메뉴 건너뛰기




Volumn 39, Issue 7, 2012, Pages 1049-1052

Re-evaluation of in vivo selectivity of [11C]SA4503 to σ1 receptors in the brain: Contributions of emopamil binding protein

Author keywords

1 receptor; 11C SA4503; Emopamil binding protein

Indexed keywords

1 [2 (3,4 DIMETHOXYPHENYL)ETHYL] 4 (3 PHENYLPROPYL)PIPERAZINE C 11; BINDING PROTEIN; CUTAMESINE; EMOPAMIL BINDING PROTEIN; HALOPERIDOL; IFENPRODIL; RADIOLIGAND; SIGMA 1 OPIATE RECEPTOR; TAMOXIFEN; TRIFLUOPERAZINE; TRIFLUPERIDOL; UNCLASSIFIED DRUG;

EID: 84866013619     PISSN: 09698051     EISSN: 18729614     Source Type: Journal    
DOI: 10.1016/j.nucmedbio.2012.03.002     Document Type: Article
Times cited : (13)

References (34)
  • 1
    • 74049130162 scopus 로고    scopus 로고
    • The role of sigma-1 receptors in the pathophysiology of neuropsychiatric diseases
    • Ishikawa M., Hashimoto K. The role of sigma-1 receptors in the pathophysiology of neuropsychiatric diseases. J Recept Ligand Channel Res 2010, 3:25-36.
    • (2010) J Recept Ligand Channel Res , vol.3 , pp. 25-36
    • Ishikawa, M.1    Hashimoto, K.2
  • 2
    • 35549006797 scopus 로고    scopus 로고
    • 2+ signaling and cell survival
    • 2+ signaling and cell survival. Cell 2007, 131:596-610.
    • (2007) Cell , vol.131 , pp. 596-610
    • Hayashi, T.1    Su, T.P.2
  • 4
    • 0030426263 scopus 로고    scopus 로고
    • Enhancement of acetylcholine release by SA4503, a novel sigma 1 receptor agonist, in the brain
    • Kobayashi T., Matsuno K., Nakata K., Mita S. Enhancement of acetylcholine release by SA4503, a novel sigma 1 receptor agonist, in the brain. J Pharmacol Exp Ther 1996, 279:106-113.
    • (1996) J Pharmacol Exp Ther , vol.279 , pp. 106-113
    • Kobayashi, T.1    Matsuno, K.2    Nakata, K.3    Mita, S.4
  • 7
    • 0030949390 scopus 로고    scopus 로고
    • The mysteries of sigma receptors: new family members reveal a role in cholesterol synthesis
    • Moebius F.F., Striessnig J., Glossmann H. The mysteries of sigma receptors: new family members reveal a role in cholesterol synthesis. Trends Pharmacol Sci 1997, 18:67-70.
    • (1997) Trends Pharmacol Sci , vol.18 , pp. 67-70
    • Moebius, F.F.1    Striessnig, J.2    Glossmann, H.3
  • 8
    • 0024281403 scopus 로고
    • Steroid binding at sigma receptors suggests a link between endocrine, nervous, and immune systems
    • Su T.P., London E.D., Jaffe J.H. Steroid binding at sigma receptors suggests a link between endocrine, nervous, and immune systems. Science 1988, 240:219-221.
    • (1988) Science , vol.240 , pp. 219-221
    • Su, T.P.1    London, E.D.2    Jaffe, J.H.3
  • 10
    • 9544223310 scopus 로고    scopus 로고
    • Emopamil-binding protein, a mammalian protein that binds a series of structurally diverse neuroprotective agents, exhibits δ8-δ7 sterol isomerase activity in yeast
    • Silve S., Dupuy P.H., Labit-Lebouteiller C., Kaghad M., Chalon P., Rahier A., et al. Emopamil-binding protein, a mammalian protein that binds a series of structurally diverse neuroprotective agents, exhibits δ8-δ7 sterol isomerase activity in yeast. J Biol Chem 1996, 271:22434-22440.
    • (1996) J Biol Chem , vol.271 , pp. 22434-22440
    • Silve, S.1    Dupuy, P.H.2    Labit-Lebouteiller, C.3    Kaghad, M.4    Chalon, P.5    Rahier, A.6
  • 12
    • 0030933902 scopus 로고    scopus 로고
    • 1-binding sites for sterol isomerization inhibitors: evidence for a pharmacological relationship with the yeast sterol δ8-δ7 isomerase
    • 1-binding sites for sterol isomerization inhibitors: evidence for a pharmacological relationship with the yeast sterol δ8-δ7 isomerase. Br J Phatmacol 1997, 121:1-6.
    • (1997) Br J Phatmacol , vol.121 , pp. 1-6
    • Moebius, F.F.1    Reiter, R.J.2    Hanner, M.3    Glossmann, H.4
  • 21
    • 33644785824 scopus 로고    scopus 로고
    • Synthesis and binding affinities of methylvesamicol analogs for the acetylcholine transporter and sigma receptor
    • Shiba K., Ogawa K., Ishiwata K., Yajima K., Mori H. Synthesis and binding affinities of methylvesamicol analogs for the acetylcholine transporter and sigma receptor. Bioorg Med Chem 2006, 14:2820-2826.
    • (2006) Bioorg Med Chem , vol.14 , pp. 2820-2826
    • Shiba, K.1    Ogawa, K.2    Ishiwata, K.3    Yajima, K.4    Mori, H.5
  • 23
    • 33645544409 scopus 로고    scopus 로고
    • Synthesis and in vitro evaluation of iodinated derivatives of piperazine as a new ligand for sigma receptor imaging by single photon emission computed tomography
    • Hirata M., Mori T., Soga S., Umeda T., Ohmomo Y. Synthesis and in vitro evaluation of iodinated derivatives of piperazine as a new ligand for sigma receptor imaging by single photon emission computed tomography. Chem Pharm Bull 2006, 54:470-475.
    • (2006) Chem Pharm Bull , vol.54 , pp. 470-475
    • Hirata, M.1    Mori, T.2    Soga, S.3    Umeda, T.4    Ohmomo, Y.5
  • 25
    • 0030843039 scopus 로고    scopus 로고
    • Synthesis, structure and quantitative structure-activity relationships of σ receptor ligands, 1-[2-(3,4-dimethoxyphenyl)ethyl]-4-(3-phenylpropyl)piperazines
    • Fujimura K., Matsumoto J., Niwa M., Kobayashi T., Kawashima Y., In Y., et al. Synthesis, structure and quantitative structure-activity relationships of σ receptor ligands, 1-[2-(3,4-dimethoxyphenyl)ethyl]-4-(3-phenylpropyl)piperazines. Bioorg Med Chem 1997, 5:1675-1683.
    • (1997) Bioorg Med Chem , vol.5 , pp. 1675-1683
    • Fujimura, K.1    Matsumoto, J.2    Niwa, M.3    Kobayashi, T.4    Kawashima, Y.5    In, Y.6
  • 30
    • 0001853507 scopus 로고
    • In vitro and in vivo steroid receptor assays in the design of estrogen radiopharmaceuticals
    • CRC Press, Boca Raton, FL, W.C. Eckelman (Ed.)
    • Katzenellenbogen J.A., Heiman D.F., Carlson K.E., Lloyd J.E. In vitro and in vivo steroid receptor assays in the design of estrogen radiopharmaceuticals. Receptor Binding Radiotracers 1982, Vol. 1:93-126. CRC Press, Boca Raton, FL. W.C. Eckelman (Ed.).
    • (1982) Receptor Binding Radiotracers , vol.1 , pp. 93-126
    • Katzenellenbogen, J.A.1    Heiman, D.F.2    Carlson, K.E.3    Lloyd, J.E.4
  • 31
    • 0001954284 scopus 로고
    • Radiolabeled adrenergic and muscarinic blockers for in vivo studies
    • CRC Press, Boca Raton, FL, W.C. Eckelman (Ed.)
    • Eckelman W.C. Radiolabeled adrenergic and muscarinic blockers for in vivo studies. Receptor Binding Radiotracers 1982, Vol. 1:69-92. CRC Press, Boca Raton, FL. W.C. Eckelman (Ed.).
    • (1982) Receptor Binding Radiotracers , vol.1 , pp. 69-92
    • Eckelman, W.C.1
  • 32
    • 0028353073 scopus 로고
    • The application of receptor theory to receptor-binding and enzyme-binding oncologic radiopharmaceuticals
    • Eckelman W.C. The application of receptor theory to receptor-binding and enzyme-binding oncologic radiopharmaceuticals. Nucl Med Biol 1994, 21:759-769.
    • (1994) Nucl Med Biol , vol.21 , pp. 759-769
    • Eckelman, W.C.1


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.