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Volumn 386, Issue 3, 2013, Pages 177-183

Pharmacological profile of β3-adrenoceptor agonists in clinical development for the treatment of overactive bladder syndrome

Author keywords

Bladder; Mirabegron; Ritobegron; Solabegron

Indexed keywords

BETA 1 ADRENERGIC RECEPTOR; BETA 2 ADRENERGIC RECEPTOR; BETA 3 ADRENERGIC RECEPTOR; KUC 7322; MIRABEGRON; RITOBEGRON; SOLABEGRON; UNCLASSIFIED DRUG;

EID: 84877917378     PISSN: 00281298     EISSN: 14321912     Source Type: Journal    
DOI: 10.1007/s00210-012-0824-1     Document Type: Review
Times cited : (72)

References (39)
  • 1
    • 84868556806 scopus 로고    scopus 로고
    • 3-adrenoceptor agonist, on the primary bladder afferent activity and bladder microcontractions in rats in comparison with those of oxybutynin
    • 3-adrenoceptor agonist, on the primary bladder afferent activity and bladder microcontractions in rats in comparison with those of oxybutynin. Eur Urol 62:1166-1173
    • (2012) Eur Urol , vol.62 , pp. 1166-1173
    • Aizawa, N.1    Homma, Y.2    Igawa, Y.3
  • 2
    • 47149118684 scopus 로고    scopus 로고
    • 3-adrenoceptor agonists on pharmacology, physiology and obesity drug discovery
    • 10.1007/s00210-008-0271-1 1:CAS:528:DC%2BD1cXosVCrsLY%3D
    • 3-adrenoceptor agonists on pharmacology, physiology and obesity drug discovery. Naunyn-Schmiedeberg's Arch Pharmacol 378:225-240
    • (2008) Naunyn-Schmiedeberg's Arch Pharmacol , vol.378 , pp. 225-240
    • Arch, J.R.S.1
  • 3
    • 33750891388 scopus 로고    scopus 로고
    • 3-adrenoceptor agonist (GW427353) on spontaneous activity and detrusor relaxation in human bladder
    • 17026593 10.1111/j.1464-410X.2006.06564.x 1:CAS:528: DC%2BD2sXktlarsw%3D%3D
    • 3-adrenoceptor agonist (GW427353) on spontaneous activity and detrusor relaxation in human bladder. BJU Int 98:1310-1314
    • (2006) BJU Int , vol.98 , pp. 1310-1314
    • Biers, S.M.1    Reynard, J.M.2    Brading, A.F.3
  • 4
    • 0026575399 scopus 로고
    • Spare receptors for β-adrenoceptor-mediated positive inotropic effects of catecholamines in the human heart
    • 1376792 10.1097/00005344-199202000-00011 1:STN:280:DyaK38zgtFSntw%3D%3D
    • Brown L, Deighton NM, Bals S, Söhlmann W, Zerkowski H-R, Michel MC, Brodde O-E (1992) Spare receptors for β-adrenoceptor-mediated positive inotropic effects of catecholamines in the human heart. J Cardiovasc Pharmacol 19:222-232
    • (1992) J Cardiovasc Pharmacol , vol.19 , pp. 222-232
    • Brown, L.1    Deighton, N.M.2    Bals, S.3    Söhlmann, W.4    Zerkowski, H.-R.5    Michel, M.C.6    Brodde, O.-E.7
  • 6
    • 84857032218 scopus 로고    scopus 로고
    • Local renin-angiotensin systems in the genitourinary tract
    • 10.1007/s00210-011-0706-y 1:CAS:528:DC%2BC38XkslCksg%3D%3D
    • Comiter C (2012) Local renin-angiotensin systems in the genitourinary tract. Naunyn-Schmiedeberg's Arch Pharmacol 385:13-26
    • (2012) Naunyn-Schmiedeberg's Arch Pharmacol , vol.385 , pp. 13-26
    • Comiter, C.1
  • 7
    • 77949417868 scopus 로고    scopus 로고
    • Ligand-directed signalling at β-adrenoceptors
    • 20132209 10.1111/j.1476-5381.2009.00602.x 1:CAS:528:DC%2BC3cXjs1ektrk%3D
    • Evans BA, Sato M, Sarwar M, Hutchinson DS, Summers RJ (2010) Ligand-directed signalling at β-adrenoceptors. Br J Pharmacol 159:1022-1038
    • (2010) Br J Pharmacol , vol.159 , pp. 1022-1038
    • Evans, B.A.1    Sato, M.2    Sarwar, M.3    Hutchinson, D.S.4    Summers, R.J.5
  • 16
    • 84864454054 scopus 로고    scopus 로고
    • Intravesical epinephrine preserves uroplakin II expression in urinary bladder from cyclophosphamide-induced rat cystitis
    • 1:CAS:528:DC%2BC38XhtVemu73E
    • Kyung YS, Park H, Lee G (2012) Intravesical epinephrine preserves uroplakin II expression in urinary bladder from cyclophosphamide-induced rat cystitis. Naunyn-Schmiedeberg's Arch Pharmacol 385:769-776
    • (2012) Naunyn-Schmiedeberg's Arch Pharmacol , vol.385 , pp. 769-776
    • Kyung, Y.S.1    Park, H.2    Lee, G.3
  • 19
    • 77955556872 scopus 로고    scopus 로고
    • 3-adrenoceptor mediates the inhibitory effects of β-adrenoceptor agonists via the urothelium in pig bladder dome
    • 20151470 10.1002/nau.20838 1:CAS:528:DC%2BC3cXht1Snur%2FF
    • 3-adrenoceptor mediates the inhibitory effects of β-adrenoceptor agonists via the urothelium in pig bladder dome. Neurourol Urodyn 29:1320-1325
    • (2010) Neurourol Urodyn , vol.29 , pp. 1320-1325
    • Masunaga, K.1    Chapple, C.R.2    McKay, N.G.3    Yoshida, M.4    Sellers, D.J.5
  • 20
    • 71249116156 scopus 로고    scopus 로고
    • Effect of pre-contraction on β-adrenoceptor-mediated relaxation of rat urinary bladder
    • 19449014 10.1007/s00345-009-0416-y 1:CAS:528:DC%2BD1MXhsVKgt7zF
    • Michel MC, Sand C (2009) Effect of pre-contraction on β-adrenoceptor-mediated relaxation of rat urinary bladder. World J Urol 27:711-715
    • (2009) World J Urol , vol.27 , pp. 711-715
    • Michel, M.C.1    Sand, C.2
  • 21
    • 32544437708 scopus 로고    scopus 로고
    • 2- and β-adrenoceptors in the urinary bladder, urethra and prostate
    • 16465187 10.1038/sj.bjp.0706619 1:CAS:528:DC%2BD28XhtFGqsLY%3D
    • 2- and β-adrenoceptors in the urinary bladder, urethra and prostate. Br J Pharmacol 147:S88-S119
    • (2006) Br J Pharmacol , vol.147
    • Michel, M.C.1    Vrydag, W.2
  • 22
    • 79956202487 scopus 로고    scopus 로고
    • β-Adrenoceptor agonist effects in experimental models of bladder dysfunction
    • 21510978 10.1016/j.pharmthera.2011.03.014 1:CAS:528:DC%2BC3MXmsVyltbo%3D
    • Michel MC, Ochodnicky P, Homma Y, Igawa Y (2011) β-Adrenoceptor agonist effects in experimental models of bladder dysfunction. Pharmacol Ther 131:40-49
    • (2011) Pharmacol Ther , vol.131 , pp. 40-49
    • Michel, M.C.1    Ochodnicky, P.2    Homma, Y.3    Igawa, Y.4
  • 25
    • 84865472825 scopus 로고    scopus 로고
    • Expression profiling of G-protein-coupled receptors in human urothelium and related cell lines
    • 22551294 10.1111/j.1464-410X.2012.011145.x 1:CAS:528:DC%2BC38Xht1CgtrnL
    • Ochodnicky P, Humphreys S, Eccles R, Poljakovic M, Wiklund P, Michel MC (2012) Expression profiling of G-protein-coupled receptors in human urothelium and related cell lines. BJU Int 110:e293-e300
    • (2012) BJU Int , vol.110
    • Ochodnicky, P.1    Humphreys, S.2    Eccles, R.3    Poljakovic, M.4    Wiklund, P.5    Michel, M.C.6
  • 27
    • 70349269052 scopus 로고    scopus 로고
    • A refocus on the bladder as the originator of storage lower urinary tract symptoms: A systematic review of the latest literature
    • 19683859 10.1016/j.eururo.2009.07.044
    • Roosen A, Chapple CR, Dmochowski RR, Fowler CJ, Gratzke C, Roehrborn CG, Stief CG, Andersson K-E (2009) A refocus on the bladder as the originator of storage lower urinary tract symptoms: a systematic review of the latest literature. Eur Urol 56:810-820
    • (2009) Eur Urol , vol.56 , pp. 810-820
    • Roosen, A.1    Chapple, C.R.2    Dmochowski, R.R.3    Fowler, C.J.4    Gratzke, C.5    Roehrborn, C.G.6    Stief, C.G.7    Andersson, K.-E.8
  • 28
    • 33746490589 scopus 로고    scopus 로고
    • 3-Adrenoceptors in the cardiovascular system: Putative roles in human pathologies
    • 16480771 10.1016/j.pharmthera.2005.12.002 1:CAS:528:DC%2BD28Xns1Sks7w%3D
    • 3-Adrenoceptors in the cardiovascular system: putative roles in human pathologies. Pharmacol Ther 111:652-673
    • (2006) Pharmacol Ther , vol.111 , pp. 652-673
    • Rozec, B.1    Gauthier, C.2
  • 29
    • 79954602236 scopus 로고    scopus 로고
    • Adrenergic control of cardiac gap junction function and expression
    • 10.1007/s00210-011-0603-4 1:CAS:528:DC%2BC3MXis1yjsrY%3D
    • Salameh A, Dhein S (2011) Adrenergic control of cardiac gap junction function and expression. Naunyn-Schmiedeberg's Arch Pharmacol 383:331-346
    • (2011) Naunyn-Schmiedeberg's Arch Pharmacol , vol.383 , pp. 331-346
    • Salameh, A.1    Dhein, S.2
  • 31
    • 84871875830 scopus 로고    scopus 로고
    • 3-adrenoceptor agonist mirabegron reduces carbachol-induced contractile activity in detrusor tissue from patients with bladder outflow obstruction with or without detrusor overactivity
    • doi: 10.1016/j.ejphar.2012.11.060
    • 3-adrenoceptor agonist mirabegron reduces carbachol-induced contractile activity in detrusor tissue from patients with bladder outflow obstruction with or without detrusor overactivity. Eur J Pharmacol doi: 10.1016/j.ejphar.2012.11.060
    • (2013) Eur J Pharmacol
    • Svalo, J.1    Nordling, J.2    Bouchelouche, K.3    Andersson, K.-E.4    Korstanje, C.5    Bouchelouche, P.6
  • 37
    • 83455210932 scopus 로고    scopus 로고
    • Muscarinic receptor subtypes and signalling involved in the attenuation of isoprenaline-induced rat urinary bladder relaxation
    • 10.1007/s00210-011-0689-8 1:CAS:528:DC%2BC3MXhsV2lsrbM
    • Witte LPW, de Haas N, Mammen M, Stangeland EL, Steinfeld T, Aiyar J, Michel MC (2011) Muscarinic receptor subtypes and signalling involved in the attenuation of isoprenaline-induced rat urinary bladder relaxation. Naunyn-Schmiedeberg's Arch Pharmacol 384:555-563
    • (2011) Naunyn-Schmiedeberg's Arch Pharmacol , vol.384 , pp. 555-563
    • Witte, L.P.W.1    De Haas, N.2    Mammen, M.3    Stangeland, E.L.4    Steinfeld, T.5    Aiyar, J.6    Michel, M.C.7
  • 39
    • 80054945654 scopus 로고    scopus 로고
    • In vivo bladder selectivity of imidafenacin, a novel antimuscarinic agent, assessed by using an effectiveness index for bladder capacity in rats
    • 10.1007/s00210-011-0675-1 1:CAS:528:DC%2BC3MXhtVegurrN
    • Yamazaki T, Muraki Y, Anraku T (2011) In vivo bladder selectivity of imidafenacin, a novel antimuscarinic agent, assessed by using an effectiveness index for bladder capacity in rats. Naunyn-Schmiedeberg's Arch Pharmacol 384:319-329
    • (2011) Naunyn-Schmiedeberg's Arch Pharmacol , vol.384 , pp. 319-329
    • Yamazaki, T.1    Muraki, Y.2    Anraku, T.3


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.