메뉴 건너뛰기




Volumn 63, Issue 3, 2011, Pages 352-361

Supersaturated dissolution data and their interpretation: The TPGS-carbamazepine model case

Author keywords

Carbamazepine; Dissolution; Solubility; Supersaturation; Vitamin E TPGS

Indexed keywords

ALPHA TOCOPHEROL; ALPHA TOCOPHERYL POLYETHYLENE GLYCOL 1000 SUCCINATE; CARBAMAZEPINE; MACROGOL; MICROCRYSTALLINE CELLULOSE; SILICON DIOXIDE; UNCLASSIFIED DRUG;

EID: 79952237126     PISSN: 00223573     EISSN: None     Source Type: Journal    
DOI: 10.1111/j.2042-7158.2010.01226.x     Document Type: Article
Times cited : (17)

References (45)
  • 2
    • 37849045222 scopus 로고    scopus 로고
    • Dissolution improvement of four poorly water soluble drugs by cogrinding with commonly used excipients
    • Vogt M et al. Dissolution improvement of four poorly water soluble drugs by cogrinding with commonly used excipients. Eur J Pharm Biopharm 2008; 68: 330-337.
    • (2008) Eur J Pharm Biopharm , vol.68 , pp. 330-337
    • Vogt, M.1
  • 3
    • 41549150839 scopus 로고    scopus 로고
    • Formulation and characterization of ternary solid dispersions made up of Itraconazole and two excipients, TPGS 1000 and PVPVA 64, that were selected based on a supersaturation screening study
    • Janssens S et al. Formulation and characterization of ternary solid dispersions made up of Itraconazole and two excipients, TPGS 1000 and PVPVA 64, that were selected based on a supersaturation screening study. Eur J Pharm Biopharm 2008; 69: 158-166.
    • (2008) Eur J Pharm Biopharm , vol.69 , pp. 158-166
    • Janssens, S.1
  • 4
    • 52949150391 scopus 로고    scopus 로고
    • Effect of polymer type on the dissolution profile of amorphous solid dispersions containing felodipine
    • Konno H et al. Effect of polymer type on the dissolution profile of amorphous solid dispersions containing felodipine. Eur J Pharm Biopharm 2008; 70: 493-499.
    • (2008) Eur J Pharm Biopharm , vol.70 , pp. 493-499
    • Konno, H.1
  • 5
    • 53849129520 scopus 로고    scopus 로고
    • Dissolution improvement and the mechanism of the improvement from cocrystallization of poorly water-soluble compounds
    • Shiraki K et al. Dissolution improvement and the mechanism of the improvement from cocrystallization of poorly water-soluble compounds. Pharm Res 2008; 25: 2581-2592.
    • (2008) Pharm Res , vol.25 , pp. 2581-2592
    • Shiraki, K.1
  • 6
    • 85047686260 scopus 로고    scopus 로고
    • Cefuroxime axetil solid dispersion with polyglycolized glycerides for improved stability and bioavailability
    • Dhumal RS et al. Cefuroxime axetil solid dispersion with polyglycolized glycerides for improved stability and bioavailability. J Pharm Pharmacol 2009; 61: 743-751.
    • (2009) J Pharm Pharmacol , vol.61 , pp. 743-751
    • Dhumal, R.S.1
  • 7
    • 0036771080 scopus 로고    scopus 로고
    • Physicochemical characterization of solid dispersions of carbamazepine formulated by supercritical carbon dioxide and conventional solvent evaporation method
    • DOI 10.1002/jps.10186
    • Sethia S, Squillante E. Physicochemical characterization of solid dispersions of carbamazepine formulated by supercritical carbon dioxide and conventional solvent evaporation methods. J Pharm Sci 2002; 91: 1948-1957. (Pubitemid 36254931)
    • (2002) Journal of Pharmaceutical Sciences , vol.91 , Issue.9 , pp. 1948-1957
    • Sethia, S.1    Squillante, E.2
  • 8
    • 1442348833 scopus 로고    scopus 로고
    • Solid dispersion of carbamazepine in PVP K30 by conventional solvent evaporation and supercritical methods
    • DOI 10.1016/j.ijpharm.2003.11.025, PII S037851730300629X
    • Sethia S, Squillante E. Solid dispersion of carbamazepine in PVP K30 by conventional solvent evaporation and supercritical methods. Int J Pharm 2004; 272: 1-10. (Pubitemid 38293005)
    • (2004) International Journal of Pharmaceutics , vol.272 , Issue.1-2 , pp. 1-10
    • Sethia, S.1    Squillante, E.2
  • 9
    • 0034607429 scopus 로고    scopus 로고
    • Membrane penetration enhancement of ibuprofen using supersaturation
    • DOI 10.1016/S0378-5173(00)00346-X, PII S037851730000346X
    • Iervolino M et al. Membrane penetration enhancement of ibuprofen using supersaturation. Int J Pharm 2000; 198: 229-238. (Pubitemid 30184859)
    • (2000) International Journal of Pharmaceutics , vol.198 , Issue.2 , pp. 229-238
    • Iervolino, M.1    Raghavan, S.L.2    Hadgraft, J.3
  • 10
    • 0036245046 scopus 로고    scopus 로고
    • Study of the complexation behavior of tenoxicam with cyclodextrins in solution: Improved solubility and percutaneous permeability
    • DOI 10.1081/DDC-120002840
    • Larrucea E et al. Study of the complexation behavior of tenoxicam with cyclodextrins in solution: improved solubility and percutaneous permeability. Drug Dev Ind Pharm 2002; 28: 245-252. (Pubitemid 34475671)
    • (2002) Drug Development and Industrial Pharmacy , vol.28 , Issue.3 , pp. 245-252
    • Larrucea, E.1    Arellano, A.2    Santoyo, S.3    Ygartua, P.4
  • 11
    • 0037965572 scopus 로고    scopus 로고
    • Processing of nimesulide-PEG 400-PG-PVP solid dispersions: Preparation, characterization, and in vitro dissolution
    • DOI 10.1081/DDC-120018203
    • Gohel MC, Patel LD. Processing of nimesulide-PEG 400-PGPVP solid dispersions: preparation, characterization, and in vitro dissolution. Drug Dev Ind Pharm 2003; 29: 299-310. (Pubitemid 36528620)
    • (2003) Drug Development and Industrial Pharmacy , vol.29 , Issue.3 , pp. 299-310
    • Gohel, M.C.1    Patel, L.D.2
  • 12
    • 33747375906 scopus 로고    scopus 로고
    • The effects of surfactants on the dissolution profiles of poorly water-soluble acidic drugs
    • Park SH, Choi HK. The effects of surfactants on the dissolution profiles of poorly water-soluble acidic drugs. Int J Pharm 2006; 321: 35-41.
    • (2006) Int J Pharm , vol.321 , pp. 35-41
    • Park, S.H.1    Choi, H.K.2
  • 14
    • 34247612824 scopus 로고    scopus 로고
    • In vitro behavior of a phosphate ester prodrug of amprenavir in human intestinal fluids and in the Caco-2 system: Illustration of intraluminal supersaturation
    • DOI 10.1016/j.ijpharm.2006.12.011, PII S0378517306010696
    • Brouwers J et al. In vitro behavior of a phosphate ester prodrug of amprenavir in human intestinal fluids and in the Caco-2 system: illustration of intraluminal supersaturation. Int J Pharm 2007; 336: 302-309. (Pubitemid 46670658)
    • (2007) International Journal of Pharmaceutics , vol.336 , Issue.2 , pp. 302-309
    • Brouwers, J.1    Tack, J.2    Augustijns, P.3
  • 15
    • 34548082187 scopus 로고    scopus 로고
    • Parallel monitoring of plasma and intraluminal drug concentrations in man after oral administration of fosamprenavir in the fasted and fed state
    • DOI 10.1007/s11095-007-9307-3
    • Brouwers J et al. Parallel monitoring of plasma and intraluminal drug concentrations in man after oral administration of fosamprenavir in the fasted and fed state. Pharm Res 2007; 24: 1862-1869. (Pubitemid 47389240)
    • (2007) Pharmaceutical Research , vol.24 , Issue.10 , pp. 1862-1869
    • Brouwers, J.1    Tack, J.2    Augustijns, P.3
  • 16
    • 67349204296 scopus 로고    scopus 로고
    • Postprandial changes in solubilizing capacity of human intestinal fluids for BCS class II drugs
    • Clarysse S et al. Postprandial changes in solubilizing capacity of human intestinal fluids for BCS class II drugs. Pharm Res 2009; 26: 1456-1466.
    • (2009) Pharm Res , vol.26 , pp. 1456-1466
    • Clarysse, S.1
  • 17
    • 0034601240 scopus 로고    scopus 로고
    • Improving drug solubility for oral delivery using solid dispersions
    • DOI 10.1016/S0939-6411(00)00076-X, PII S093964110000076X
    • Leuner C, Dressman J. Improving drug solubility for oral delivery using solid dispersions. Eur J Pharm Biopharm 2000; 50: 47-60. (Pubitemid 30326688)
    • (2000) European Journal of Pharmaceutics and Biopharmaceutics , vol.50 , Issue.1 , pp. 47-60
    • Leuner, C.1    Dressman, J.2
  • 18
    • 1142303337 scopus 로고    scopus 로고
    • What is the true solubility advantage for amorphous pharmaceuticals?
    • DOI 10.1023/A:1007516718048
    • Hancock B, Parks M. What is the true solubility advantage for amorphous pharmaceuticals? Pharm Res 2001; 17: 397-404. (Pubitemid 30395293)
    • (2000) Pharmaceutical Research , vol.17 , Issue.4 , pp. 397-404
    • Hancock, B.C.1    Parks, M.2
  • 20
    • 0033986929 scopus 로고    scopus 로고
    • Effect of cellulose polymers on supersaturation and in vitro membrane transport of hydrocortisone acetate
    • DOI 10.1016/S0378-5173(99)00345-2, PII S0378517399003452
    • Raghavan SL et al. Effect of cellulose polymers on supersaturation and in vitro membrane transport of hydrocortisone acetate. Int J Pharm 2000; 193: 231-237. (Pubitemid 30001867)
    • (2000) International Journal of Pharmaceutics , vol.193 , Issue.2 , pp. 231-237
    • Raghavan, S.L.1    Trividic, A.2    Davis, A.F.3    Hadgraft, J.4
  • 22
    • 33646689478 scopus 로고    scopus 로고
    • Structural relaxation of acetaminophen glass
    • Gunawan LG et al. Structural relaxation of acetaminophen glass. Pharm Res 2006; 23: 967-979.
    • (2006) Pharm Res , vol.23 , pp. 967-979
    • Gunawan, L.G.1
  • 23
    • 0017178826 scopus 로고
    • Dissolution behavior and bioavailability of phenytoin from a ground mixture with microcrystalline cellulose
    • Yamamoto K et al. Dissolution behavior and bioavailability of phenytoin from a ground mixture with microcrystalline cellulose. J Pharm Sci 1976; 65: 1484-1488.
    • (1976) J Pharm Sci , vol.65 , pp. 1484-1488
    • Yamamoto, K.1
  • 24
    • 0025830658 scopus 로고
    • Dissolution and bioavailability of phenobarbital in solid dispersion with phosphatidylcholine
    • Fujii M et al. Dissolution and bioavailability of phenobarbital in solid dispersion with phosphatidylcholine. Chem Pharm Bull 1991; 39: 1886-1888.
    • (1991) Chem Pharm Bull , vol.39 , pp. 1886-1888
    • Fujii, M.1
  • 25
    • 0031958399 scopus 로고    scopus 로고
    • Influence of water-soluble polymers on the dissolution of Nifedipine solid dispersions with combined carriers
    • Suzki H, Sunada H. Influence of water-soluble polymers on the dissolution of nifedipine solid dispersions with combined carriers. Chem Pharm Bull 1998; 46: 482-487. (Pubitemid 28188567)
    • (1998) Chemical and Pharmaceutical Bulletin , vol.46 , Issue.3 , pp. 482-487
    • Suzuki, H.1    Sunada, H.2
  • 26
    • 33644881395 scopus 로고    scopus 로고
    • Stabilization of solid dispersions of nimodipine and polyethylene glycol 2000
    • Urbanetz NA. Stabilization of solid dispersions of nimodipine and polyethylene glycol 2000. Eur J Pharm Sci 2006; 28: 67-76.
    • (2006) Eur J Pharm Sci , vol.28 , pp. 67-76
    • Urbanetz, N.A.1
  • 29
    • 41349116109 scopus 로고    scopus 로고
    • Development of a reaction-limited model of dissolution: Application to official dissolution tests experiments
    • Dokoumetzidis A et al. Development of a reaction-limited model of dissolution: Application to official dissolution tests experiments. Int J Pharm 2008; 355: 114-125.
    • (2008) Int J Pharm , vol.355 , pp. 114-125
    • Dokoumetzidis, A.1
  • 30
    • 67650569218 scopus 로고    scopus 로고
    • A simulation of oral absorption using classical nucleation theory
    • Sugano K. A simulation of oral absorption using classical nucleation theory. Int J Pharm 2009; 378: 142-145.
    • (2009) Int J Pharm , vol.378 , pp. 142-145
    • Sugano, K.1
  • 31
    • 72449149167 scopus 로고    scopus 로고
    • Computational oral absorption simulation for low-solubility compounds
    • Sugano K. Computational oral absorption simulation for low-solubility compounds. Chem Biodivers 2009; 6: 2014-2029.
    • (2009) Chem Biodivers , vol.6 , pp. 2014-2029
    • Sugano, K.1
  • 32
    • 0033988596 scopus 로고    scopus 로고
    • Physicochemical properties and bioavailability of carbamazepine polymorphs and dihydrate
    • DOI 10.1016/S0378-5173(99)00315-4, PII S0378517399003154
    • Kobayashi Y et al. Physicochemical properties and bioavailability of carbamazepine polymorphs and dihydrate. Int J Pharm 2000; 193: 137-146. (Pubitemid 30001856)
    • (2000) International Journal of Pharmaceutics , vol.193 , Issue.2 , pp. 137-146
    • Kobayashi, Y.1    Ito, S.2    Itai, S.3    Yamamoto, K.4
  • 34
    • 0025880233 scopus 로고
    • Improvement of cyclosporin absorption in children after liver transplantation by means of water-soluble vitamin E
    • Sokol RJ et al. Improvement of cyclosporin absorption in children after liver transplantation by means of water-soluble vitamin E. Lancet 1991; 338: 212-214.
    • (1991) Lancet , vol.338 , pp. 212-214
    • Sokol, R.J.1
  • 36
    • 33747373878 scopus 로고    scopus 로고
    • A century of dissolution research: From Noyes and Whitney to the Biopharmaceutics Classification System
    • DOI 10.1016/j.ijpharm.2006.07.011, PII S0378517306005813
    • Dokoumetzidis A, Macheras P. A century of dissolution research: From Noyes and Whitney to the Biopharmaceutics Classification System. Int J Pharm 2006; 321: 1-11. (Pubitemid 44247428)
    • (2006) International Journal of Pharmaceutics , vol.321 , Issue.1-2 , pp. 1-11
    • Dokoumetzidis, A.1    Macheras, P.2
  • 37
    • 0005491022 scopus 로고    scopus 로고
    • A statistical rate theory study of interface concentration during crystal growth or dissolution
    • Dejmek M, Ward CA. A statistical rate theory study of interface concentration during crystal growth or dissolution. J Chem Phys 1998; 108: 8698-8704. (Pubitemid 128597379)
    • (1998) Journal of Chemical Physics , vol.108 , Issue.20 , pp. 8698-8704
    • Dejmek, M.1    Ward, C.A.2
  • 39
    • 0036482959 scopus 로고    scopus 로고
    • A novel method for estimation of transition temperature for polymorphic pairs in pharmaceuticals using heat of solution and solubility data
    • DOI 10.1248/cpb.50.263
    • Urakami K et al. A novel method for estimation of transition temperature for polymorphic pairs in pharmaceuticals using heat of solution and solubility data. Chem Pharm Bull (Tokyo) 2002; 50: 263-267. (Pubitemid 41694591)
    • (2002) Chemical and Pharmaceutical Bulletin , vol.50 , Issue.2 , pp. 263-267
    • Urakami, K.1    Shono, Y.2    Higashi, A.3    Umemoto, K.4    Godo, M.5
  • 40
    • 62849110155 scopus 로고    scopus 로고
    • Solvent-mediated solid phase transformations of carbamazepine: Effects of simulated intestinal fluid and fasted state simulated intestinal fluid
    • Lehto P et al. Solvent-mediated solid phase transformations of carbamazepine: effects of simulated intestinal fluid and fasted state simulated intestinal fluid. J Pharm Sci 2009; 98: 985-996.
    • (2009) J Pharm Sci , vol.98 , pp. 985-996
    • Lehto, P.1
  • 41
    • 0026499481 scopus 로고
    • Determination of association constants in cyclodextrin/drug complexation using the Scatchard plot: Application to beta-cyclodextrin- anilinonaphthalenesulfonates
    • Sideris EE et al. Determination of association constants in cyclodextrin/drug complexation using the Scatchard plot: application to beta-cyclodextrin-anilinonaphthalenesulfonates. Pharm Res 1992; 9: 1568-1574.
    • (1992) Pharm Res , vol.9 , pp. 1568-1574
    • Sideris, E.E.1
  • 42
    • 0003347739 scopus 로고
    • Disperse systems. Surfactant properties in solutions and micelle formulation
    • 18th edn. Easton, Pennsylvania: Mack Publishing Company, 18042
    • Zografi G et al. Disperse systems. Surfactant properties in solutions and micelle formulation. Remington's Pharmaceutical Sciences, 18th edn. Easton, Pennsylvania: Mack Publishing Company, 18042, 1990: 257-309.
    • (1990) Remington's Pharmaceutical Sciences , pp. 257-309
    • Zografi, G.1
  • 43
    • 33744544180 scopus 로고
    • Fractal reaction-kinetics
    • Kopelman R. Fractal reaction-kinetics. Science 1988; 241: 1620-1626.
    • (1988) Science , vol.241 , pp. 1620-1626
    • Kopelman, R.1
  • 44
    • 0034058121 scopus 로고    scopus 로고
    • On the heterogeneity of drug dissolution and release
    • DOI 10.1023/A:1007596709657
    • Macheras P, Dokoumetzidis A. On the heterogeneity of drug dissolution and release. Pharm Res 2000; 17: 108-112. (Pubitemid 30158357)
    • (2000) Pharmaceutical Research , vol.17 , Issue.2 , pp. 108-112
    • Macheras, P.1    Dokoumetzidis, A.2


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.