Multiple inhibitory actions of lidocaine on Torpedo nicotinic acetylcholine receptors transplanted to Xenopus oocytes

Journal of Neurochemistry

Volumn 117, Issue 6, 2011, Pages 1009-1019

  Alberola Die, Armando ^a   Martinez Pinna, Juan ^a   González Ros, José Manuel ^b   Ivorra, Isabel ^a   Morales, Andrés ^a  

^a UNIVERSITY OF ALICANTE   (Spain)

^b MIGUEL HERNÁNDEZ UNIVERSITY   (Spain)

Author keywords

lidocaine; local anaesthetics; microtransplantation; nicotinic acetylcholine receptors; QX 314; Xenopus oocytes

Indexed keywords

1,5 BIS(4 ALLYLDIMETHYLAMMONIUMPHENYL)PENTAN 3 ONE DIBROMIDE; 2 (TRIETHYLAMMONIO) N (2,6 DIMETHYLPHENYL)ACETAMIDE BROMIDE; ACETYLCHOLINE; EDROPHONIUM; LIDOCAINE; NICOTINIC RECEPTOR; QUATERNARY AMMONIUM DERIVATIVE; UNCLASSIFIED DRUG;

ANESTHESIA MECHANISM; ANIMAL CELL; ARTICLE; CELL MEMBRANE; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG BINDING SITE; ELECTRIC FIELD; FEMALE; IC 50; INHIBITION KINETICS; NONHUMAN; OOCYTE; PRIORITY JOURNAL; RECEPTOR BLOCKING; TORPEDO MARMORATA; XENOPUS LAEVIS;

ACETYLCHOLINE; ANESTHETICS, LOCAL; ANIMALS; BENZENAMINIUM, 4,4'-(3-OXO-1,5-PENTANEDIYL)BIS(N,N-DIMETHYL-N-2-PROPENYL-), DIBROMIDE; DOSE-RESPONSE RELATIONSHIP, DRUG; DRUG SYNERGISM; EDROPHONIUM; FEMALE; ION CHANNEL GATING; LIDOCAINE; MEMBRANE POTENTIALS; NICOTINIC ANTAGONISTS; OOCYTES; RECEPTORS, NICOTINIC; TORPEDO; XENOPUS LAEVIS;

EID: 79957979913     PISSN: 00223042     EISSN: 14714159     Source Type: Journal    
DOI: 10.1111/j.1471-4159.2011.07271.x     Document Type: Article

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