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Volumn 6, Issue 12, 2011, Pages 2233-2242

New Prodrugs of the Antiprotozoal Drug Pentamidine

(8) Kotthaus, Joscha a Kotthaus, Jürke a Schade, Dennis a Schwering, Ulrike a Hungeling, Helen a Müller Fielitz, Helge b Raasch, Walter b Clement, Bernd a

a UNIVERSITY OF KIEL (Germany)

b UNIVERSITY OF LÜBECK (Germany)

Author keywords

Amidoximes; Oral bioavailability; Pentamidines; Prodrugs; Trypanosomiasis

Indexed keywords

AMIDOXIMES; ANTIPROTOZOAL AGENT; PENTAMIDINE; PRODRUG; UNCLASSIFIED DRUG;

ALKYLATION; ANIMAL EXPERIMENT; ANIMAL MODEL; ANIMAL TISSUE; ANTIPROTOZOAL ACTIVITY; ARTICLE; CONTROLLED STUDY; DRUG BIOAVAILABILITY; DRUG DELIVERY SYSTEM; DRUG DETERMINATION; DRUG DISTRIBUTION; DRUG PENETRATION; DRUG SOLUBILITY; DRUG STABILITY; IN VITRO STUDY; IN VIVO STUDY; MALE; NONHUMAN; PRIORITY JOURNAL; RAT;

ADMINISTRATION, ORAL; ANIMALS; ANTIPROTOZOAL AGENTS; CELL LINE; CELL MEMBRANE PERMEABILITY; CYTOCHROME P-450 ENZYME SYSTEM; DRUG STABILITY; HUMANS; HYDROGEN-ION CONCENTRATION; MALE; MICROSOMES, LIVER; PENTAMIDINE; PRODRUGS; PROTEIN BINDING; RATS; RATS, SPRAGUE-DAWLEY; SWINE; TISSUE DISTRIBUTION;

EID: 82955161528 PISSN: 18607179 EISSN: 18607187 Source Type: Journal
DOI: 10.1002/cmdc.201100422 Document Type: Article

Times cited : (22)

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