Characterization of dequalinium as a XIAP antagonist that targets the BIR2 domain

Apoptosis

Volumn 16, Issue 5, 2011, Pages 460-467

  Orzáez, Mar ^a   Gortat, Anna ^a   Sancho, Mónica ^a   Carbajo, Rodrigo J ^a   Pineda Lucena, Antonio ^a   Palacios Rodríguez, Yadira ^a,b   Pérez Payá, Enrique ^a,b  

^a CENTRO DE INVESTIGACIÓN PRÍNCIPE FELIPE   (Spain)

^b INSTITUTO DE BIOMEDICINA DE VALENCIA   (Spain)

Author keywords

Anti tumour; Apoptosis; Dequalinium; IAP; Inhibitor; Screening; XIAP

Indexed keywords

CASPASE 3; CASPASE 9; DEQUALINIUM; X LINKED INHIBITOR OF APOPTOSIS;

ANTINEOPLASTIC ACTIVITY; ARTICLE; CELL DEATH; CONTROLLED STUDY; ENZYME ACTIVITY; HUMAN; HUMAN CELL; IN VITRO STUDY; PRIORITY JOURNAL; PROTEIN DOMAIN; PROTEIN PROTEIN INTERACTION;

APOPTOSIS; BINDING SITES; CASPASE 3; DEQUALINIUM; HELA CELLS; HUMANS; MAGNETIC RESONANCE SPECTROSCOPY; PROTEIN BINDING; PROTEIN STRUCTURE, TERTIARY; X-LINKED INHIBITOR OF APOPTOSIS PROTEIN;

INTRACISTERNAL A-PARTICLES;

EID: 79955813671     PISSN: 13608185     EISSN: 1573675X     Source Type: Journal    
DOI: 10.1007/s10495-011-0582-4     Document Type: Article

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