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Volumn 13, Issue , 2012, Pages

Microneedle pretreatment enhances the percutaneous permeation of hydrophilic compounds with high melting points

Author keywords

In vitro permeation study; LogKow; Melting point; Microneedles; Non steroidal anti inflammatory drug; Physical penetration enhancement; Transdermal drug delivery

Indexed keywords

DICLOFENAC; IBUPROFEN; KETOPROFEN; METHYLENE BLUE; PARACETAMOL; NONSTEROID ANTIINFLAMMATORY AGENT;

EID: 84872035866     PISSN: 20506511     EISSN: None     Source Type: Journal    
DOI: 10.1186/2050-6511-13-5     Document Type: Article
Times cited : (46)

References (39)
  • 1
    • 0035859979 scopus 로고    scopus 로고
    • Skin, the final frontier 32
    • Hadgraft J. Skin, the final frontier 32. IntJPharm 2001, 224:1-18.
    • (2001) IntJPharm , vol.224 , pp. 1-18
    • Hadgraft, J.1
  • 4
    • 0029188379 scopus 로고
    • Transdermal iontophoresis: effect of penetration enhancer and iontophoresis on drug transport and surface characteristics of human epidermis
    • Singh J, Singh S. Transdermal iontophoresis: effect of penetration enhancer and iontophoresis on drug transport and surface characteristics of human epidermis. Curr Probl Dermatol 1995, 22:179-183.
    • (1995) Curr Probl Dermatol , vol.22 , pp. 179-183
    • Singh, J.1    Singh, S.2
  • 5
    • 0024841175 scopus 로고
    • Transdermal iontophoretic drug delivery: mechanistic analysis and application to polypeptide delivery
    • 10.1002/jps.2600780506, 2664125
    • Srinivasan V, Higuchi WI, Sims SM, Ghanem AH, Behl CR. Transdermal iontophoretic drug delivery: mechanistic analysis and application to polypeptide delivery. J Pharm Sci 1989, 78:370-375. 10.1002/jps.2600780506, 2664125.
    • (1989) J Pharm Sci , vol.78 , pp. 370-375
    • Srinivasan, V.1    Higuchi, W.I.2    Sims, S.M.3    Ghanem, A.H.4    Behl, C.R.5
  • 7
    • 0031852494 scopus 로고    scopus 로고
    • Microfabricated microneedles: A novel approach to transdermal drug delivery
    • 10.1021/js980042+, 9687334
    • Henry S, McAllister DV, Allen MG, Prausnitz MR. Microfabricated microneedles: A novel approach to transdermal drug delivery. J Pharm Sci 1998, 87:922-925. 10.1021/js980042+, 9687334.
    • (1998) J Pharm Sci , vol.87 , pp. 922-925
    • Henry, S.1    McAllister, D.V.2    Allen, M.G.3    Prausnitz, M.R.4
  • 10
    • 59349105168 scopus 로고    scopus 로고
    • Skin penetration enhancement by a microneedle device (Dermaroller) in vitro: dependency on needle size and applied formulation
    • 10.1016/j.ejps.2008.12.008, 19146954
    • Badran MM, Kuntsche J, Fahr A. Skin penetration enhancement by a microneedle device (Dermaroller) in vitro: dependency on needle size and applied formulation. Eur J Pharm Sci 2009, 36:511-523. 10.1016/j.ejps.2008.12.008, 19146954.
    • (2009) Eur J Pharm Sci , vol.36 , pp. 511-523
    • Badran, M.M.1    Kuntsche, J.2    Fahr, A.3
  • 11
    • 48749105332 scopus 로고    scopus 로고
    • Microneedle-based drug delivery: studies on delivery parameters and biocompatibility
    • 10.1007/s10544-008-9171-x, 18324474
    • Wu Y, Qiu Y, Zhang S, Qin G, Gao Y. Microneedle-based drug delivery: studies on delivery parameters and biocompatibility. Biomed Microdevices 2008, 10:601-610. 10.1007/s10544-008-9171-x, 18324474.
    • (2008) Biomed Microdevices , vol.10 , pp. 601-610
    • Wu, Y.1    Qiu, Y.2    Zhang, S.3    Qin, G.4    Gao, Y.5
  • 13
    • 33747748467 scopus 로고    scopus 로고
    • Feasibility of microneedles for percutaneous absorption of insulin
    • 10.1016/j.ejps.2006.05.011, 16828268
    • Ito Y, Hagiwara E, Saeki A, Sugioka N, Takada K. Feasibility of microneedles for percutaneous absorption of insulin. Eur J Pharm Sci 2006, 29:82-88. 10.1016/j.ejps.2006.05.011, 16828268.
    • (2006) Eur J Pharm Sci , vol.29 , pp. 82-88
    • Ito, Y.1    Hagiwara, E.2    Saeki, A.3    Sugioka, N.4    Takada, K.5
  • 14
    • 40049112272 scopus 로고    scopus 로고
    • Dissolving microneedles for transdermal drug delivery
    • 10.1016/j.biomaterials.2007.12.048, 2293299, 18261792
    • Lee JW, Park JH, Prausnitz MR. Dissolving microneedles for transdermal drug delivery. Biomaterials 2008, 29:2113-2124. 10.1016/j.biomaterials.2007.12.048, 2293299, 18261792.
    • (2008) Biomaterials , vol.29 , pp. 2113-2124
    • Lee, J.W.1    Park, J.H.2    Prausnitz, M.R.3
  • 16
    • 1542358759 scopus 로고    scopus 로고
    • Microneedles for transdermal drug delivery
    • 10.1016/j.addr.2003.10.023, 15019747
    • Prausnitz MR. Microneedles for transdermal drug delivery. Adv Drug Deliv Rev 2004, 56:581-587. 10.1016/j.addr.2003.10.023, 15019747.
    • (2004) Adv Drug Deliv Rev , vol.56 , pp. 581-587
    • Prausnitz, M.R.1
  • 17
    • 77952744825 scopus 로고    scopus 로고
    • Transdermal delivery of insulin using microneedle rollers in vivo
    • 10.1016/j.ijpharm.2010.03.041, 20347024
    • Zhou CP, Liu YL, Wang HL, Zhang PX, Zhang JL. Transdermal delivery of insulin using microneedle rollers in vivo. Int J Pharm 2010, 392:127-133. 10.1016/j.ijpharm.2010.03.041, 20347024.
    • (2010) Int J Pharm , vol.392 , pp. 127-133
    • Zhou, C.P.1    Liu, Y.L.2    Wang, H.L.3    Zhang, P.X.4    Zhang, J.L.5
  • 18
    • 0344270926 scopus 로고    scopus 로고
    • Microfabricated needles for transdermal delivery of macromolecules and nanoparticles: fabrication methods and transport studies
    • 10.1073/pnas.2331316100, 283494, 14623977
    • McAllister DV, Wang PM, Davis SP, Park JH, Canatella PJ, Allen MG, Prausnitz MR. Microfabricated needles for transdermal delivery of macromolecules and nanoparticles: fabrication methods and transport studies. Proc Natl Acad Sci U S A 2003, 100:13755-13760. 10.1073/pnas.2331316100, 283494, 14623977.
    • (2003) Proc Natl Acad Sci U S A , vol.100 , pp. 13755-13760
    • McAllister, D.V.1    Wang, P.M.2    Davis, S.P.3    Park, J.H.4    Canatella, P.J.5    Allen, M.G.6    Prausnitz, M.R.7
  • 19
    • 33846542514 scopus 로고    scopus 로고
    • Assembled microneedle arrays enhance the transport of compounds varying over a large range of molecular weight across human dermatomed skin
    • 10.1016/j.jconrel.2006.11.009, 17196697
    • Verbaan FJ, Bal SM, van den Berg DJ, Groenink WH, Verpoorten H, Luttge R, Bouwstra JA. Assembled microneedle arrays enhance the transport of compounds varying over a large range of molecular weight across human dermatomed skin. J Control Release 2007, 117:238-245. 10.1016/j.jconrel.2006.11.009, 17196697.
    • (2007) J Control Release , vol.117 , pp. 238-245
    • Verbaan, F.J.1    Bal, S.M.2    van den Berg, D.J.3    Groenink, W.H.4    Verpoorten, H.5    Luttge, R.6    Bouwstra, J.A.7
  • 20
  • 21
    • 0030347018 scopus 로고    scopus 로고
    • Histological and histochemical investigations on the structure of udder skin of cattle with special reference to changes during in vivo udder perfusion models
    • Ludewig T, Michel G, Gutte G. Histological and histochemical investigations on the structure of udder skin of cattle with special reference to changes during in vivo udder perfusion models. Dtsch Tierarztl Wochenschr 1996, 103:501-505.
    • (1996) Dtsch Tierarztl Wochenschr , vol.103 , pp. 501-505
    • Ludewig, T.1    Michel, G.2    Gutte, G.3
  • 22
    • 80052657580 scopus 로고    scopus 로고
    • The correlation between epidermal lipid composition and morphologic skin characteristics with percutaneous permeation: an interspecies comparison of substances with different lipophilicity
    • 10.1111/j.1365-2885.2010.01246.x, 21906081
    • Stahl J, Niedorf F, Kietzmann M. The correlation between epidermal lipid composition and morphologic skin characteristics with percutaneous permeation: an interspecies comparison of substances with different lipophilicity. J Vet Pharmacol Ther 2011, 34:502-507. 10.1111/j.1365-2885.2010.01246.x, 21906081.
    • (2011) J Vet Pharmacol Ther , vol.34 , pp. 502-507
    • Stahl, J.1    Niedorf, F.2    Kietzmann, M.3
  • 23
    • 45549105562 scopus 로고    scopus 로고
    • The automated, accurate and reproducible determination of steady-state permeation parameters from percutaneous permeation data
    • Niedorf F, Schmidt E, Kietzmann M. The automated, accurate and reproducible determination of steady-state permeation parameters from percutaneous permeation data. Altern Lab Anim 2008, 36:201-213.
    • (2008) Altern Lab Anim , vol.36 , pp. 201-213
    • Niedorf, F.1    Schmidt, E.2    Kietzmann, M.3
  • 25
    • 0036105150 scopus 로고    scopus 로고
    • Improved genetic immunization via micromechanical disruption of skin-barrier function and targeted epidermal delivery
    • 10.1038/nm0402-415, 11927950
    • Mikszta JA, Alarcon JB, Brittingham JM, Sutter DE, Pettis RJ, Harvey NG. Improved genetic immunization via micromechanical disruption of skin-barrier function and targeted epidermal delivery. Nat Med 2002, 8:415-419. 10.1038/nm0402-415, 11927950.
    • (2002) Nat Med , vol.8 , pp. 415-419
    • Mikszta, J.A.1    Alarcon, J.B.2    Brittingham, J.M.3    Sutter, D.E.4    Pettis, R.J.5    Harvey, N.G.6
  • 26
    • 77957019129 scopus 로고    scopus 로고
    • Effects of microneedle length, density, insertion time and multiple applications on human skin barrier function: assessments by transepidermal water loss
    • 10.1016/j.tiv.2010.08.012, 20732409
    • Gomaa YA, Morrow DI, Garland MJ, Donnelly RF, El-Khordagui LK, Meidan VM. Effects of microneedle length, density, insertion time and multiple applications on human skin barrier function: assessments by transepidermal water loss. Toxicol In Vitro 2010, 24:1971-1978. 10.1016/j.tiv.2010.08.012, 20732409.
    • (2010) Toxicol In Vitro , vol.24 , pp. 1971-1978
    • Gomaa, Y.A.1    Morrow, D.I.2    Garland, M.J.3    Donnelly, R.F.4    El-Khordagui, L.K.5    Meidan, V.M.6
  • 27
    • 70350215864 scopus 로고    scopus 로고
    • Microneedle arrays allow lower microbial penetration than hypodermic needles in vitro
    • 10.1007/s11095-009-9967-2, 2900181, 19756972
    • Donnelly RF, Singh TR, Tunney MM, Morrow DI, McCarron PA, O'Mahony C, Woolfson AD. Microneedle arrays allow lower microbial penetration than hypodermic needles in vitro. Pharm Res 2009, 26:2513-2522. 10.1007/s11095-009-9967-2, 2900181, 19756972.
    • (2009) Pharm Res , vol.26 , pp. 2513-2522
    • Donnelly, R.F.1    Singh, T.R.2    Tunney, M.M.3    Morrow, D.I.4    McCarron, P.A.5    O'Mahony, C.6    Woolfson, A.D.7
  • 28
    • 77957280275 scopus 로고    scopus 로고
    • A microneedle roller for transdermal drug delivery
    • 10.1016/j.ejpb.2010.07.001, 20624460
    • Park JH, Choi SO, Seo S, Choy YB, Prausnitz MR. A microneedle roller for transdermal drug delivery. Eur J Pharm Biopharm 2010, 76:282-289. 10.1016/j.ejpb.2010.07.001, 20624460.
    • (2010) Eur J Pharm Biopharm , vol.76 , pp. 282-289
    • Park, J.H.1    Choi, S.O.2    Seo, S.3    Choy, Y.B.4    Prausnitz, M.R.5
  • 29
    • 48149083798 scopus 로고    scopus 로고
    • Influence of the delivery systems using a microneedle array on the permeation of a hydrophilic molecule, calcein
    • 10.1016/j.ejpb.2008.02.009, 18411045
    • Oh JH, Park HH, Do KY, Han M, Hyun DH, Kim CG, Kim CH, Lee SS, Hwang SJ, Shin SC, Cho CW. Influence of the delivery systems using a microneedle array on the permeation of a hydrophilic molecule, calcein. Eur J Pharm Biopharm 2008, 69:1040-1045. 10.1016/j.ejpb.2008.02.009, 18411045.
    • (2008) Eur J Pharm Biopharm , vol.69 , pp. 1040-1045
    • Oh, J.H.1    Park, H.H.2    Do, K.Y.3    Han, M.4    Hyun, D.H.5    Kim, C.G.6    Kim, C.H.7    Lee, S.S.8    Hwang, S.J.9    Shin, S.C.10    Cho, C.W.11
  • 30
    • 33845740999 scopus 로고    scopus 로고
    • Ibuprofen Transport into and through Skin from Topical Formulations: In Vitro-In Vivo Comparison 1
    • Herkenne C, Naik A, Kalia YN, Hadgraft J, Guy RH. Ibuprofen Transport into and through Skin from Topical Formulations: In Vitro-In Vivo Comparison 1. J Invest Dermatol 2006, 127:135-142.
    • (2006) J Invest Dermatol , vol.127 , pp. 135-142
    • Herkenne, C.1    Naik, A.2    Kalia, Y.N.3    Hadgraft, J.4    Guy, R.H.5
  • 32
    • 9144227054 scopus 로고    scopus 로고
    • In vitro percutaneous penetration of five pesticides-effects of molecular weight and solubility characteristics 3
    • Nielsen JB, Nielsen F, Sorensen JA. In vitro percutaneous penetration of five pesticides-effects of molecular weight and solubility characteristics 3. AnnOccupHyg 2004, 48:697-705.
    • (2004) AnnOccupHyg , vol.48 , pp. 697-705
    • Nielsen, J.B.1    Nielsen, F.2    Sorensen, J.A.3
  • 33
    • 20944438241 scopus 로고    scopus 로고
    • Percutaneous penetration through slightly damaged skin
    • 10.1007/s00403-005-0555-y, 15834614
    • Nielsen JB. Percutaneous penetration through slightly damaged skin. Arch Dermatol Res 2005, 296:560-567. 10.1007/s00403-005-0555-y, 15834614.
    • (2005) Arch Dermatol Res , vol.296 , pp. 560-567
    • Nielsen, J.B.1
  • 34
    • 0032841637 scopus 로고    scopus 로고
    • Microfabricated microneedles: A novel approach to transdermal drug delivery
    • Henry S, McAllister DV, Allen MG, Prausnitz MR. Microfabricated microneedles: A novel approach to transdermal drug delivery. J Pharm Sci 1999, 88:948.
    • (1999) J Pharm Sci , vol.88 , pp. 948
    • Henry, S.1    McAllister, D.V.2    Allen, M.G.3    Prausnitz, M.R.4
  • 36
    • 80054093391 scopus 로고    scopus 로고
    • Dynamic in-situ eutectic formation for topical drug delivery
    • Fiala S, Brown MB, Jones SA. Dynamic in-situ eutectic formation for topical drug delivery. J Pharm Pharmacol 2011, 63:1428-1436.
    • (2011) J Pharm Pharmacol , vol.63 , pp. 1428-1436
    • Fiala, S.1    Brown, M.B.2    Jones, S.A.3
  • 37
    • 0035927202 scopus 로고    scopus 로고
    • Mechanistic study into the enhanced transdermal permeation of a model beta-blocker, propranolol, by fatty acids: a melting point depression effect
    • 10.1016/S0378-5173(01)00645-7, 11337176
    • Stott PW, Williams AC, Barry BW. Mechanistic study into the enhanced transdermal permeation of a model beta-blocker, propranolol, by fatty acids: a melting point depression effect. Int J Pharm 2001, 219:161-176. 10.1016/S0378-5173(01)00645-7, 11337176.
    • (2001) Int J Pharm , vol.219 , pp. 161-176
    • Stott, P.W.1    Williams, A.C.2    Barry, B.W.3
  • 38
    • 50449085359 scopus 로고    scopus 로고
    • In vivo assessment of safety of microneedle arrays in human skin
    • 10.1016/j.ejps.2008.06.016, 18657610
    • Bal SM, Caussin J, Pavel S, Bouwstra JA. In vivo assessment of safety of microneedle arrays in human skin. Eur J Pharm Sci 2008, 35:193-202. 10.1016/j.ejps.2008.06.016, 18657610.
    • (2008) Eur J Pharm Sci , vol.35 , pp. 193-202
    • Bal, S.M.1    Caussin, J.2    Pavel, S.3    Bouwstra, J.A.4
  • 39
    • 67649096926 scopus 로고    scopus 로고
    • Microporation applications for enhancing drug delivery
    • 10.1517/17425240902841935, 19348604
    • Banga AK. Microporation applications for enhancing drug delivery. Expert Opin Drug Deliv 2009, 6:343-354. 10.1517/17425240902841935, 19348604.
    • (2009) Expert Opin Drug Deliv , vol.6 , pp. 343-354
    • Banga, A.K.1


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.