Genetically encoded photo-cross-linkers map the binding site of an allosteric drug on a G protein-coupled receptor

ACS Chemical Biology

Volumn 7, Issue 6, 2012, Pages 967-972

  Grunbeck, Amy ^a   Huber, Thomas ^a   Abrol, Ravinder ^b   Trzaskowski, Bartosz ^b   Goddard III, William A ^b   Sakmar, Thomas P ^a  

^a ROCKEFELLER UNIVERSITY   (United States)

^b CALIFORNIA INSTITUTE OF TECHNOLOGY   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

G PROTEIN COUPLED RECEPTOR; MARAVIROC;

ARTICLE; CROSS LINKING; CRYSTAL STRUCTURE; DRUG BINDING SITE; DRUG LABELING; DRUG RECEPTOR BINDING; ISOTOPE LABELING; PHOTO CROSS LINKING; PRIORITY JOURNAL;

ALLOSTERIC SITE; CROSS-LINKING REAGENTS; CYCLOHEXANES; HEK293 CELLS; HIV FUSION INHIBITORS; HIV INFECTIONS; HIV-1; HUMANS; MODELS, MOLECULAR; MUTAGENESIS, SITE-DIRECTED; MUTATION; RECEPTORS, CCR5; TRIAZOLES; ULTRAVIOLET RAYS; VIRUS INTERNALIZATION;

EID: 84862526546     PISSN: 15548929     EISSN: 15548937     Source Type: Journal    
DOI: 10.1021/cb300059z     Document Type: Article

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