A derivative of the natural compound kakuol affects DNA relaxation of topoisomerase IB inhibiting the cleavage reaction

Archives of Biochemistry and Biophysics

Volumn 530, Issue 1, 2013, Pages 7-12

  Castelli, Silvia ^a   Vieira, Sara ^a   D'Annessa, Ilda ^a   Katkar, Prafulla ^a   Musso, Loana ^b   Dallavalle, Sabrina ^b   Desideri, Alessandro ^a  

^a UNIVERSITY OF ROME TOR VERGATA   (Italy)

^b UNIVERSITY OF MILAN   (Italy)

Author keywords

Catalytic inhibitor; Cleavage; Docking; Kakuol; Natural compound; Topoisomerase IB

Indexed keywords

DNA TOPOISOMERASE; DNA TOPOISOMERASE INHIBITOR; KAKUOL; KAKUOL DERIVATIVE; PLANT MEDICINAL PRODUCT; TOPOISOMERASE 1B; UNCLASSIFIED DRUG;

ARTICLE; ASARUM; ASARUM SIEBOLDII; CATALYSIS; DNA BINDING; DNA CLEAVAGE; DNA SYNTHESIS INHIBITION; DRUG BINDING; DRUG STRUCTURE; DRUG SYNTHESIS; ENZYME ACTIVE SITE; HUMAN; MOLECULAR DOCKING; NONHUMAN; PRIORITY JOURNAL; RHIZOME;

BASE SEQUENCE; BENZODIOXOLES; BIOLOGICAL AGENTS; CATALYTIC DOMAIN; DNA; DNA TOPOISOMERASES, TYPE I; HUMANS; MODELS, MOLECULAR; NUCLEIC ACID CONFORMATION; PROPIOPHENONES; TOPOISOMERASE I INHIBITORS;

ASARUM SIEBOLDII;

EID: 84872135865     PISSN: 00039861     EISSN: 10960384     Source Type: Journal    
DOI: 10.1016/j.abb.2012.12.013     Document Type: Article

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