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Volumn 32, Issue 8, 2012, Pages 1546-1558

Measurement of 5-HT 1A receptor density and in-vivo binding parameters of 18Fmefway in the nonhuman primate

Author keywords

5 HT 1A; 18F mefway; B max; K D; multiple injection PET

Indexed keywords

MEFWAY FLUORINE F 18; RADIOPHARMACEUTICAL AGENT; SEROTONIN 1A RECEPTOR; UNCLASSIFIED DRUG;

EID: 84864535033     PISSN: 0271678X     EISSN: 15597016     Source Type: Journal    
DOI: 10.1038/jcbfm.2012.43     Document Type: Article
Times cited : (12)

References (46)
  • 1
    • 0018757980 scopus 로고
    • Serotonin and dopamine metabolites in brain regions and cerebrospinal fluid of primate species: Effects of ketamine and fluphenazine
    • Bacopoulos NG, Redmond DE, Roth RH (1979) Serotonin and dopamine metabolites in brain regions and cerebrospinal fluid of primate species: effects of ketamine and fluphenazine. J Neurochem 32:1215-8
    • (1979) J Neurochem , vol.32 , pp. 1215-1218
    • Bacopoulos, N.G.1    Redmond, D.E.2    Roth, R.H.3
  • 2
    • 0030610492 scopus 로고    scopus 로고
    • 3HWAY-100635 for 5-HT1A receptor autoradiography in human brain: A comparison with 3H8-OH-DPAT and demonstration of increased binding in the frontal cortex in schizophrenia
    • Burnet PWJ, Eastwood SL, Harrison PJ (1997) 3HWAY-100635 for 5-HT1A receptor autoradiography in human brain: a comparison with 3H8-OH-DPAT and demonstration of increased binding in the frontal cortex in schizophrenia. Neurochem Int 30:565-74
    • (1997) Neurochem Int , vol.30 , pp. 565-574
    • Burnet, P.W.J.1    Eastwood, S.L.2    Harrison, P.J.3
  • 3
    • 0033624542 scopus 로고    scopus 로고
    • PET evaluation of 18FFCWAY, an analog of the 5-HT1A receptor antagonist,WAY-100635
    • Carson RE, Lang L,Watabe H, Der MG, Adams HR, Jagoda E (2000) PET evaluation of 18FFCWAY, an analog of the 5-HT1A receptor antagonist,WAY-100635. Nucl Med Biol 27:493-7
    • (2000) Nucl Med Biol , vol.27 , pp. 493-497
    • Carson, R.E.1    Lang Lwatabe, H.2    Der, M.G.3    Adams, H.R.4    Jagoda, E.5
  • 4
    • 1542286816 scopus 로고    scopus 로고
    • Measuring the in vivo binding parameters of 18F-fallypride in monkeys using a PET multiple-injection protocol
    • Christian BT, Narayanan T, Shi B, Morris ED, Mantil J, Mukherjee J (2004) Measuring the in vivo binding parameters of 18F-fallypride in monkeys using a PET multiple-injection protocol. J Cereb Blood Flow Metab 24:309-22
    • (2004) J Cereb Blood Flow Metab , vol.24 , pp. 309-322
    • Christian, B.T.1    Narayanan, T.2    Shi, B.3    Morris, E.D.4    Mantil, J.5    Mukherjee, J.6
  • 6
    • 0036263314 scopus 로고    scopus 로고
    • Modeling 18FMPPF positron emission tomography kinetics for the determination of 5-hydroxytryptamine (1A) receptor concentration with multiinjection
    • Costes N, Merlet I, Zimmer L, Lavenne F, Cinotti L, Delforge J, Luxen A, Pujol J-F, Le Bars D (2002) Modeling 18FMPPF positron emission tomography kinetics for the determination of 5-hydroxytryptamine (1A) receptor concentration with multiinjection. J Cereb Blood Flow Metab 22:753-65
    • (2002) J Cereb Blood Flow Metab , vol.22 , pp. 753-765
    • Costes, N.1    Merlet, I.2    Zimmer, L.3    Lavenne, F.4    Cinotti, L.5    Delforge, J.6    Luxen, A.7    Pujol, J.-F.8    Le Bars, D.9
  • 10
    • 0025455847 scopus 로고
    • Identifiability analysis and parameter identification of an in vivo ligand-receptor model from PET data
    • Delforge J, Syrota A, Mazoyer BM (1990) Identifiability analysis and parameter identification of an in vivo ligand-receptor model from PET data. IEEE Trans Biomed Eng 37:653-61
    • (1990) IEEE Trans Biomed Eng , vol.37 , pp. 653-661
    • Delforge, J.1    Syrota, A.2    Mazoyer, B.M.3
  • 11
    • 0025936652 scopus 로고
    • Effects of in utero ethanol exposure on the developing serotonergic system
    • Druse MJ, Kuo A, Tajuddin N (1991) Effects of in utero ethanol exposure on the developing serotonergic system. Alcohol Clin Exp Res 15:678-84
    • (1991) Alcohol Clin Exp Res , vol.15 , pp. 678-684
    • Druse, M.J.1    Kuo, A.2    Tajuddin, N.3
  • 16
    • 2442642743 scopus 로고    scopus 로고
    • Positron emission tomography receptor assay with multiple ligand concentrations: An equilibrium approach
    • (Abelson JN, Simon MI, eds) New York: Academic Press
    • Holden JE, Doudet DJ (2004) Positron emission tomography receptor assay with multiple ligand concentrations: an equilibrium approach. In: Methods in enzymology (Abelson JN, Simon MI, eds), vol. 385. New York: Academic Press, 169-84
    • (2004) Methods in Enzymology , vol.385 , pp. 169-184
    • Holden, J.E.1    Doudet, D.J.2
  • 18
    • 0028988544 scopus 로고
    • Characterization of the binding of 3HWAY-100635, a novel 5-hydroxytryptamine1A receptor antagonist, to rat brain
    • Khawaja X, Evans N, Reilly Y, Ennis C, Minchin MCW (1995) Characterization of the binding of 3HWAY-100635, a novel 5-hydroxytryptamine1A receptor antagonist, to rat brain. J Neurochem 64:2716-26
    • (1995) J Neurochem , vol.64 , pp. 2716-2726
    • Khawaja, X.1    Evans, N.2    Reilly, Y.3    Ennis, C.4    Minchin, M.C.W.5
  • 19
    • 0022974030 scopus 로고
    • Distribution of serotonin-1A receptors in the monkey and the postmortem human hippocampal region. A quantitative autoradiographic study using the selective agonist 3H8-OH-DPAT
    • Köhler C, Radesäter A-C, Lang W, Chan-Palay V (1986) Distribution of serotonin-1A receptors in the monkey and the postmortem human hippocampal region. A quantitative autoradiographic study using the selective agonist 3H8-OH-DPAT. Neurosci Lett 72:43-8
    • (1986) Neurosci Lett , vol.72 , pp. 43-48
    • Köhler, C.1    Radesäter, A.-C.2    Lang, W.3    Chan-Palay, V.4
  • 20
  • 27
    • 27544446126 scopus 로고    scopus 로고
    • Multiinjection approach for D2 receptor binding quantification in living rats using 11Craclopride and the b-microprobe: Crossvalidation with in vitro binding data
    • Mauger G, Saba W, Hantraye P, Dolle F, Coulon C, Bramoulle Y, Chalon S, Grégoire M-C (2005) Multiinjection approach for D2 receptor binding quantification in living rats using 11Craclopride and the b-microprobe: crossvalidation with in vitro binding data. J Cereb Blood Flow Metab 25:1517-27
    • (2005) J Cereb Blood Flow Metab , vol.25 , pp. 1517-1527
    • Mauger, G.1    Saba, W.2    Hantraye, P.3    Dolle, F.4    Coulon, C.5    Bramoulle, Y.6    Chalon, S.7    Grégoire, M.-C.8
  • 30
    • 2442700315 scopus 로고    scopus 로고
    • Estimation of local receptor density, B'max, and other parameters via multiple-injection positron emission tomography experiments
    • (Abelson JN, Simon MI, eds) New York: Academic Press
    • Morris ED, Christian BT, Yoder KK, Muzic RF (2004) Estimation of local receptor density, B'max, and other parameters via multiple-injection positron emission tomography experiments. In: Methods in enzymology (Abelson JN, Simon MI, eds), vol. 385. New York: Academic Press, 184-213
    • (2004) Methods in Enzymology , vol.385 , pp. 184-213
    • Morris, E.D.1    Christian, B.T.2    Yoder, K.K.3    Muzic, R.F.4
  • 31
    • 31844443045 scopus 로고    scopus 로고
    • Evaluation of objective functions for estimation of kinetic parameters
    • Muzic RF, Christian BT (2006) Evaluation of objective functions for estimation of kinetic parameters. Med Phys 33:342-53
    • (2006) Med Phys , vol.33 , pp. 342-353
    • Muzic, R.F.1    Christian, B.T.2
  • 32
    • 0035047852 scopus 로고    scopus 로고
    • COMKAT: Compartment model kinetic analysis tool
    • Muzic RF, Cornelius S (2001) COMKAT: compartment model kinetic analysis tool. J Nucl Med 42:636-45
    • (2001) J Nucl Med , vol.42 , pp. 636-645
    • Muzic, R.F.1    Cornelius, S.2
  • 33
    • 0034318949 scopus 로고    scopus 로고
    • Iterative optimal design of PET experiments for estimating b-adrenergic receptor concentration
    • Muzic RF, Saidel GM, Zhu N, Nelson AD, Zheng L, Berridge MS (2000) Iterative optimal design of PET experiments for estimating b-adrenergic receptor concentration. Med Biol Eng 38:593-602
    • (2000) Med Biol Eng , vol.38 , pp. 593-602
    • Muzic, R.F.1    Saidel, G.M.2    Zhu, N.3    Nelson, A.D.4    Zheng, L.5    Berridge, M.S.6
  • 34
    • 2942622711 scopus 로고    scopus 로고
    • Differentiation of extrastriatal dopamine D2 receptor density and affinity in the human brain using PET
    • Olsson H, Halldin C, Farde L (2004) Differentiation of extrastriatal dopamine D2 receptor density and affinity in the human brain using PET. Neuroimage 22:794-803
    • (2004) Neuroimage , vol.22 , pp. 794-803
    • Olsson, H.1    Halldin, C.2    Farde, L.3
  • 38
    • 34547233630 scopus 로고    scopus 로고
    • Synthesis and biologic evaluation of a novel serotonin 5-HT1A receptor radioligand, 18F-labeled mefway, in rodents and imaging by PET in a nonhuman primate
    • Saigal N, Pichika R, Easwaramoorthy B, Collins D, Christian BT, Shi B, Narayanan TK, Potkin SG, Mukherjee J (2006) Synthesis and biologic evaluation of a novel serotonin 5-HT1A receptor radioligand, 18F-labeled mefway, in rodents and imaging by PET in a nonhuman primate. J Nucl Med 47:1697-706
    • (2006) J Nucl Med , vol.47 , pp. 1697-1706
    • Saigal, N.1    Pichika, R.2    Easwaramoorthy, B.3    Collins, D.4    Christian, B.T.5    Shi, B.6    Narayanan, T.K.7    Potkin, S.G.8    Mukherjee, J.9
  • 39
    • 33845919225 scopus 로고    scopus 로고
    • Robust experiment design for estimating myocardial beta adrenergic receptor concentration using PET
    • Salinas C, Muzic RF, Ernsberger P, Saidel GM (2007) Robust experiment design for estimating myocardial beta adrenergic receptor concentration using PET. Med Phys 34:151-65
    • (2007) Med Phys , vol.34 , pp. 151-165
    • Salinas, C.1    Muzic, R.F.2    Ernsberger, P.3    Saidel, G.M.4
  • 44
    • 0032793091 scopus 로고    scopus 로고
    • Analogues ofWAY-100635 as radiotracers for in vivo imaging of 5-HT1A receptors
    • Wilson AA, Garcia A, Li J, Dasilva JN, Houle S (1999) Analogues ofWAY-100635 as radiotracers for in vivo imaging of 5-HT1A receptors. J Labelled Compd Rad 42:611-20
    • (1999) J Labelled Compd Rad , vol.42 , pp. 611-620
    • Wilson, A.A.1    Garcia, A.2    Li, J.3    Dasilva, J.N.4    Houle, S.5


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.