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Bioorganic and Medicinal Chemistry Letters

Volumn 22, Issue 10, 2012, Pages 3425-3430

Conjugates of 5-isoquinolinesulfonylamides and oligo-d-arginine possess high affinity and selectivity towards Rho kinase (ROCK)

(9) Lavogina, Darja a Kalind, Katrin a Bredihhina, Jevgenia a Hurt, Madis a Vaasa, Angela a Kasari, Marje a Enkvist, Erki a Raidaru, Gerda a Uri, Asko a

a UNIVERSITY OF TARTU (Estonia)

Author keywords

ARC; Inhibitor; Isoquinoline; Luminescent probe; Protein kinase; Rho kinase (ROCK)

Indexed keywords

5 ISOQUINOLINESULFONYLAMIDE DERIVATIVE; ARC 3002; ARGININE DERIVATIVE; ISOQUINOLINE DERIVATIVE; OLIGO DEXTRO ARGININE DERIVATIVE; RHO KINASE; RHO KINASE INHIBITOR; UNCLASSIFIED DRUG;

ARTICLE; DRUG POTENCY; DRUG SELECTIVITY; DRUG STRUCTURE; DRUG SYNTHESIS; ENZYME INHIBITION; REACTION ANALYSIS; STRUCTURE ANALYSIS;

ARGININE; ISOQUINOLINES; RHO-ASSOCIATED KINASES; SULFONAMIDES;

EID: 84860462617 PISSN: 0960894X EISSN: 14643405 Source Type: Journal
DOI: 10.1016/j.bmcl.2012.03.101 Document Type: Article

Times cited : (14)

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