹¹

21
- 84862610399
- K.F. Speer, C.L. Cosimini, and K.E. Splan Biopolymers 98 2012 122
- (2012) Biopolymers , vol.98 , pp. 122
- Speer, K.F.¹ Cosimini, C.L.² Splan, K.E.³

22
- 42149087042
- B.P. Eckelman, M. Drag, S.J. Snipas, and G.S. Salvesen Cell Death Differ. 15 2008 920
- (2008) Cell Death Differ. , vol.15 , pp. 920
- Eckelman, B.P.¹ Drag, M.² Snipas, S.J.³ Salvesen, G.S.⁴

23
- 84876803988
- Antagonists of IAP-family anti-apoptotic proteins - Probe 2
- National Center for Biotechnology Information (US); Bethesda, MD, 2010-2009
- Lopez, M.; Welsh, K.; Yuan, H.; Stonich, D.; Su, Y.; Garcia, X.; Cuddy, M.; Houghten, R.; Sergienko, E.; Reed, J. C.; Ardecky, R.; Reddy, S.; Finlay, D.; Vuori, K.; Dad, S.; Chung, T. D. Y.; Cosford, N. D. P. Antagonists of IAP-family anti-apoptotic proteins - Probe 2. In Probe Reports from the NIH Molecular Libraries Program [Internet]; National Center for Biotechnology Information (US); Bethesda, MD, 2010-2009.
- Probe Reports from the NIH Molecular Libraries Program [Internet]
- Lopez, M.¹ Welsh, K.² Yuan, H.³ Stonich, D.⁴ Su, Y.⁵ Garcia, X.⁶ Cuddy, M.⁷ Houghten, R.⁸ Sergienko, E.⁹ Reed, J.C.¹⁰ Ardecky, R.¹¹ Reddy, S.¹² Finlay, D.¹³ Vuori, K.¹⁴ Dad, S.¹⁵ Chung, T.D.Y.¹⁶ Cosford, N.D.P.¹⁷

24
- 84876525212
- M. Vamos, K. Welsh, D. Finlay, P. San Lee, P.D. Mace, S.J. Snipas, M.L. Gonzalez, S. Reddy Ganji, R.J. Ardecky, S.J. Riedl, G.S. Salvesen, K. Vuori, J.C. Reed, and N.D.P Cosford ACS Chem. Biol. 8 2013 725
- (2013) ACS Chem. Biol. , vol.8 , pp. 725
- Vamos, M.¹ Welsh, K.² Finlay, D.³ San Lee, P.⁴ Mace, P.D.⁵ Snipas, S.J.⁶ Gonzalez, M.L.⁷ Reddy Ganji, S.⁸ Ardecky, R.J.⁹ Riedl, S.J.¹⁰ Salvesen, G.S.¹¹ Vuori, K.¹² Reed, J.C.¹³ Cosford, D.P.¹⁴

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