Block of cloned Kv4.3 potassium channels by dapoxetine

Neuropharmacology

Volumn 62, Issue 7, 2012, Pages 2261-2266

  Jeong, Imju ^a   Kim, Sae Woong ^a   Yoon, Shin Hee ^a   Hahn, Sang June ^a  

^a The Catholic University of Korea   (South Korea)

Author keywords

Closed state inactivation; Dapoxetine; Kv4.3; Open channel block; Premature ejaculation; SSRI

Indexed keywords

DAPOXETINE; POTASSIUM CHANNEL KV4.3; SHAL POTASSIUM CHANNEL; UNCLASSIFIED DRUG;

AMPLITUDE MODULATION; ANIMAL CELL; ARTICLE; CHO CELL; CONCENTRATION RESPONSE; CONTROLLED STUDY; DISSOCIATION; HYPERPOLARIZATION; IC 50; MEMBRANE POTENTIAL; NONHUMAN; PATCH CLAMP; PHARMACOLOGICAL BLOCKING; PRIORITY JOURNAL; PROTEIN EXPRESSION; STEADY STATE;

EID: 84862831596     PISSN: 00283908     EISSN: 18737064     Source Type: Journal    
DOI: 10.1016/j.neuropharm.2011.12.006     Document Type: Article

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