Fluoro analogs of WAY-100635 with varying pharmacokinetics properties

Nuclear Medicine and Biology

Volumn 27, Issue 5, 2000, Pages 457-462

  Lang, Lixin ^a   Jagoda, Elaine ^a   Schmall, Bernard ^a   Sassaman, Mark ^a   Ma, Ying ^a   Eckelman, William C ^a  

^a NATIONAL INSTITUTES OF HEALTH   (United States)

Author keywords

5 HT(1A) subtype; FCWAY; Fluorine 18; MeFBWAY; Serotonin receptor

Indexed keywords

CARBANILAMIDE DERIVATIVE; CYCLOHEXANECARBOXYLIC ACID DERIVATIVE; FLUORINE 18; N [2 [4 (2 METHOXYPHENYL) 1 PIPERAZINYL]ETHYL] N (2 PYRIDYL)CYCLOHEXANECARBOXAMIDE; RADIOLIGAND; RECEPTOR SUBTYPE; SEROTONIN 1A RECEPTOR;

CHEMICAL ANALYSIS; CHEMICAL STRUCTURE; FLUORINATION; HUMAN; IN VIVO STUDY; ISOTOPE LABELING; PHARMACOKINETICS; POSITRON EMISSION TOMOGRAPHY; RECEPTOR BINDING; RECEPTOR SENSITIVITY; REVIEW; STOICHIOMETRY; STRUCTURE ACTIVITY RELATION;

EID: 0033827025     PISSN: 09698051     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0969-8051(00)00111-6     Document Type: Article

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