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Volumn 46, Issue 9, 2011, Pages 4100-4106

Synthesis, characterization and pharmacological activity of 4-{[1-substituted aminomethyl-4-arylideneamino-5-sulfanyl-4,5-dihydro-1H-1,2,4- triazol-3-yl]methyl}-2H-1,4-benzothiazin-3(4H)-ones

(5) Gowda, J a Khader, A M A a Kalluraya, B a Shree, Padma b Shabaraya, A R b

a MANGALORE UNIVERSITY (India)

b SRINIVAS COLLEGE OF PHARMACY (India)

Author keywords

1,4 Benzothiazin 3(4H) one; Analgesic activity; Anti inflammatory activity

Indexed keywords

(3 OXO 2,3 DIHYDRO 4H 1,4 BENZOTHIAZIN 4 YL)ACETIC ACID; 4 [(1 MORPHOLINOMETHYL 4 BENZYLIDENEAMINO 5 SULFANYL 4,5 DIHYDRO 1H 1,2,4 TRIAZOL 3 YL)METHYL] 2H 1,4 BENZOTHIAZIN 3(4H) ONE; 4 [(1 N METHYL PIPERAZINOMETHYL 4 BENZYLIDENEAMINO 5 SULFANYL 4,5 DIHYDRO 1H 1,2,4 TRIAZOL 3 YL)METHYL] 2H 1,4 BENZOTHIAZIN 3(4H) ONE; 4 [(1 PIPERIDINOMETHYL 4 BENZYLIDENEAMINO 5 SULFANYL 4,5 DIHYDRO 1H 1,2,4 TRIAZOL 3 YL)METHYL] 2H 1,4 BENZOTHIAZIN 3(4H) ONE; 4 [[1 MORPHOLINOMETHYL 4 (PARA CHLORO BENZYLIDENEAMINO) 5 SULFANYL 4,5 DIHYDRO 1H 1,2,4 TRIAZOL 3 YL]METHYL] 2H 1,4 BENZOTHIAZIN 3(4H) ONE; 4 [[1 MORPHOLINOMETHYL 4 (PARA HYDROXY BENZYLIDENEAMINO) 5 SULFANYL 4,5 DIHYDRO 1H 1,2,4 TRIAZOL 3 YL]METHYL] 2H 1,4-BENZOTHIAZIN 3(4H) ONE; 4 [[1 MORPHOLINOMETHYL 4 (PARA NITRO BENZYLIDENENEAMINO) 5 SULFANYL 4,5 DIHYDRO 1H 1,2,4 TRIAZOL 3 YL]METHYL] 2H 1,4 BENZOTHIAZIN 3(4H) ONE; 4 [[1 N METHYL PIPERAZINOMETHYL 4 (PARA CHLORO BENZYLIDENEAMINO) 5 SULFANYL 4,5 DIHYDRO 1H 1,2,4 TRIAZOL 3 YL]METHYL] 2H 1,4 BENZOTHIAZIN 3(4H) ONE; 4 [[1 N METHYL PIPERAZINOMETHYL 4 (PARA NITRO BENZYLIDENENEAMINO) 5 SULFANYL 4,5 DIHYDRO 1H 1,2,4 TRIAZOL 3 YL]METHYL] 2H 1,4 BENZOTHIAZIN 3(4H) ONE; 4 [[1 PIPERIDINOMETHYL 4 (PARA CHLORO BENZYLIDENEAMINO) 5 SULFANYL 4,5 DIHYDRO 1H 1,2,4 TRIAZOL 3 YL]METHYL] 2H 1,4 BENZOTHIAZIN 3(4H) ONE; 4 [[1 PIPERIDINOMETHYL 4 (PARA HYDROXY BENZYLIDENEAMINO) 5 SULFANYL 4,5 DIHYDRO 1H 1,2,4 TRIAZOL 3 YL]METHYL] 2H 1,4 BENZOTHIAZIN 3(4H) ONE; 4 [[1 PIPERIDINOMETHYL 4 (PARA NITRO BENZYLIDENENEAMINO) 5 SULFANYL 4,5 DIHYDRO 1H 1,2,4 TRIAZOL 3 YL]METHYL] 2H 1,4 BENZOTHIAZIN 3(4H) ONE; ANALGESIC AGENT; ANTIINFLAMMATORY AGENT; CARBOXYLIC ACID; INDOMETACIN; MANNICH BASE; PENTAZOCINE; SCHIFF BASE; UNCLASSIFIED DRUG;

ANALGESIC ACTIVITY; ANIMAL EXPERIMENT; ANIMAL MODEL; ANTIINFLAMMATORY ACTIVITY; ARTICLE; CONTROLLED STUDY; DERIVATIZATION; DRUG SCREENING; DRUG STRUCTURE; DRUG SYNTHESIS; FEMALE; INFRARED RADIATION; MALE; MASS SPECTROMETRY; NONHUMAN; PAW EDEMA; PROTON NUCLEAR MAGNETIC RESONANCE; RAT;

ANIMALS; ANTI-INFLAMMATORY AGENTS; FEMALE; MAGNETIC RESONANCE SPECTROSCOPY; MALE; MASS SPECTROMETRY; RATS; RATS, WISTAR; SPECTROPHOTOMETRY, INFRARED; THIAZINES;

EID: 80052923006 PISSN: 02235234 EISSN: 17683254 Source Type: Journal
DOI: 10.1016/j.ejmech.2011.06.010 Document Type: Article

Times cited : (49)

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