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Volumn 281, Issue 1, 2000, Pages 62-67

High-throughput screening of enzyme inhibitors: Automatic determination of tight-binding inhibition constants

(6) Kuzmič, Petr a Sideris, Steve b Cregar, Lynne M b Elrod, Kyle C b Rice, Kenneth D b Janc, James W b

b Axys Pharmaceuticals Inc (United States)

Author keywords

Data analysis; Enzyme kinetics; High throughput screening; Inhibition constant; Mast cell tryptase; Mathematics; Statistics; Tight binding

Indexed keywords

DATA REDUCTION; ENZYME KINETICS; ESTIMATION; MATHEMATICAL TECHNIQUES; STATISTICS;

AUTOMATIC DETERMINATION; AUTOMATIC PROCEDURES; HIGH THROUGHPUT SCREENING; HUMAN INTERVENTION; INHIBITION CONSTANTS; MAST CELLS; NON-LINEAR LEAST SQUARES; TIGHT BINDING;

ENZYME INHIBITION;

APC 1390; ENZYME INHIBITOR; PHENYLGUANIDINE; UNCLASSIFIED DRUG;

ARTICLE; COMPUTER PROGRAM; DOSE RESPONSE; ENZYME INHIBITOR COMPLEX; HUMAN; HUMAN CELL; INHIBITION KINETICS; INTERMETHOD COMPARISON; LABORATORY AUTOMATION; MAST CELL; MATHEMATICAL ANALYSIS; PRIORITY JOURNAL; RELIABILITY;

EID: 0034657809 PISSN: 00032697 EISSN: None Source Type: Journal
DOI: 10.1006/abio.2000.4501 Document Type: Article

Times cited : (55)

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