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Volumn 63, Issue , 2013, Pages 892-896

Optimizing the control of apoptosis by amide/triazole isosteric substitution in a constrained peptoid

(7) Corredor, Miriam a Bujons, Jordi a Orzáez, Mar b Sancho, Mónica b Pérez Payá, Enrique b,c Alfonso, Ignacio a Messeguer, Angel a

a INSTITUTE OF ADVANCED CHEMISTRY OF CATALONIA IQAC CSIC (Spain)

b CENTRO DE INVESTIGACIÓN PRÍNCIPE FELIPE (Spain)

c INSTITUTO DE BIOMEDICINA DE VALENCIA (Spain)

Author keywords

lactam; Apoptosis inhibitors; Click chemistry; Molecular docking; Triazole; Ugi 4CC

Indexed keywords

1,2,3 TRIAZOLE DERIVATIVE; AMIDE; BETA LACTAM; PEPTOID; TRIAZOLE;

APOPTOSIS; ARTICLE; BIOLOGICAL ACTIVITY; CYCLIZATION; DRUG SYNTHESIS; IN VITRO STUDY; ISOMER; MOLECULAR DOCKING;

AMIDES; APOPTOSIS; BINDING SITES; CYCLIZATION; HUMANS; MODELS, CHEMICAL; MODELS, MOLECULAR; MOLECULAR STRUCTURE; PEPTOIDS; PROTEIN BINDING; PROTEIN STRUCTURE, TERTIARY; TRIAZOLES;

EID: 84877050340 PISSN: 02235234 EISSN: 17683254 Source Type: Journal
DOI: 10.1016/j.ejmech.2013.03.004 Document Type: Article

Times cited : (18)

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