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Volumn 12, Issue 17, 2011, Pages 2640-2646

Dynamic substrate enhancement for the identification of specific, second-site-binding fragments targeting a set of protein tyrosine phosphatases

(3) Schmidt, Marco F b,c,e Groves, Matthew R d Rademann, Jörg a,b

a UNIVERSITY OF LEIPZIG (Germany)

b LEIBNIZ INSTITUT FÜR MOLEKULARE PHARMAKOLOGIE (Germany)

c FREIE UNIVERSITÄT BERLIN (Germany)

d EUROPEAN MOLECULAR BIOLOGY LABORATORY (Germany)

e UNIVERSITY OF CAMBRIDGE (United Kingdom)

Author keywords

Drug discovery; Dynamic ligation assay; Mycobacterium tuberculosis; Protein tyrosine phosphatases; Second site binders

Indexed keywords

BACTERIAL ENZYME; HEMATOPOIETIC PROTEIN TYROSINE PHOSPHATASE; PHOSPHOTYROSINE; PROTEIN TYROSINE PHOSPHATASE; PROTEIN TYROSINE PHOSPHATASE 1B; PROTEIN TYROSINE PHOSPHATASE A; PROTEIN TYROSINE PHOSPHATASE INHIBITOR; PROTEIN TYROSINE PHOSPHATASE SHP 2; UNCLASSIFIED DRUG;

ARTICLE; BINDING SITE; CONTROLLED STUDY; COVALENT BOND; ENZYME SUBSTRATE; ENZYME SUBSTRATE COMPLEX; PRIORITY JOURNAL; SCREENING;

BACTERIAL PROTEINS; BINDING SITES; CATALYTIC DOMAIN; COMPUTER SIMULATION; ENZYME INHIBITORS; HUMANS; KINETICS; PROTEIN TYROSINE PHOSPHATASE, NON-RECEPTOR TYPE 1; PROTEIN TYROSINE PHOSPHATASES; SUBSTRATE SPECIFICITY;

BACTERIA (MICROORGANISMS); MYCOBACTERIUM TUBERCULOSIS;

EID: 81555205139 PISSN: 14394227 EISSN: 14397633 Source Type: Journal
DOI: 10.1002/cbic.201100414 Document Type: Article

Times cited : (22)

References (30)

1
- 0034614490
- T. Hunter, Cell 2000, 100, 113-127.
- (2000) Cell , vol.100 , pp. 113-127
- Hunter, T.¹

2
- 2942581416
- A. Alonso, J. Sasin, N. Bottini, I. Friedberg, I. Friedberg, A. Osterman, A. Godzik, T. Hunter, J. Dixon, T. Mustelin, Cell 2004, 117, 699-711.
- (2004) Cell , vol.117 , pp. 699-711
- Alonso, A.¹ Sasin, J.² Bottini, N.³ Friedberg, I.⁴ Friedberg, I.⁵ Osterman, A.⁶ Godzik, A.⁷ Hunter, T.⁸ Dixon, J.⁹ Mustelin, T.¹⁰

3
- 0042071479
- O. M. Fischer, S. Streit, S. Hart, A. Ullrich, Curr. Opin. Chem. Biol. 2003, 7, 490-495.
- (2003) Curr. Opin. Chem. Biol. , vol.7 , pp. 490-495
- Fischer, O.M.¹ Streit, S.² Hart, S.³ Ullrich, A.⁴

4
- 1642323740
- M. E. Noble, J. A. Endicott, L. N. Johnson, Science 2004, 303, 1800-1805.
- (2004) Science , vol.303 , pp. 1800-1805
- Noble, M.E.¹ Endicott, J.A.² Johnson, L.N.³

5
- 21244444303
- L. Bialy, H. Waldmann, Angew. Chem. 2005, 117, 3880-3906; Angew. Chem. Int. Ed. 2005, 44, 3814-3839.
- (2005) Angew. Chem. 2005, 117, 3880-3906; Angew. Chem. Int. Ed. , vol.44 , pp. 3814-3839
- Bialy, L.¹ Waldmann, H.²

6
- 33846460390
- A. K. H. Hirsch, F. R. Fischer, F. Diederich, Angew. Chem. 2007, 119, 342-357; Angew. Chem. Int. Ed. 2007, 46, 338-352.
- (2007) Angew. Chem. 2007, 119, 342-357; Angew. Chem. Int. Ed. , vol.46 , pp. 338-352
- Hirsch, A.K.H.¹ Fischer, F.R.² Diederich, F.³

7
- 67949124765
- M. A. T. Blaskovich, Curr. Med. Chem. 2009, 16, 2095-2176.
- (2009) Curr. Med. Chem. , vol.16 , pp. 2095-2176
- Blaskovich, M.A.T.¹

8
- 58249138122
- A. J. Barr, E. Ugochukwu, K. W. Lee, O. N. King, P. Filippakopoulos, I. Alfano, P. Savitsky, N. A. Burgess-Brown, S. Müller, S. Knapp, Cell 2009, 136, 352-363.
- (2009) Cell , vol.136 , pp. 352-363
- Barr, A.J.¹ Ugochukwu, E.² Lee, K.W.³ King, O.N.⁴ Filippakopoulos, P.⁵ Alfano, I.⁶ Savitsky, P.⁷ Burgess-Brown, N.A.⁸ Müller, S.⁹ Knapp, S.¹⁰

9
- 37549048176
- A. Ciulli, C. Abell, Curr. Opin. Biotechnol. 2007, 18, 489-496.
- (2007) Curr. Opin. Biotechnol. , vol.18 , pp. 489-496
- Ciulli, A.¹ Abell, C.²

10
- 68749088518
- M. F. Schmidt, J. Rademann, Trends Biotechnol. 2009, 27, 512-521.
- (2009) Trends Biotechnol. , vol.27 , pp. 512-521
- Schmidt, M.F.¹ Rademann, J.²

11
- 44949155667
- M. F. Schmidt, A. Isidro-Llobet, M. Lisurek, A. El-Dahshan, J. Tan, R. Hilgenfeld, J. Rademann, Angew. Chem. 2008, 120, 3319-3323; Angew. Chem. Int. Ed. 2008, 47, 3275-3278.
- (2008) Angew. Chem. 2008, 120, 3319-3323; Angew. Chem. Int. Ed. , vol.47 , pp. 3275-3278
- Schmidt, M.F.¹ Isidro-Llobet, A.² Lisurek, M.³ El-Dahshan, A.⁴ Tan, J.⁵ Hilgenfeld, R.⁶ Rademann, J.⁷

12
- 70349907092
- M. F. Schmidt, A. El-Dahshan, S. Keller, J. Rademann, Angew. Chem. 2009, 121, 6464-6467; Angew. Chem. Int. Ed. 2009, 48, 6346-6349.
- (2009) Angew. Chem. 2009, 121, 6464-6467; Angew. Chem. Int. Ed. , vol.48 , pp. 6346-6349
- Schmidt, M.F.¹ El-Dahshan, A.² Keller, S.³ Rademann, J.⁴

13
- 34547758886
- M. B. Soellner, K. A. Rawls, H. Tsuruoka, R. K. Jain, J. A. Ellman, J. Am. Chem. Soc. 2007, 129, 9613-9615.
- (2007) J. Am. Chem. Soc. , vol.129 , pp. 9613-9615
- Soellner, M.B.¹ Rawls, K.A.² Tsuruoka, H.³ Jain, R.K.⁴ Ellman, J.A.⁵

14
- 0023917654
- A. A. Baykov, O. A. Evtushenko, S. M. Avaeva, Anal. Biochem. 1988, 171, 266-270.
- (1988) Anal. Biochem. , vol.171 , pp. 266-270
- Baykov, A.A.¹ Evtushenko, O.A.² Avaeva, S.M.³

15
- 43049181499
- H. Bach, K. G. Papavinasasundaram, D. Wong, Z. Hmama, Y. Av-Gay, Cell Host Microbe 2008, 3, 316-322.
- (2008) Cell Host Microbe , vol.3 , pp. 316-322
- Bach, H.¹ Papavinasasundaram, K.G.² Wong, D.³ Hmama, Z.⁴ Av-Gay, Y.⁵

16
- 0033525870
- M. Elchebly, P. Payette, E. Michaliszyn, W. Cromlish, S. Collins, A. L. Loy, D. Normandin, A. Cheng, J. Himms-Hagen, C.-C. Chan, C. Ramachandran, M. J. Gresser, M. L. Tremblay, B. P. Kennedy, Science 1999, 283, 1544-1548.
- (1999) Science , vol.283 , pp. 1544-1548
- Elchebly, M.¹ Payette, P.² Michaliszyn, E.³ Cromlish, W.⁴ Collins, S.⁵ Loy, A.L.⁶ Normandin, D.⁷ Cheng, A.⁸ Himms-Hagen, J.⁹ Chan, C.-C.¹⁰ Ramachandran, C.¹¹ Gresser, M.J.¹² Tremblay, M.L.¹³ Kennedy, B.P.¹⁴

17
- 0027957970
- B. Zanke, J. Squire, H. Griesser, M. Henry, H. Suzuki, B. Patterson, M. Minden, T. W. Mak, Leukemia 1994, 8, 236-244.
- (1994) Leukemia , vol.8 , pp. 236-244
- Zanke, B.¹ Squire, J.² Griesser, H.³ Henry, M.⁴ Suzuki, H.⁵ Patterson, B.⁶ Minden, M.⁷ Mak, T.W.⁸

18
- 44449083477
- K. Hellmuth, S. Grosskopf, C. T. Lum, M. Würtele, N. Röder, J. P. von Kries, M. Rosario, J. Rademann, W. Birchmeier, Proc. Natl. Acad. Sci. USA 2008, 105, 7275-7280.
- (2008) Proc. Natl. Acad. Sci. USA , vol.105 , pp. 7275-7280
- Hellmuth, K.¹ Grosskopf, S.² Lum, C.T.³ Würtele, M.⁴ Röder, N.⁵ von Kries, J.P.⁶ Rosario, M.⁷ Rademann, J.⁸ Birchmeier, W.⁹

19
- 77954684593
- M. Lisurek, B. Rupp, J. Wichard, M. Neuenschwander, J. P. von Kries, R. Frank, J. Rademann, R. Kühne, Mol. Diversity 2010, 14, 401-408.
- (2010) Mol. Diversity , vol.14 , pp. 401-408
- Lisurek, M.¹ Rupp, B.² Wichard, J.³ Neuenschwander, M.⁴ von Kries, J.P.⁵ Frank, R.⁶ Rademann, J.⁷ Kühne, R.⁸

20
- 34249052551
- L. Tautz, T. Mustelin, Methods 2007, 42, 250-260.
- (2007) Methods , vol.42 , pp. 250-260
- Tautz, L.¹ Mustelin, T.²

21
- 67049137557
- R. Maccari, R. Ottanà, R. Ciurleo, P. Paoli, G. Manao, G. Camici, C. Laggner, T. Langer, ChemMedChem 2009, 4, 957-962.
- (2009) ChemMedChem , vol.4 , pp. 957-962
- Maccari, R.¹ Ottanà, R.² Ciurleo, R.³ Paoli, P.⁴ Manao, G.⁵ Camici, G.⁶ Laggner, C.⁷ Langer, T.⁸

22
- 0000468730
- M. M. Mader, P. A. Bartlett, Chem. Rev. 1997, 97, 1281-1301.
- (1997) Chem. Rev. , vol.97 , pp. 1281-1301
- Mader, M.M.¹ Bartlett, P.A.²

23
- 84859477826
- S. Großkopf, J. Rademann, unpublished results;
- S. Großkopf, J. Rademann, unpublished results.

24
- 0037377337
- P. Huang, J. Ramphal, J. Wei, C. Liang, B. Jallal, G. McMahon, C. Tang, Bioorg. Med. Chem. 2003, 11, 1835-1849.
- (2003) Bioorg. Med. Chem. , vol.11 , pp. 1835-1849
- Huang, P.¹ Ramphal, J.² Wei, J.³ Liang, C.⁴ Jallal, B.⁵ McMahon, G.⁶ Tang, C.⁷

25
- 14644438366
- C. Madhurantakam, E. Rajakumara, P. A. Mazumdar, B. Saha, D. Mitra, H. G. Wiker, R. Sankaranarayanan, A. K. Das, J. Bacteriol. 2005, 187, 2175-2181.
- (2005) J. Bacteriol. , vol.187 , pp. 2175-2181
- Madhurantakam, C.¹ Rajakumara, E.² Mazumdar, P.A.³ Saha, B.⁴ Mitra, D.⁵ Wiker, H.G.⁶ Sankaranarayanan, R.⁷ Das, A.K.⁸

26
- 26944488334
- M. Manger, M. Scheck, H. Prinz, J. P. von Kries, T. Langer, K. Saxena, H. Schwalbe, A. Fuerstner, J. Rademann, H. Waldmann, ChemBioChem 2005, 6, 1749-1753.
- (2005) ChemBioChem , vol.6 , pp. 1749-1753
- Manger, M.¹ Scheck, M.² Prinz, H.³ von Kries, J.P.⁴ Langer, T.⁵ Saxena, K.⁶ Schwalbe, H.⁷ Fuerstner, A.⁸ Rademann, J.⁹ Waldmann, H.¹⁰

27
- 55549140118
- L. D. Chiaradia, A. Mascarello, M. Purifição, J. Vernal, M. N. S. Cordeiro, M. E. Zenteno, A. Villarino, R. J. Nunes, R. A. Yunes, H. Terenzi, Bioorg. Med. Chem. Lett. 2008, 18, 6227-6230.
- (2008) Bioorg. Med. Chem. Lett. , vol.18 , pp. 6227-6230
- Chiaradia, L.D.¹ Mascarello, A.² Purifição, M.³ Vernal, J.⁴ Cordeiro, M.N.S.⁵ Zenteno, M.E.⁶ Villarino, A.⁷ Nunes, R.J.⁸ Yunes, R.A.⁹ Terenzi, H.¹⁰

28
- 71849090071
- K. A. Rawls, P. T. Lang, J. Takeuchi, S. Imamura, T. D. Baguley, C. Grundner, T. Alber, J. A. Ellman, Bioorg. Med. Chem. Lett. 2009, 19, 6851-6854.
- (2009) Bioorg. Med. Chem. Lett. , vol.19 , pp. 6851-6854
- Rawls, K.A.¹ Lang, P.T.² Takeuchi, J.³ Imamura, S.⁴ Baguley, T.D.⁵ Grundner, C.⁶ Alber, T.⁷ Ellman, J.A.⁸

29
- 76649119460
- G. Kemmer, S. Keller, Nat. Protoc. 2010, 5, 267-281.
- (2010) Nat. Protoc. , vol.5 , pp. 267-281
- Kemmer, G.¹ Keller, S.²

30
- 0003845223
- v.0.99, DeLano Scientific, San Carlos.
- W. L. DeLano, The PyMOL Molecular Graphics System, v.0.99, DeLano Scientific, San Carlos, 2002.
- (2002) The PyMOL Molecular Graphics System
- DeLano, W.L.¹

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