-
1
-
-
0036285999
-
Hydrophobic ion pairing of isoniazid using a prodrug approach
-
DOI 10.1002/jps.10116
-
Zhou H et al. Hydrophobic ion pairing of isoniazid using a prodrug approach. J Pharm 2002; 91: 1502-1511. (Pubitemid 34633965)
-
(2002)
Journal of Pharmaceutical Sciences
, vol.91
, Issue.6
, pp. 1502-1511
-
-
Zhou, H.1
Lengsfeld, C.2
Claffey, D.J.3
Ruth, J.A.4
Hybertson, B.5
Randolph, T.W.6
Ng, K.-Y.7
Manning, M.C.8
-
2
-
-
37849045222
-
Dissolution improvement of four poorly water soluble drugs by cogrinding with commonly used excipients
-
Vogt M et al. Dissolution improvement of four poorly water soluble drugs by cogrinding with commonly used excipients. Eur J Pharm Biopharm 2008; 68: 330-337.
-
(2008)
Eur J Pharm Biopharm
, vol.68
, pp. 330-337
-
-
Vogt, M.1
-
3
-
-
41549150839
-
Formulation and characterization of ternary solid dispersions made up of Itraconazole and two excipients, TPGS 1000 and PVPVA 64, that were selected based on a supersaturation screening study
-
Janssens S et al. Formulation and characterization of ternary solid dispersions made up of Itraconazole and two excipients, TPGS 1000 and PVPVA 64, that were selected based on a supersaturation screening study. Eur J Pharm Biopharm 2008; 69: 158-166.
-
(2008)
Eur J Pharm Biopharm
, vol.69
, pp. 158-166
-
-
Janssens, S.1
-
4
-
-
52949150391
-
Effect of polymer type on the dissolution profile of amorphous solid dispersions containing felodipine
-
Konno H et al. Effect of polymer type on the dissolution profile of amorphous solid dispersions containing felodipine. Eur J Pharm Biopharm 2008; 70: 493-499.
-
(2008)
Eur J Pharm Biopharm
, vol.70
, pp. 493-499
-
-
Konno, H.1
-
5
-
-
53849129520
-
Dissolution improvement and the mechanism of the improvement from cocrystallization of poorly water-soluble compounds
-
Shiraki K et al. Dissolution improvement and the mechanism of the improvement from cocrystallization of poorly water-soluble compounds. Pharm Res 2008; 25: 2581-2592.
-
(2008)
Pharm Res
, vol.25
, pp. 2581-2592
-
-
Shiraki, K.1
-
6
-
-
85047686260
-
Cefuroxime axetil solid dispersion with polyglycolized glycerides for improved stability and bioavailability
-
Dhumal RS et al. Cefuroxime axetil solid dispersion with polyglycolized glycerides for improved stability and bioavailability. J Pharm Pharmacol 2009; 61: 743-751.
-
(2009)
J Pharm Pharmacol
, vol.61
, pp. 743-751
-
-
Dhumal, R.S.1
-
7
-
-
0036771080
-
Physicochemical characterization of solid dispersions of carbamazepine formulated by supercritical carbon dioxide and conventional solvent evaporation method
-
DOI 10.1002/jps.10186
-
Sethia S, Squillante E. Physicochemical characterization of solid dispersions of carbamazepine formulated by supercritical carbon dioxide and conventional solvent evaporation methods. J Pharm Sci 2002; 91: 1948-1957. (Pubitemid 36254931)
-
(2002)
Journal of Pharmaceutical Sciences
, vol.91
, Issue.9
, pp. 1948-1957
-
-
Sethia, S.1
Squillante, E.2
-
8
-
-
1442348833
-
Solid dispersion of carbamazepine in PVP K30 by conventional solvent evaporation and supercritical methods
-
DOI 10.1016/j.ijpharm.2003.11.025, PII S037851730300629X
-
Sethia S, Squillante E. Solid dispersion of carbamazepine in PVP K30 by conventional solvent evaporation and supercritical methods. Int J Pharm 2004; 272: 1-10. (Pubitemid 38293005)
-
(2004)
International Journal of Pharmaceutics
, vol.272
, Issue.1-2
, pp. 1-10
-
-
Sethia, S.1
Squillante, E.2
-
9
-
-
0034607429
-
Membrane penetration enhancement of ibuprofen using supersaturation
-
DOI 10.1016/S0378-5173(00)00346-X, PII S037851730000346X
-
Iervolino M et al. Membrane penetration enhancement of ibuprofen using supersaturation. Int J Pharm 2000; 198: 229-238. (Pubitemid 30184859)
-
(2000)
International Journal of Pharmaceutics
, vol.198
, Issue.2
, pp. 229-238
-
-
Iervolino, M.1
Raghavan, S.L.2
Hadgraft, J.3
-
10
-
-
0036245046
-
Study of the complexation behavior of tenoxicam with cyclodextrins in solution: Improved solubility and percutaneous permeability
-
DOI 10.1081/DDC-120002840
-
Larrucea E et al. Study of the complexation behavior of tenoxicam with cyclodextrins in solution: improved solubility and percutaneous permeability. Drug Dev Ind Pharm 2002; 28: 245-252. (Pubitemid 34475671)
-
(2002)
Drug Development and Industrial Pharmacy
, vol.28
, Issue.3
, pp. 245-252
-
-
Larrucea, E.1
Arellano, A.2
Santoyo, S.3
Ygartua, P.4
-
11
-
-
0037965572
-
Processing of nimesulide-PEG 400-PG-PVP solid dispersions: Preparation, characterization, and in vitro dissolution
-
DOI 10.1081/DDC-120018203
-
Gohel MC, Patel LD. Processing of nimesulide-PEG 400-PGPVP solid dispersions: preparation, characterization, and in vitro dissolution. Drug Dev Ind Pharm 2003; 29: 299-310. (Pubitemid 36528620)
-
(2003)
Drug Development and Industrial Pharmacy
, vol.29
, Issue.3
, pp. 299-310
-
-
Gohel, M.C.1
Patel, L.D.2
-
12
-
-
33747375906
-
The effects of surfactants on the dissolution profiles of poorly water-soluble acidic drugs
-
Park SH, Choi HK. The effects of surfactants on the dissolution profiles of poorly water-soluble acidic drugs. Int J Pharm 2006; 321: 35-41.
-
(2006)
Int J Pharm
, vol.321
, pp. 35-41
-
-
Park, S.H.1
Choi, H.K.2
-
13
-
-
33745377516
-
Canine intestinal contents vs. simulated media for the assessment of solubility of two weak bases in the human small intestinal contents
-
DOI 10.1007/s11095-006-0207-8
-
Kalantzi L et al. Canine intestinal contents vs. simulated media for the assessment of solubility of two weak bases in the human small intestinal contents. Pharm Res 2006; 23: 1373-1381. (Pubitemid 43946159)
-
(2006)
Pharmaceutical Research
, vol.23
, Issue.6
, pp. 1373-1381
-
-
Kalantzi, L.1
Persson, E.2
Polentarutti, B.3
Abrahamsson, B.4
Goumas, K.5
Dressman, J.B.6
Reppas, C.7
-
14
-
-
34247612824
-
In vitro behavior of a phosphate ester prodrug of amprenavir in human intestinal fluids and in the Caco-2 system: Illustration of intraluminal supersaturation
-
DOI 10.1016/j.ijpharm.2006.12.011, PII S0378517306010696
-
Brouwers J et al. In vitro behavior of a phosphate ester prodrug of amprenavir in human intestinal fluids and in the Caco-2 system: illustration of intraluminal supersaturation. Int J Pharm 2007; 336: 302-309. (Pubitemid 46670658)
-
(2007)
International Journal of Pharmaceutics
, vol.336
, Issue.2
, pp. 302-309
-
-
Brouwers, J.1
Tack, J.2
Augustijns, P.3
-
15
-
-
34548082187
-
Parallel monitoring of plasma and intraluminal drug concentrations in man after oral administration of fosamprenavir in the fasted and fed state
-
DOI 10.1007/s11095-007-9307-3
-
Brouwers J et al. Parallel monitoring of plasma and intraluminal drug concentrations in man after oral administration of fosamprenavir in the fasted and fed state. Pharm Res 2007; 24: 1862-1869. (Pubitemid 47389240)
-
(2007)
Pharmaceutical Research
, vol.24
, Issue.10
, pp. 1862-1869
-
-
Brouwers, J.1
Tack, J.2
Augustijns, P.3
-
16
-
-
67349204296
-
Postprandial changes in solubilizing capacity of human intestinal fluids for BCS class II drugs
-
Clarysse S et al. Postprandial changes in solubilizing capacity of human intestinal fluids for BCS class II drugs. Pharm Res 2009; 26: 1456-1466.
-
(2009)
Pharm Res
, vol.26
, pp. 1456-1466
-
-
Clarysse, S.1
-
17
-
-
0034601240
-
Improving drug solubility for oral delivery using solid dispersions
-
DOI 10.1016/S0939-6411(00)00076-X, PII S093964110000076X
-
Leuner C, Dressman J. Improving drug solubility for oral delivery using solid dispersions. Eur J Pharm Biopharm 2000; 50: 47-60. (Pubitemid 30326688)
-
(2000)
European Journal of Pharmaceutics and Biopharmaceutics
, vol.50
, Issue.1
, pp. 47-60
-
-
Leuner, C.1
Dressman, J.2
-
18
-
-
1142303337
-
What is the true solubility advantage for amorphous pharmaceuticals?
-
DOI 10.1023/A:1007516718048
-
Hancock B, Parks M. What is the true solubility advantage for amorphous pharmaceuticals? Pharm Res 2001; 17: 397-404. (Pubitemid 30395293)
-
(2000)
Pharmaceutical Research
, vol.17
, Issue.4
, pp. 397-404
-
-
Hancock, B.C.1
Parks, M.2
-
19
-
-
21644446038
-
Development and characterization of a scalable controlled precipitation process to enhance the dissolution of poorly water-soluble drugs
-
DOI 10.1023/B:PHAM.0000048196.61887.e5
-
Rogers TL et al. Development and characterization of a scalable controlled precipitation process to enhance the dissolution of poorly water-soluble drugs. Pharm Res 2004; 21: 2048-2057. (Pubitemid 40941225)
-
(2004)
Pharmaceutical Research
, vol.21
, Issue.11
, pp. 2048-2057
-
-
Rogers, T.L.1
Gillespie, I.B.2
Hitt, J.E.3
Fransen, K.L.4
Crowl, C.A.5
Tucker, C.J.6
Kupperblatt, G.B.7
Becker, J.N.8
Wilson, D.L.9
Todd, C.10
Broomall, C.F.11
Evans, J.C.12
Elder, E.J.13
-
20
-
-
0033986929
-
Effect of cellulose polymers on supersaturation and in vitro membrane transport of hydrocortisone acetate
-
DOI 10.1016/S0378-5173(99)00345-2, PII S0378517399003452
-
Raghavan SL et al. Effect of cellulose polymers on supersaturation and in vitro membrane transport of hydrocortisone acetate. Int J Pharm 2000; 193: 231-237. (Pubitemid 30001867)
-
(2000)
International Journal of Pharmaceutics
, vol.193
, Issue.2
, pp. 231-237
-
-
Raghavan, S.L.1
Trividic, A.2
Davis, A.F.3
Hadgraft, J.4
-
22
-
-
33646689478
-
Structural relaxation of acetaminophen glass
-
Gunawan LG et al. Structural relaxation of acetaminophen glass. Pharm Res 2006; 23: 967-979.
-
(2006)
Pharm Res
, vol.23
, pp. 967-979
-
-
Gunawan, L.G.1
-
23
-
-
0017178826
-
Dissolution behavior and bioavailability of phenytoin from a ground mixture with microcrystalline cellulose
-
Yamamoto K et al. Dissolution behavior and bioavailability of phenytoin from a ground mixture with microcrystalline cellulose. J Pharm Sci 1976; 65: 1484-1488.
-
(1976)
J Pharm Sci
, vol.65
, pp. 1484-1488
-
-
Yamamoto, K.1
-
24
-
-
0025830658
-
Dissolution and bioavailability of phenobarbital in solid dispersion with phosphatidylcholine
-
Fujii M et al. Dissolution and bioavailability of phenobarbital in solid dispersion with phosphatidylcholine. Chem Pharm Bull 1991; 39: 1886-1888.
-
(1991)
Chem Pharm Bull
, vol.39
, pp. 1886-1888
-
-
Fujii, M.1
-
25
-
-
0031958399
-
Influence of water-soluble polymers on the dissolution of Nifedipine solid dispersions with combined carriers
-
Suzki H, Sunada H. Influence of water-soluble polymers on the dissolution of nifedipine solid dispersions with combined carriers. Chem Pharm Bull 1998; 46: 482-487. (Pubitemid 28188567)
-
(1998)
Chemical and Pharmaceutical Bulletin
, vol.46
, Issue.3
, pp. 482-487
-
-
Suzuki, H.1
Sunada, H.2
-
26
-
-
33644881395
-
Stabilization of solid dispersions of nimodipine and polyethylene glycol 2000
-
Urbanetz NA. Stabilization of solid dispersions of nimodipine and polyethylene glycol 2000. Eur J Pharm Sci 2006; 28: 67-76.
-
(2006)
Eur J Pharm Sci
, vol.28
, pp. 67-76
-
-
Urbanetz, N.A.1
-
29
-
-
41349116109
-
Development of a reaction-limited model of dissolution: Application to official dissolution tests experiments
-
Dokoumetzidis A et al. Development of a reaction-limited model of dissolution: Application to official dissolution tests experiments. Int J Pharm 2008; 355: 114-125.
-
(2008)
Int J Pharm
, vol.355
, pp. 114-125
-
-
Dokoumetzidis, A.1
-
30
-
-
67650569218
-
A simulation of oral absorption using classical nucleation theory
-
Sugano K. A simulation of oral absorption using classical nucleation theory. Int J Pharm 2009; 378: 142-145.
-
(2009)
Int J Pharm
, vol.378
, pp. 142-145
-
-
Sugano, K.1
-
31
-
-
72449149167
-
Computational oral absorption simulation for low-solubility compounds
-
Sugano K. Computational oral absorption simulation for low-solubility compounds. Chem Biodivers 2009; 6: 2014-2029.
-
(2009)
Chem Biodivers
, vol.6
, pp. 2014-2029
-
-
Sugano, K.1
-
32
-
-
0033988596
-
Physicochemical properties and bioavailability of carbamazepine polymorphs and dihydrate
-
DOI 10.1016/S0378-5173(99)00315-4, PII S0378517399003154
-
Kobayashi Y et al. Physicochemical properties and bioavailability of carbamazepine polymorphs and dihydrate. Int J Pharm 2000; 193: 137-146. (Pubitemid 30001856)
-
(2000)
International Journal of Pharmaceutics
, vol.193
, Issue.2
, pp. 137-146
-
-
Kobayashi, Y.1
Ito, S.2
Itai, S.3
Yamamoto, K.4
-
33
-
-
33947500641
-
Influence of polymorphic form, morphology, and excipient interactions on the dissolution of carbamazepine compacts
-
DOI 10.1002/jps.20756
-
Tian F et al. Influence of polymorphic form, morphology, and excipient interactions on the dissolution of carbamazepine compacts. J Pharm Sci 2007; 96: 584-594. (Pubitemid 46466080)
-
(2007)
Journal of Pharmaceutical Sciences
, vol.96
, Issue.3
, pp. 584-594
-
-
Tian, F.1
Sandler, N.2
Aaltonen, J.3
Lang, C.4
Saville, D.J.5
Gordon, K.C.6
Strachan, C.J.7
Rantanen, J.8
Rades, T.9
-
34
-
-
0025880233
-
Improvement of cyclosporin absorption in children after liver transplantation by means of water-soluble vitamin E
-
Sokol RJ et al. Improvement of cyclosporin absorption in children after liver transplantation by means of water-soluble vitamin E. Lancet 1991; 338: 212-214.
-
(1991)
Lancet
, vol.338
, pp. 212-214
-
-
Sokol, R.J.1
-
36
-
-
33747373878
-
A century of dissolution research: From Noyes and Whitney to the Biopharmaceutics Classification System
-
DOI 10.1016/j.ijpharm.2006.07.011, PII S0378517306005813
-
Dokoumetzidis A, Macheras P. A century of dissolution research: From Noyes and Whitney to the Biopharmaceutics Classification System. Int J Pharm 2006; 321: 1-11. (Pubitemid 44247428)
-
(2006)
International Journal of Pharmaceutics
, vol.321
, Issue.1-2
, pp. 1-11
-
-
Dokoumetzidis, A.1
Macheras, P.2
-
37
-
-
0005491022
-
A statistical rate theory study of interface concentration during crystal growth or dissolution
-
Dejmek M, Ward CA. A statistical rate theory study of interface concentration during crystal growth or dissolution. J Chem Phys 1998; 108: 8698-8704. (Pubitemid 128597379)
-
(1998)
Journal of Chemical Physics
, vol.108
, Issue.20
, pp. 8698-8704
-
-
Dejmek, M.1
Ward, C.A.2
-
39
-
-
0036482959
-
A novel method for estimation of transition temperature for polymorphic pairs in pharmaceuticals using heat of solution and solubility data
-
DOI 10.1248/cpb.50.263
-
Urakami K et al. A novel method for estimation of transition temperature for polymorphic pairs in pharmaceuticals using heat of solution and solubility data. Chem Pharm Bull (Tokyo) 2002; 50: 263-267. (Pubitemid 41694591)
-
(2002)
Chemical and Pharmaceutical Bulletin
, vol.50
, Issue.2
, pp. 263-267
-
-
Urakami, K.1
Shono, Y.2
Higashi, A.3
Umemoto, K.4
Godo, M.5
-
40
-
-
62849110155
-
Solvent-mediated solid phase transformations of carbamazepine: Effects of simulated intestinal fluid and fasted state simulated intestinal fluid
-
Lehto P et al. Solvent-mediated solid phase transformations of carbamazepine: effects of simulated intestinal fluid and fasted state simulated intestinal fluid. J Pharm Sci 2009; 98: 985-996.
-
(2009)
J Pharm Sci
, vol.98
, pp. 985-996
-
-
Lehto, P.1
-
41
-
-
0026499481
-
Determination of association constants in cyclodextrin/drug complexation using the Scatchard plot: Application to beta-cyclodextrin- anilinonaphthalenesulfonates
-
Sideris EE et al. Determination of association constants in cyclodextrin/drug complexation using the Scatchard plot: application to beta-cyclodextrin-anilinonaphthalenesulfonates. Pharm Res 1992; 9: 1568-1574.
-
(1992)
Pharm Res
, vol.9
, pp. 1568-1574
-
-
Sideris, E.E.1
-
42
-
-
0003347739
-
Disperse systems. Surfactant properties in solutions and micelle formulation
-
18th edn. Easton, Pennsylvania: Mack Publishing Company, 18042
-
Zografi G et al. Disperse systems. Surfactant properties in solutions and micelle formulation. Remington's Pharmaceutical Sciences, 18th edn. Easton, Pennsylvania: Mack Publishing Company, 18042, 1990: 257-309.
-
(1990)
Remington's Pharmaceutical Sciences
, pp. 257-309
-
-
Zografi, G.1
-
43
-
-
33744544180
-
Fractal reaction-kinetics
-
Kopelman R. Fractal reaction-kinetics. Science 1988; 241: 1620-1626.
-
(1988)
Science
, vol.241
, pp. 1620-1626
-
-
Kopelman, R.1
-
44
-
-
0034058121
-
On the heterogeneity of drug dissolution and release
-
DOI 10.1023/A:1007596709657
-
Macheras P, Dokoumetzidis A. On the heterogeneity of drug dissolution and release. Pharm Res 2000; 17: 108-112. (Pubitemid 30158357)
-
(2000)
Pharmaceutical Research
, vol.17
, Issue.2
, pp. 108-112
-
-
Macheras, P.1
Dokoumetzidis, A.2
-
45
-
-
29244445764
-
The effects of food on the dissolution of poorly soluble drugs in human and in model small intestinal fluids
-
DOI 10.1007/s11095-005-8192-x
-
Persson EM et al. The effects of food on the dissolution of poorly soluble drugs in human and in model small intestinal fluids. Pharm Res 2005; 22: 2141-2151. (Pubitemid 41821594)
-
(2005)
Pharmaceutical Research
, vol.22
, Issue.12
, pp. 2141-2151
-
-
Persson, E.M.1
Gustafsson, A.-S.2
Carlsson, A.S.3
Nilsson, R.G.4
Knutson, L.5
Forsell, P.6
Hanisch, G.7
Lennernas, H.8
Abrahamsson, B.9
|