Synthesis and biological evaluation of substituted 4-arylthiazol-2-amino derivatives as potent growth inhibitors of replicating Mycobacterium tuberculosis H 37R V

Bioorganic and Medicinal Chemistry Letters

Volumn 21, Issue 18, 2011, Pages 5589-5593

  Roy, Kuldeep K ^a   Singh, Supriya ^a   Sharma, Sandeep K ^a   Srivastava, Ranjana ^a   Chaturvedi, Vinita ^a   Saxena, Anil K ^a  

^a CENTRAL DRUG RESEARCH INSTITUTE   (India)

Author keywords

Anti tubercular; Minimum inhibitory concentration (MIC); Mycobacterium tuberculosis; Nitazoxanide; Phenylthiazole

Indexed keywords

4 ARYLTHIAZOL 2 AMINO DERIVATIVE; ISONIAZID; NITAZOXANIDE; RIFAMPICIN; STREPTOMYCIN; THIAZOLE DERIVATIVE; TIZOXANIDE; TUBERCULOSTATIC AGENT; UNCLASSIFIED DRUG;

ARTICLE; BACTERIAL STRAIN; BIOLOGICAL ACTIVITY; DRUG SYNTHESIS; MINIMUM INHIBITORY CONCENTRATION; MYCOBACTERIUM TUBERCULOSIS; NONHUMAN;

ANTI-BACTERIAL AGENTS; CHEMISTRY TECHNIQUES, SYNTHETIC; DOSE-RESPONSE RELATIONSHIP, DRUG; MICROBIAL SENSITIVITY TESTS; MOLECULAR STRUCTURE; MYCOBACTERIUM TUBERCULOSIS; STEREOISOMERISM; STRUCTURE-ACTIVITY RELATIONSHIP; THIAZOLES;

MYCOBACTERIUM TUBERCULOSIS;

EID: 80051940406     PISSN: 0960894X     EISSN: 14643405     Source Type: Journal    
DOI: 10.1016/j.bmcl.2011.06.076     Document Type: Article

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