SCOPUS 정보 검색 플랫폼

Volumn 85, Issue 8, 2012, Pages 1897-1911

Design, synthesis and biological activity evaluation of 2-mercapto-4(3H)-quinazolinone derivatives as novel inhibitors of protein tyrosine phosphatase 1B

(8) Li, Hui a Wang, Jin Ping a Yang, Fan a Liu, Ting a Qiu, Wen Wei a Li, Jing Ya b Li, Jia b Tang, Jie a

a EAST CHINA NORMAL UNIVERSITY (China)

b SHANGHAI INSTITUTE OF MATERIA MEDICA (China)

Author keywords

[No Author keywords available]

Indexed keywords

EID: 84864359321 PISSN: 03855414 EISSN: 18810942 Source Type: Journal
DOI: 10.3987/COM-12-12477 Document Type: Article

Times cited : (11)

References (44)

1
- 2942581416
- A. Alonso, J. Sasin, N. Bottini, I. Friedberg, A. Osterman, A. Godzik, T. Hunter, J. Dixon, and T. Mustelin, Cell, 2004, 117, 699.
- (2004) Cell , vol.117 , pp. 699
- Alonso, A.¹ Sasin, J.² Bottini, N.³ Friedberg, I.⁴ Osterman, A.⁵ Godzik, A.⁶ Hunter, T.⁷ Dixon, J.⁸ Mustelin, T.⁹

2
- 0036183603
- A. Cheng, N. Dubè, F. Gu, and M. L. Tremblay, Eur. J. Biochem., 2002, 269, 1050.
- (2002) Eur. J. Biochem , vol.269 , pp. 1050
- Cheng, A.¹ Dubè, N.² Gu, F.³ Tremblay, M.L.⁴

3
- 0035990925
- Z. Zhang, B. Zhou, and L. Xie, Pharmacol. Therap., 2002, 93, 307.
- (2002) Pharmacol. Therap , vol.93 , pp. 307
- Zhang, Z.¹ Zhou, B.² Xie, L.³

4
- 0035415662
- Z. Y. Zhang, Curr. Opin. Chem. Biol., 2001, 5, 416.
- (2001) Curr. Opin. Chem. Biol , vol.5 , pp. 416
- Zhang, Z.Y.¹

5
- 0036807325
- R. H. Van Huijsduijnen, A. Bombrun, and D. Swinnen, Drugs Discov. Today, 2002, 7, 1013.
- (2002) Drugs Discov. Today , vol.7 , pp. 1013
- Van Huijsduijnen, R.H.¹ Bombrun, A.² Swinnen, D.³

6
- 38949123683
- W. J. Hendriks, A. Elson, S. Harroch, and A. W. Stoker, FEBS J., 2008, 275, 816.
- (2008) FEBS J , vol.275 , pp. 816
- Hendriks, W.J.¹ Elson, A.² Harroch, S.³ Stoker, A.W.⁴

7
- 33847202286
- S. G. Julien, N. Dubé, M. Read, J. Penney, M. Paquet, Y. X. Han, B. P. Kennedy, W. J. Muller, and M. L. Tremblay, Nat. Genet., 2007, 39, 338.
- (2007) Nat. Genet , vol.39 , pp. 338
- Julien, S.G.¹ Dubé, N.² Read, M.³ Penney, J.⁴ Paquet, M.⁵ Han, Y.X.⁶ Kennedy, B.P.⁷ Muller, W.J.⁸ Tremblay, M.L.⁹

8
- 0039619868
- S. Wälchli, M. L. Curchod, R. P. Gobert, S. Arkinstall, and R. H. Van Huijsduijnen, J. Biol. Chem., 2000, 275, 9792.
- (2000) J. Biol. Chem , vol.275 , pp. 9792
- Wälchli, S.¹ Curchod, M.L.² Gobert, R.P.³ Arkinstall, S.⁴ Van Huijsduijnen, R.H.⁵

9
- 0034635374
- B. J. Goldstein, A. Bittner-Kowalczyk, M. F. White, and M. Harbeck, J. Biol. Chem., 2000, 275, 4283.
- (2000) J. Biol. Chem , vol.275 , pp. 4283
- Goldstein, B.J.¹ Bittner-Kowalczyk, A.² White, M.F.³ Harbeck, M.⁴

10
- 0036228770
- A. Cheng, N. Uetani, P. D. Simoncic, V. P. Chaubey, A. Lee-Loy, C. J. McGlade, B. P. Kennedy, and M. L. Tremblay, Dev. Cell, 2002, 2, 497.
- (2002) Dev. Cell , vol.2 , pp. 497
- Cheng, A.¹ Uetani, N.² Simoncic, P.D.³ Chaubey, V.P.⁴ Lee-Loy, A.⁵ McGlade, C.J.⁶ Kennedy, B.P.⁷ Tremblay, M.L.⁸

11
- 18344379861
- J. M. Zabolotny, K. K. Bence-Hanulec, A. Stricker-Krongrad, F. Haj, Y. Wang, Y. Minokoshi, Y. B. Kim, J. K. Elmquist, L. A. Tartaglia, B. B. Kahn, and B. G. Neel, Dev. Cell, 2002, 2, 489.
- (2002) Dev. Cell , vol.2 , pp. 489
- Zabolotny, J.M.¹ Bence-Hanulec, K.K.² Stricker-Krongrad, A.³ Haj, F.⁴ Wang, Y.⁵ Minokoshi, Y.⁶ Kim, Y.B.⁷ Elmquist, J.K.⁸ Tartaglia, L.A.⁹ Kahn, B.B.¹⁰ Neel, B.G.¹¹

12
- 0033525870
- M. Elchebly, P. Payette, E. Michaliszyn, W. Cromlish, S. Collins, A. L. Loy, D. Normandin, A. Cheng, J. Himms-Hagen, C. C. Chan, C. Ramachandran, M. J. Gresser, M. L. Tremblay, and B. P. Kennedy, Science, 1999, 283, 1544.
- (1999) Science , vol.283 , pp. 1544
- Elchebly, M.¹ Payette, P.² Michaliszyn, E.³ Cromlish, W.⁴ Collins, S.⁵ Loy, A.L.⁶ Normandin, D.⁷ Cheng, A.⁸ Himms-Hagen, J.⁹ Chan, C.C.¹⁰ Ramachandran, C.¹¹ Gresser, M.J.¹² Tremblay, M.L.¹³ Kennedy, B.P.¹⁴

13
- 0033942614
- L. D. Klaman, O. Boss, O. D. Peroni, J. K. Kim, J. L. Martino, J. M. Zabolotny, N. Moghal, M. Lubkin, Y. B. Kim, A. H. Sharpe, A. Stricker-Krongrad, G. I. Shulman, B. G. Neel, and B. B. Kahn, Mol. Cell. Biol., 2000, 20, 5479.
- (2000) Mol. Cell. Biol , vol.20 , pp. 5479
- Klaman, L.D.¹ Boss, O.² Peroni, O.D.³ Kim, J.K.⁴ Martino, J.L.⁵ Zabolotny, J.M.⁶ Moghal, N.⁷ Lubkin, M.⁸ Kim, Y.B.⁹ Sharpe, A.H.¹⁰ Stricker-Krongrad, A.¹¹ Shulman, G.I.¹² Neel, B.G.¹³ Kahn, B.B.¹⁴

14
- 79960073235
- D. Popov, Biochem. Biophys. Res. Commun., 2011, 410, 377.
- (2011) Biochem. Biophys. Res. Commun , vol.410 , pp. 377
- Popov, D.¹

15
- 0034308201
- B. P. Kennedy and C. Ramachandran, Biochem. Pharmacol., 2000, 60, 877.
- (2000) Biochem. Pharmacol , vol.60 , pp. 877
- Kennedy, B.P.¹ Ramachandran, C.²

16
- 0036715628
- T. O. Johnson, J. Ermolieff, and M. R. Jirousek, Nat. Rev. Drug Discov., 2002, 1, 696.
- (2002) Nat. Rev. Drug Discov , vol.1 , pp. 696
- Johnson, T.O.¹ Ermolieff, J.² Jirousek, M.R.³

17
- 34247362854
- S. Zhang and Z. Y. Zhang, Drug Discov. Today, 2007, 12, 373.
- (2007) Drug Discov. Today , vol.12 , pp. 373
- Zhang, S.¹ Zhang, Z.Y.²

18
- 34347260715
- S. Lee and Q. Wang, Med. Res. Rev., 2007, 27, 553.
- (2007) Med. Res. Rev , vol.27 , pp. 553
- Lee, S.¹ Wang, Q.²

19
- 38749150385
- L. Shi, H. P. Yu, Y. Y. Zhou, J. Q. Du, Q. Shen, J. Y. Li, and J. Li, Acta Pharmacol. Sin., 2008, 29, 278.
- (2008) Acta Pharmacol. Sin , vol.29 , pp. 278
- Shi, L.¹ Yu, H.P.² Zhou, Y.Y.³ Du, J.Q.⁴ Shen, Q.⁵ Li, J.Y.⁶ Li, J.⁷

20
- 64849096634
- Y. Zhang, Y. Li, Y. W. Guo, H. L. Jiang, and X. Shen, Acta Pharmacol. Sin., 2009, 30, 333.
- (2009) Acta Pharmacol. Sin , vol.30 , pp. 333
- Zhang, Y.¹ Li, Y.² Guo, Y.W.³ Jiang, H.L.⁴ Shen, X.⁵

21
- 77955461653
- Z. Liu, Q. Chai, Y. Y. Li, Q. Shen, L. P. Ma, L. N. Zhang, X. Wang, L. Sheng, J. Y. Li, J. Li, and J. K. Shen, Acta Pharmacol. Sin., 2010, 31, 1005.
- (2010) Acta Pharmacol. Sin , vol.31 , pp. 1005
- Liu, Z.¹ Chai, Q.² Li, Y.Y.³ Shen, Q.⁴ Ma, L.P.⁵ Zhang, L.N.⁶ Wang, X.⁷ Sheng, L.⁸ Li, J.Y.⁹ Li, J.¹⁰ Shen, J.K.¹¹

22
- 12344318177
- M. J. Hartshorn, C. W. Murray, A. Cleasby, M. Frederickson, I. J. Tickle, and H. Jhoti, J. Med. Chem., 2005, 48, 403.
- (2005) J. Med. Chem , vol.48 , pp. 403
- Hartshorn, M.J.¹ Murray, C.W.² Cleasby, A.³ Frederickson, M.⁴ Tickle, I.J.⁵ Jhoti, H.⁶

23
- 34648833338
- D. P. Wilson, Z. K. Wan, W. X. Xu, S. J. Kirincich, B. C. Follows, D. Joseph-McCarthy, K. Foreman, A. Moretto, J. J. Wu, M. Zhu, E. Binnun, Y. L. Zhang, M. Tam, D. V. Erbe, J. Tobin, X. Xu, L. Leung, A. Shilling, S. Y. Tam, T. S. Mansour, and J. Lee, J. Med. Chem., 2007, 50, 4681.
- (2007) J. Med. Chem , vol.50 , pp. 4681
- Wilson, D.P.¹ Wan, Z.K.² Xu, W.X.³ Kirincich, S.J.⁴ Follows, B.C.⁵ Joseph-Mccarthy, D.⁶ Foreman, K.⁷ Moretto, A.⁸ Wu, J.J.⁹ Zhu, M.¹⁰ Binnun, E.¹¹ Zhang, Y.L.¹² Tam, M.¹³ Erbe, D.V.¹⁴ Tobin, J.¹⁵ Xu, X.¹⁶ Leung, L.¹⁷ Shilling, A.¹⁸ Tam, S.Y.¹⁹ Mansour, T.S.²⁰ Lee, J.²¹ more..

24
- 47349122949
- M. Hussain, V. Ahmed, B. Hill, Z. Ahmed, and S. D. Taylor, Bioorg. Med. Chem., 2008, 16, 6764.
- (2008) Bioorg. Med. Chem , vol.16 , pp. 6764
- Hussain, M.¹ Ahmed, V.² Hill, B.³ Ahmed, Z.⁴ Taylor, S.D.⁵

25
- 0020637625
- P. Kumar, K. N. Dhawan, S. Vrat, K. P. Bhargava, and K. Kishore, Arch. Pharm., 1983, 316, 759.
- (1983) Arch. Pharm , vol.316 , pp. 759
- Kumar, P.¹ Dhawan, K.N.² Vrat, S.³ Bhargava, K.P.⁴ Kishore, K.⁵

26
- 0021271988
- N. S. Habib and M. A. Khalils, J. Pharm. Sci., 1984, 73, 982.
- (1984) J. Pharm. Sci , vol.73 , pp. 982
- Habib, N.S.¹ Khalils, M.A.²

27
- 50949089653
- V. Jatav, P. Mishra, S. Kashaw, and J. P. Stables, Eur. J. Med. Chem., 2008, 43, 1945.
- (2008) Eur. J. Med. Chem , vol.43 , pp. 1945
- Jatav, V.¹ Mishra, P.² Kashaw, S.³ Stables, J.P.⁴

28
- 0013817762
- S. Hayao, H. J. Havera, W. G. Strycker, T. J. Leipzig, R. A. Kulp, and H. E. Hartzler, J. Med. Chem., 1965, 8, 807.29. J. A.
- (1965) J. Med. Chem , vol.8 , pp. 807
- Hayao, S.¹ Havera, H.J.² Strycker, W.G.³ Leipzig, T.J.⁴ Kulp, R.A.⁵ Hartzler, H.E.⁶

29
- 0026073884
- J.A. 3rd. Lowe, R. L. Archer, D. S. Chapin, J. B. Cheng, D. Helweg, J. L. Johnson, B. K. Koe, L. A. Lebel, and P. F. Moore, J. Med. Chem., 1991, 34, 624.
- (1991) J. Med. Chem , vol.34 , pp. 624
- Lowe III, J.A.¹ Archer, R.L.² Chapin, D.S.³ Cheng, J.B.⁴ Helweg, D.⁵ Johnson, J.L.⁶ Koe, B.K.⁷ Lebel, L.A.⁸ Moore, P.F.⁹

30
- 0033598323
- C. Qi, L. Deng, H. Shih, L. M. Leoni, D. Genini, D. A. Carson, and H. B. Cottam, J. Med. Chem., 1999, 42, 3860.
- (1999) J. Med. Chem , vol.42 , pp. 3860
- Qi, C.¹ Deng, L.² Shih, H.³ Leoni, L.M.⁴ Genini, D.⁵ Carson, D.A.⁶ Cottam, H.B.⁷

31
- 17444372597
- B. R. Baker, R. E. Schaub, J. P. Joseph, F. J. McEvoy, and J. H. Williams, J. Org. Chem., 1952, 17, 149.
- (1952) J. Org. Chem , vol.17 , pp. 149
- Baker, B.R.¹ Schaub, R.E.² Joseph, J.P.³ McEvoy, F.J.⁴ Williams, J.H.⁵

32
- 8444233942
- A. R. Maarouf, E. R. El-Bendary, and F. E. Goda, Arch. Pharm. Pharm. Med. Chem., 2004, 337, 527.
- (2004) Arch. Pharm. Pharm. Med. Chem , vol.337 , pp. 527
- Maarouf, A.R.¹ El-Bendary, E.R.² Goda, F.E.³

33
- 56249112648
- T. Nagase, T. Mizutani, E. Sekino, S. Ishikawa, S. Ito, Y. Mitobe, Y. Miyamoto, R. Yoshimoto, T. Tanaka, A. Ishihara, N. Takenaga, S. Tokita, and N. Sato, J. Med. Chem., 2008, 51, 6889.
- (2008) J. Med. Chem , vol.51 , pp. 6889
- Nagase, T.¹ Mizutani, T.² Sekino, E.³ Ishikawa, S.⁴ Ito, S.⁵ Mitobe, Y.⁶ Miyamoto, Y.⁷ Yoshimoto, R.⁸ Tanaka, T.⁹ Ishihara, A.¹⁰ Takenaga, N.¹¹ Tokita, S.¹² Sato, N.¹³

34
- 0026718844
- M. J. Yu, J. R. McCowan, N. R. Mason, J. B. Deeter, and L. G. Mendelsohn, J. Med. Chem., 1992, 35, 2534.
- (1992) J. Med. Chem , vol.35 , pp. 2534
- Yu, M.J.¹ McCowan, J.R.² Mason, N.R.³ Deeter, J.B.⁴ Mendelsohn, L.G.⁵

35
- 14444274329
- J. K. Padia, M. Field, J. Hinton, K. Meecham, J. Pablo, R. Pinnock, B. D. Roth, L. Singh, N. Suman-Chauhan, B. K. Trivedi, and L. Webdale, J. Med. Chem., 1998, 41, 1042.
- (1998) J. Med. Chem , vol.41 , pp. 1042
- Padia, J.K.¹ Field, M.² Hinton, J.³ Meecham, K.⁴ Pablo, J.⁵ Pinnock, R.⁶ Roth, B.D.⁷ Singh, L.⁸ Suman-Chauhan, N.⁹ Trivedi, B.K.¹⁰ Webdale, L.¹¹

36
- 0030064335
- K. Smith, G. A. El-Hiti, M. F. Abdel-Megeed, and M. A. Abdo, J. Org. Chem., 1996, 61, 647.
- (1996) J. Org. Chem , vol.61 , pp. 647
- Smith, K.¹ El-Hiti, G.A.² Abdel-Megeed, M.F.³ Abdo, M.A.⁴

37
- 40749097325
- V. Alagarsamy, D. Shankar, and S. Murugesan, Biomed. Pharmacother., 2008, 62, 173.
- (2008) Biomed. Pharmacother , vol.62 , pp. 173
- Alagarsamy, V.¹ Shankar, D.² Murugesan, S.³

38
- 33750949952
- V. Alagarsamy, V. R. Solomon, and K. Dhanaba, Bioorg. Med. Chem., 2007, 15, 235.
- (2007) Bioorg. Med. Chem , vol.15 , pp. 235
- Alagarsamy, V.¹ Solomon, V.R.² Dhanaba, K.³

39
- 9344269616
- L. M. Yun, S. Yangibaev, K. M. Shakhidoyatov, V. Ya. Alekseeva, and K. A. V'yunov, Chem. Heterocycl. Comp., 1987, 23, 214.
- (1987) Chem. Heterocycl. Comp , vol.23 , pp. 214
- Yun, L.M.¹ Yangibaev, S.² Shakhidoyatov, K.M.³ Ya. Alekseeva, V.⁴ V'Yunov, K.A.⁵

40
- 0037194618
- Y. T. Chen and C. T. Seto, J. Med. Chem., 2002, 45, 3946.
- (2002) J. Med. Chem , vol.45 , pp. 3946
- Chen, Y.T.¹ Seto, C.T.²

41
- 0037140871
- F. R. Alexandre, A. Berecibara, and T. Besson, Tetrahedron Lett., 2002, 43, 3911.
- (2002) Tetrahedron Lett , vol.43 , pp. 3911
- Alexandre, F.R.¹ Berecibara, A.² Besson, T.³

42
- 0018397695
- R. M. Shafik, A. A. B. Hazzaa, and N. S. Habib, Pharmazie, 1979, 34, 148.
- (1979) Pharmazie , vol.34 , pp. 148
- Shafik, R.M.¹ Hazzaa, A.A.B.² Habib, N.S.³

43
- 9344269616
- L. M. Yun, S. Yangibaev, Kh. M. Shakhidoyatov, V. Ya. Alekseeva, and K. A. V'yunov, Chem. Heterocycl. Comp., 1987, 23, 214.
- (1987) Chem. Heterocycl. Comp , vol.23 , pp. 214
- Yun, L.M.¹ Yangibaev, S.² Shakhidoyatov, K.M.³ Ya. Alekseeva, V.⁴ V'Yunov, K.A.⁵

44
- 33645188851
- J. E. McCarty, E. L. Haines, and C. A. VanderWerf, J. Am. Chem. Soc., 1960, 82, 964.
- (1960) J. Am. Chem. Soc , vol.82 , pp. 964
- McCarty, J.E.¹ Haines, E.L.² Vanderwerf, C.A.³

* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.