Differential effects of two major neurosteroids on cerebellar and cortical GABAA receptor binding and function

European Journal of Pharmacology

Volumn 650, Issue 1, 2011, Pages 94-101

  Maksay, Gábor ^a   Fodor, László ^b  

^a INSTITUTE OF EXPERIMENTAL MEDICINE   (Hungary)

^b GEDEON RICHTER LTD   (Hungary)

Author keywords

6 GABAA receptor; 6KO mouse; 5 THDOC; 3H EBOB binding; Allopregnanolone; Gaboxadol

Indexed keywords

3ALPHA HYDROXY 5ALPHA PREGNAN 20 ONE; 3ALPHA,21 DIHYDROXY 5ALPHA PREGNAN 20 ONE; 4 AMINOBUTYRIC ACID A RECEPTOR; 4 AMINOBUTYRIC ACID A RECEPTOR ALPHA6; 4 AMINOBUTYRIC ACID A RECEPTOR DELTA; 4 AMINOBUTYRIC ACID RECEPTOR STIMULATING AGENT; 5ALPHA TETRAHYDRODEOXYCORTICOSTERONE; 5BETA PREGNAN 3ALPHA,21 DIOL 20 ONE; CHLORIDE; ETHYNYLBICYCLOORTHOBENZOATE; FUROSEMIDE; GABOXADOL; MINERALOCORTICOID; UNCLASSIFIED DRUG;

ANIMAL CELL; ANIMAL TISSUE; ARTICLE; BINDING AFFINITY; BRAIN CORTEX; BRAIN TISSUE; CEREBELLUM; CHLORIDE CURRENT; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG RECEPTOR BINDING; GRANULE CELL; INCUBATION TIME; MALE; MOUSE; NONHUMAN; PRIORITY JOURNAL; PROTEIN FUNCTION; RAT; RECEPTOR OCCUPANCY; WILD TYPE;

ANIMALS; BICYCLO COMPOUNDS, HETEROCYCLIC; CEREBELLUM; CEREBRAL CORTEX; DESOXYCORTICOSTERONE; DOSE-RESPONSE RELATIONSHIP, DRUG; DRUG SYNERGISM; FUROSEMIDE; GABA-A RECEPTOR AGONISTS; GENE KNOCKOUT TECHNIQUES; MALE; MICE; NEUROTRANSMITTER AGENTS; PREGNANOLONE; PROTEIN BINDING; RATS; RECEPTORS, GABA-A;

EID: 78649737740     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.ejphar.2010.10.003     Document Type: Article

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