Lack of evidence that nebivolol is a β 3-adrenoceptor agonist

European Journal of Pharmacology

Volumn 654, Issue 1, 2011, Pages 86-91

  Frazier, Elfaridah P ^a   Michel Reher, Martina B ^a   Van Loenen, Pieter ^a   Sand, Carsten ^b   Schneider, Tim ^b   Peters, Stephan L M ^a   Michel, Martin C ^a  

^a UNIVERSITY OF AMSTERDAM   (Netherlands)

^b UNIVERSITY OF DUISBURG ESSEN   (Germany)

Author keywords

3 Adrenoceptor; Chinese hamster ovary cell; Nebivolol; Urinary bladder

Indexed keywords

1 (2 ETHYLPHENOXY) 3 (1,2,3,4 TETRAHYDRO 1 NAPHTHYLAMINO) 2 PROPANOL OXALATE; BETA 3 ADRENERGIC RECEPTOR; CYCLIC AMP; ISOPRENALINE; NEBIVOLOL; RADIOLIGAND;

ANIMAL CELL; ANIMAL TISSUE; ARTICLE; BINDING AFFINITY; BLADDER; CHO CELL; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG POTENCY; DRUG RECEPTOR BINDING; GENETIC TRANSFECTION; HUMAN; HUMAN TISSUE; MALE; NONHUMAN; PRIORITY JOURNAL; RAT; SMOOTH MUSCLE FIBER; SMOOTH MUSCLE RELAXATION; VASODILATATION;

ADRENERGIC BETA-1 RECEPTOR ANTAGONISTS; ANIMALS; BENZOPYRANS; CHO CELLS; CRICETINAE; CRICETULUS; CYCLIC AMP; DOSE-RESPONSE RELATIONSHIP, DRUG; ETHANOLAMINES; HUMANS; MALE; PROPANOLAMINES; RATS; RATS, WISTAR; RECEPTORS, ADRENERGIC, BETA-3; URINARY BLADDER;

EID: 78951471093     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.ejphar.2010.11.036     Document Type: Article

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