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ChemMedChem

Volumn 8, Issue 6, 2013, Pages 909-913

Selective Bisubstrate Inhibitors with Sub-nanomolar Affinity for Protein Kinase Pim-1

(7) Ekambaram, Ramesh a Enkvist, Erki a Vaasa, Angela a Kasari, Marje a Raidaru, Gerda a Knapp, Stefan b Uri, Asko a

a UNIVERSITY OF TARTU (Estonia)

b UNIVERSITY OF OXFORD (United Kingdom)

Author keywords

Bisubstrate inhibitors; Fluorescent probes; Pim 1; Protein kinases

Indexed keywords

PROTEIN KINASE PIM 1; PROTEIN KINASE PIM 2; PROTEIN SERINE THREONINE KINASE; UNCLASSIFIED DRUG;

APOPTOSIS; ARTICLE; BINDING SITE; CELL DIFFERENTIATION; CELL PROLIFERATION; CELL SURVIVAL; HEMATOLOGIC MALIGNANCY; HUMAN; HYDROGEN BOND; MOLONEY LEUKEMIA ONCOVIRUS; NONHODGKIN LYMPHOMA; PRIORITY JOURNAL; PROSTATE CANCER;

DOSE-RESPONSE RELATIONSHIP, DRUG; MOLECULAR STRUCTURE; NANOSTRUCTURES; PROTEIN KINASE INHIBITORS; PROTO-ONCOGENE PROTEINS C-PIM-1; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 84878346308 PISSN: 18607179 EISSN: 18607187 Source Type: Journal
DOI: 10.1002/cmdc.201300042 Document Type: Article

Times cited : (18)

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