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Journal of Biological Inorganic Chemistry

Volumn 16, Issue 1, 2011, Pages 137-155

Synthesis and biological evaluation of new [Tc(N)(PS)]-based mixed-ligand compounds useful in the design of target-specific radiopharmaceuticals: The 2-methoxyphenylpiperazine dithiocarbamate derivatives as an example

(8) Bolzati, Cristina a,b Salvarese, Nicola b Carta, Davide b Refosco, Fiorenzo a Dolmella, Alessandro b Pietzsch, Hans Jürgen c Bergmann, Ralf c Bandoli, Giuliano b

a CNR (Italy)

b UNIVERSITY OF PADOVA (Italy)

c INSTITUTE OF ION BEAM PHYSICS AND MATERIALS RESEARCH (Germany)

Author keywords

5HT1A receptor; Brain; Dithiocarbamate; Phosphinothiolate; Technetium

Indexed keywords

2 METHOXYPHENYLPIPERAZINE DITHIOCARBAMATE DERIVATIVE; CYSTEINE; DITHIOCARBAMIC ACID; DITHIOCARBAMIC ACID DERIVATIVE; GLUTATHIONE; SEROTONIN 1A RECEPTOR; TECHNETIUM 99M; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ARTICLE; BINDING AFFINITY; BIOTRANSFORMATION; CHEMICAL ANALYSIS; CHEMICAL REACTION; CHEMICAL STRUCTURE; CONTROLLED STUDY; FEMALE; IC 50; LIPOPHILICITY; NONHUMAN; PH; PHARMACOPHORE; PRIORITY JOURNAL; RAT; RECEPTOR BINDING; ROOM TEMPERATURE; SYNTHESIS;

ANIMALS; DRUG DESIGN; LIGANDS; MOLECULAR STRUCTURE; ORGANOTECHNETIUM COMPOUNDS; PIPERAZINES; RADIOPHARMACEUTICALS; RATS; RECEPTOR, SEROTONIN, 5-HT1A; SULFHYDRYL COMPOUNDS; TECHNETIUM; THIOCARBAMATES; TISSUE DISTRIBUTION;

EID: 79951549586 PISSN: 09498257 EISSN: None Source Type: Journal
DOI: 10.1007/s00775-010-0712-4 Document Type: Article

Times cited : (14)

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