Synthesis and evaluation of some novel quinazolinone derivatives as diuretic agents

Archiv der Pharmazie

Volumn 337, Issue 10, 2004, Pages 527-532

  Maarouf, Azza R ^a   El Bendary, Eman R ^a   Goda, Fatma E ^a  

^a MANSOURA UNIVERSITY   (Egypt)

Author keywords

4(3H) Quinazolinones; Diuretic activity; Thiadiazolylquinazolinones; Thiazolylquinazolinones

Indexed keywords

2 [2 (4 CHLOROPHENYL)VINYL] 7 CHLORO 3 (2 SULFAMOYL 1,3,4 THIADIAZOL 5 YL)QUINAZOLIN 4(3H) ONE; 4(3H) QUINAZOLINONE DERIVATIVE; 7 CHLORO 2 METHYL 3 (1,3,4 THIADIAZOL 2 YL)QUINAZOLIN 4(3H) ONE; 7 CHLORO 2 METHYL 3 (1,3,4 THIAZOL 2 YL)QUINAZOLIN 4(3H) ONE; 7 CHLORO 2 METHYL 3 (2 SULFAMOYL 1,3,4 THIADIAZOL 5 YL)QUINAZOLIN 4(3H) ONE; 7 CHLORO 3 (2 MERCAPTO 1,3,4 THIADIAZOL 5 YL) 2 METHYLQUINAZOLIN 4(3H) ONE; DIURETIC AGENT; FUROSEMIDE; QUINAZOLINONE DERIVATIVE; THIADIAZOLYLQUINAZOLINONE; THIAZOLYLQUINAZOLINONE; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ARTICLE; CONTROLLED STUDY; DIURETIC THERAPY; DRUG STRUCTURE; DRUG SYNTHESIS; FEMALE; MALE; NONHUMAN; PRIORITY JOURNAL; PROTON NUCLEAR MAGNETIC RESONANCE; RAT; SPECTROPHOTOMETRY;

ANIMALS; DIURETICS; LETHAL DOSE 50; QUINAZOLINES; RATS; STRUCTURE-ACTIVITY RELATIONSHIP; THIADIAZOLES; THIAZOLES;

EID: 8444233942     PISSN: 03656233     EISSN: None     Source Type: Journal    
DOI: 10.1002/ardp.200400869     Document Type: Article

References (31)

1. H. A. Parish Jr., R. D. Gilliom, W. P. Purcell, R. K. Browne, R. F. Spirk, H. D. White, J. Med. Chem. 1982, 25, 93-102.
2. S. Jantova, D. Hudecova, K. Spirkova, S. Stankovsky, Folia Microbiol. 1994, 39(6), 471-474.
3. J. Bartroli, E. Turmo, M. Alguerd, E. Boncompte, M. L. Vericat, L. Conte, J. Ramis, M. Merlos, J. G. Rafanell, J. Form, J. Med. Chem. 1998, 41(11), 1869-1882.
4. M. Shrimali, R. Kalsi, K. Dixit, J. P. Barthwal, Arzneimittel-Forschung 1991, 41, 514-519.
5. M. Y. Ebeid, H. H. Hassanein, M. V. Riad, A. B. Hassan, Egypt. J. Pharm. Sci. 1990, 31 (1-4), 267; M. Y. Ebeid, Z. I. Gad, N. M. El-Sayed, El-S. Ahmed, B. El-Sayeh, Egypt. J. Pharm. Sci. 1991, 32(3-4), 441-455.
6. M. Y. Ebeid, H. H. Hassanein, M. V. Riad, A. B. Hassan, Egypt. J. Pharm. Sci. 1990, 31 (1-4), 267; M. Y. Ebeid, Z. I. Gad, N. M. El-Sayed, El-S. Ahmed, B. El-Sayeh, Egypt. J. Pharm. Sci. 1991, 32(3-4), 441-455.
7. E. R. El-Bendary, M. A. El-Sherbeny, F. A. Badria, Boll. Chim. Farm. 1998, 137(4), 115-119.
8. M. A. El-Sherbeny, Arch. Pharm. Pharm. Med. Chem. 2000, 333, 323-328.
9. H. M. Eisa, M. B. El-Ashmawy, M. M. Tayel, S. A. Abo El-Magd, H. A. El-Kashef, Boll. Chim. Farm. 1996, 135(10), 585-590.
10. A. Monge, V. Martinez-Merino, V. Sanmartin, M. C. Ochoa, F. Fernadez-Alvarez, Arzneim-Forsch. 1990, 40, 1349-1352.
11. M. M. Gineinah, M. A. El-Sherbeny, M. N. Nasr, A. R. Maarouf, Arch. Pharm. Pharm. Med. Chem., 2002, 335, 556-562.
12. M. M. Gineinah, M. N. Nasr, A. M. Abdelal, A. A. El-Emam, S. A. Said, Med. Chem. Res. 2000, 10, 243-252.
13. S. El-Meligie, A. K. El-Ansary, M. M. Said, M. M. M. Hussein, Indian J. Chem. 2001, 40B, 62-69.
14. J. V. Partin, I. E. Anglin, N. Kyprianou, Br. J. Cancer. 2003, 88(10), 1615-1621.
15. D. R. Huron, M. E. Gorre, A. J. Kraker, C. L. Sawyers, N. Rosen, M. M. Moasser, Clin. Cancer Res. 2003, 9(4), 1267-1273.
16. A. M. Farghaly, R. Soliman, M. A. Khalil, A. A. Bekhit, A. el-Din, A. Bekhit, Boll. Chem. Farm. 2002, 141(5), 372-378.
17. C. Parkanyi, D. S. Schmidt, J. Heterocycl. Chem. 2000, 37, 725-729.
18. H. Kikuchi, H. Tasaka, S. Hirai, Y. Takaya, Y. Iwabuchi, H. Ooi, S. Hatakeyama, H. S. Kim, Y. Wataya, Y. Oshima, J. Med. Chem. 2002, 45(12), 2563-2570.
19. E. Cohen, B. Klarberg, J. R. Vaughan Jr., J. Am. Chem. Soc. 1959, 81, 5508-5509; E. Cohen, B. Klarberg, J. R. Vaughan Jr., J. Am. Chem. Soc. 1960, 82, 2731-2735.
20. E. Cohen, B. Klarberg, J. R. Vaughan Jr., J. Am. Chem. Soc. 1959, 81, 5508-5509; E. Cohen, B. Klarberg, J. R. Vaughan Jr., J. Am. Chem. Soc. 1960, 82, 2731-2735.
21. th Edition (Eds.: J. N. Delgado, W. A. Remers), Lippincott Raven, Philadelphia, 1998, chapter 2, 3-42.
22. B. J. Materson, J. L. Hotchkiss, J. S. Barkin, Curr. Ther. Res. 1972, 14, 454-460.
23. R. W. Yaung, K. H. Wood, J. A. Eichler, J. A. Vaughan Jr., G. W. Anderson, J. Chem. Soc. 1956, 78, 4649-4654.
24. A. K. Shakya, P. Mishra, G. K. Patnaik, R. Sukla, R. C. Srimal, Arch. Pharm. Res. 1998, 21(6), 753-758.
25. A. Scoozzafava, C. T. Supuran, J. Enzyme Inhib. 1998, 13(2), 103-123.
26. K. Nishikawa, H. Shimakawa, Y. Inada, Y. Shibouta, S. Kikuchi, S. Yurugi, Y. Oka, Chem. Pharm. Bull. 1976, 24, 2057-2077.
27. M. T. Bogert, G. D. Beal, J. Am. Chem. Soc. 1924, 4, 1294-1301.
28. D. R. Desai, V. S. Patel, S. R. Patel, J. Indian Chem. Soc. 1966, 43, 531-537.
29. V. Patrow, O. Stephenson, A. J. Thomas, A. M. Wild, J. Chem. Soc. 1958, 1508-1515.
30. K. M. Modi, N. N. Vortoak, N. N. Shah, K. Lotlikar, U. K. Sheth, Arch. Intern. Pharmacodyn. 1963, 144, 51-57.
31. J. T. Litchfield, T. Wilcoxon, J. Pharmacol. Exp. Ther. 1949, 96, 99-113.