-
3
-
-
34848848499
-
-
K. Müller, C. Faeh, F. Diederich, Science 2007, 317, 1881 - 1886.
-
(2007)
Science
, vol.317
, pp. 1881-1886
-
-
Müller, K.1
Faeh, C.2
Diederich, F.3
-
7
-
-
62949236412
-
-
M. S. Wiehn, S. D. Lindell, S. Bräse, Angew. Chem. 2008, 120, 8240 - 8242
-
(2008)
Angew. Chem.
, vol.120
, pp. 8240-8242
-
-
Wiehn, M.S.1
Lindell, S.D.2
Bräse, S.3
-
8
-
-
54049122258
-
-
Angew. Chem. Int. Ed. 2008, 47, 8120 - 8122
-
(2008)
Angew. Chem. Int. Ed.
, vol.47
, pp. 8120-8122
-
-
-
10
-
-
33747265243
-
-
G. K. Prakash, R. Mogi, G. A. Olah, Org. Lett. 2006, 8, 3589 - 3592
-
(2006)
Org. Lett.
, vol.8
, pp. 3589-3592
-
-
Prakash, G.K.1
Mogi, R.2
Olah, G.A.3
-
11
-
-
55049117569
-
-
V. V. Levin, A. D. Dilman, P. A. Belyakov, M. I. Struchkova, V. A. Tartakovsky, Eur. J. Org. Chem. 2008, 31, 5226 - 5230
-
(2008)
Eur. J. Org. Chem.
, vol.31
, pp. 5226-5230
-
-
Levin, V.V.1
Dilman, A.D.2
Belyakov, P.A.3
Struchkova, M.I.4
Tartakovsky, V.A.5
-
12
-
-
37249001484
-
-
N. V. Kirij, L. A. Babadzhanova, V. N. Movchun, Y. L. Yagupolskii, W. Tyrra, D. Naumann, H. T. M. Fischer, H. Scherer, J. Fluorine Chem. 2008, 129, 14 - 21
-
(2008)
J. Fluorine Chem.
, vol.129
, pp. 14-21
-
-
Kirij, N.V.1
Babadzhanova, L.A.2
Movchun, V.N.3
Yagupolskii, Y.L.4
Tyrra, W.5
Naumann, D.6
Fischer, H.T.M.7
Scherer, H.8
-
13
-
-
35548947177
-
-
A. D. Dilman, D. E. Arkhipov, V. V. Levin, P. A. Belyakov, A. A. Korlyukov, M. I. Struchkova, V. A. Tartakovsky, J. Org. Chem. 2007, 72, 8604 - 8607
-
(2007)
J. Org. Chem.
, vol.72
, pp. 8604-8607
-
-
Dilman, A.D.1
Arkhipov, D.E.2
Levin, V.V.3
Belyakov, P.A.4
Korlyukov, A.A.5
Struchkova, M.I.6
Tartakovsky, V.A.7
-
14
-
-
0035917368
-
-
D. W. Nelson, J. Owens, D. Hiraldo, J. Org. Chem. 2001, 66, 2572 - 2582.
-
(2001)
J. Org. Chem.
, vol.66
, pp. 2572-2582
-
-
Nelson, D.W.1
Owens, J.2
Hiraldo, D.3
-
16
-
-
0036969976
-
-
Y. Gong, K. Kato, H. Kimoto, Bull. Chem. Soc. Jpn. 2002, 75, 2637 - 2645.
-
(2002)
Bull. Chem. Soc. Jpn.
, vol.75
, pp. 2637-2645
-
-
Gong, Y.1
Kato, K.2
Kimoto, H.3
-
17
-
-
0035035271
-
-
B. Crousse, S. Narizuka, D. Bonnet-Delpon, J.-P. Bégué, Synlett 2001, 679 - 681.
-
(2001)
Synlett
, pp. 679-681
-
-
Crousse, B.1
Narizuka, S.2
Bonnet-Delpon, D.3
Bégué, J.-P.4
-
18
-
-
10744227548
-
-
A. Volonterio, S. Bellosta, F. Bravin, M. C. Bellucci, L. Bruche, G. Colombo, L. Malpezzi, S. Mazzini, S. V. Meille, M. Meli, C. Ramirez de Arellano, M. Zanda, Chem. Eur. J. 2003, 9, 4510 - 4522
-
(2003)
Chem. Eur. J.
, vol.9
, pp. 4510-4522
-
-
Volonterio, A.1
Bellosta, S.2
Bravin, F.3
Bellucci, M.C.4
Bruche, L.5
Colombo, G.6
Malpezzi, L.7
Mazzini, S.8
Meille, S.V.9
Meli, M.10
De Arellano, C.R.11
Zanda, M.12
-
19
-
-
0034729603
-
-
1833. For some recent examples of fluorine-containing peptidomimetics
-
A. Volonterio, P. Bravo, M. Zanda, Org. Lett. 2000, 2, 1827 - 1833. For some recent examples of fluorine-containing peptidomimetics
-
(2000)
Org. Lett.
, vol.2
, pp. 1827
-
-
Volonterio, A.1
Bravo, P.2
Zanda, M.3
-
20
-
-
0033535071
-
-
G. S. Garrett, S. J. McPhail, K. Tornheim, P. E. Correa, J. M. McIver, Bioorg. Med. Chem. Lett. 1999, 9, 301 - 306
-
(1999)
Bioorg. Med. Chem. Lett.
, vol.9
, pp. 301-306
-
-
Garrett, G.S.1
McPhail, S.J.2
Tornheim, K.3
Correa, P.E.4
McIver, J.M.5
-
21
-
-
0033582779
-
-
M.-A. Poupart, G. Fazal, S. Goulet, L.-T. Mar, J. Org. Chem. 1999, 64, 1356 - 1361
-
(1999)
J. Org. Chem.
, vol.64
, pp. 1356-1361
-
-
Poupart, M.-A.1
Fazal, G.2
Goulet, S.3
Mar, L.-T.4
-
22
-
-
17144462307
-
-
924, and references cited therein
-
M. Eda, A. Ashimori, F. Akahoshi, T. Yoshimura, Y. Inoue, C. Fukaya, M. Nakajima, H. Fukuyama, T. Imada, N. Nakamura, Bioorg. Med. Chem. Lett. 1998, 8, 919 - 924, and references cited therein
-
(1998)
Bioorg. Med. Chem. Lett.
, vol.8
, pp. 919
-
-
Eda, M.1
Ashimori, A.2
Akahoshi, F.3
Yoshimura, T.4
Inoue, Y.5
Fukaya, C.6
Nakajima, M.7
Fukuyama, H.8
Imada, T.9
Nakamura, N.10
-
25
-
-
0027968473
-
-
L. G. Boros, B. Decorte, R. H. Gimi, J. T. Welch, Y. Wu, R. E. Handschumacher, Tetrahedron Lett. 1994, 35, 6033 - 6036
-
(1994)
Tetrahedron Lett.
, vol.35
, pp. 6033-6036
-
-
Boros, L.G.1
Decorte, B.2
Gimi, R.H.3
Welch, J.T.4
Wu, Y.5
Handschumacher, R.E.6
-
26
-
-
0027946242
-
-
L. Revesz, C. Briswalter, R. Heng, A. Leutwiler, R. Mueller, H.-J. Wuethrich, Tetrahedron Lett. 1994, 35, 9693 - 9696
-
(1994)
Tetrahedron Lett.
, vol.35
, pp. 9693-9696
-
-
Revesz, L.1
Briswalter, C.2
Heng, R.3
Leutwiler, A.4
Mueller, R.5
Wuethrich, H.-J.6
-
28
-
-
38749144762
-
-
J. Y. Gauthier, N. Chauret, W. Cromlish, S. Desmarais, L. T. Duong, J.-P. Falgueyret, D. B. Kimmel, S. Lamontagne, S. Léger, T. LeRiche, C. S. Li, F. Massé, D. J. McKay, D. A. Nicoll-Griffith, R. M. Oballa, J. T. Palmer, M. D. Percival, D. Riendeau, J. Robichaud, G. A. Rodan, S. B. Rodan, C. Seto, M. Thérien, V.-L. Truong, M. C. Venuti, G. Wesolowski, R. N. Young, R. Zambonia, W. C. Black, Bioorg. Med. Chem. Lett. 2008, 18, 923 - 928.
-
(2008)
Bioorg. Med. Chem. Lett.
, vol.18
, pp. 923-928
-
-
Gauthier, J.Y.1
Chauret, N.2
Cromlish, W.3
Desmarais, S.4
Duong, L.T.5
Falgueyret, J.-P.6
Kimmel, D.B.7
Lamontagne, S.8
Léger, S.9
Leriche, T.10
Li, C.S.11
Massé, F.12
McKay, D.J.13
Nicoll-Griffith, D.A.14
Oballa, R.M.15
Palmer, J.T.16
Percival, M.D.17
Riendeau, D.18
Robichaud, J.19
Rodan, G.A.20
Rodan, S.B.21
Seto, C.22
Thérien, M.23
Truong, V.-L.24
Venuti, M.C.25
Wesolowski, G.26
Young, R.N.27
Zambonia, R.28
Black, W.C.29
more..
-
30
-
-
78349255229
-
-
Reductive amination
-
Reductive amination
-
-
-
-
32
-
-
13444302540
-
-
F. Gosselin, P. D. O'Shea, S. Roy, R. A. Reamer, C.-Y. Chen, R. P. Volante, Org. Lett. 2005, 7, 355 - 358
-
(2005)
Org. Lett.
, vol.7
, pp. 355-358
-
-
Gosselin, F.1
O'Shea, P.D.2
Roy, S.3
Reamer, R.A.4
Chen, C.-Y.5
Volante, R.P.6
-
33
-
-
53849092219
-
-
G. Hughes, P. N. Devine, J. R. Naber, P. D. O'Shea, B. S. Foster, D. J. McKay, R. P. Volante, Angew. Chem. 2007, 119, 1871 - 1874
-
(2007)
Angew. Chem.
, vol.119
, pp. 1871-1874
-
-
Hughes, G.1
Devine, P.N.2
Naber, J.R.3
O'Shea, P.D.4
Foster, B.S.5
McKay, D.J.6
Volante, R.P.7
-
34
-
-
34249718561
-
-
Angew. Chem. Int. Ed. 2007, 46, 1839 - 1842.
-
(2007)
Angew. Chem. Int. Ed.
, vol.46
, pp. 1839-1842
-
-
-
35
-
-
0033165877
-
-
J.-C. Blazejewski, E. Anselmi, M. P. Wilmshurst, Tetrahedron Lett. 1999, 40, 5475 - 5478.
-
(1999)
Tetrahedron Lett.
, vol.40
, pp. 5475-5478
-
-
Blazejewski, J.-C.1
Anselmi, E.2
Wilmshurst, M.P.3
-
36
-
-
41349118976
-
-
P. V. Khodakovskiy, D. M. Volochnyuk, D. M. Panov, I. I. Pervak, E. V. Zarudnitskii, O. V. Shishkin, A. A. Yurchenko, A. Shivanyuk, A. A. Tolmachev, Synthesis 2008, 6, 948 - 956
-
(2008)
Synthesis
, vol.6
, pp. 948-956
-
-
Khodakovskiy, P.V.1
Volochnyuk, D.M.2
Panov, D.M.3
Pervak, I.I.4
Zarudnitskii, E.V.5
Shishkin, O.V.6
Yurchenko, A.A.7
Shivanyuk, A.8
Tolmachev, A.A.9
-
37
-
-
78349292096
-
-
According to Chemical Abstracts over 270 aryl trifluoro ketones are commercially available.
-
According to Chemical Abstracts over 270 aryl trifluoro ketones are commercially available.
-
-
-
-
38
-
-
53849146708
-
-
For a very useful synthesis of heterocyclic systems, which have a different substitution pattern, see:
-
For a very useful synthesis of heterocyclic systems, which have a different substitution pattern, see:, G.-W. Zhang, L. Wang, J. Nie, J.-A. Ma, Adv. Synth. Catal. 2008, 350, 1457 - 1463.
-
(2008)
Adv. Synth. Catal.
, vol.350
, pp. 1457-1463
-
-
Zhang, G.-W.1
Wang, L.2
Nie, J.3
Ma, J.-A.4
-
39
-
-
0030970293
-
-
For an alternative synthesis, see:
-
For an alternative synthesis, see:, Y. Yokoyama, K. Mochida, Tetrahedron Lett. 1997, 38, 3443 - 3446.
-
(1997)
Tetrahedron Lett.
, vol.38
, pp. 3443-3446
-
-
Yokoyama, Y.1
Mochida, K.2
-
40
-
-
42949168465
-
-
P. Fu, M. L. Snapper, A. H. Hoveyda, J. Am. Chem. Soc. 2008, 130, 5530 - 5541.
-
(2008)
J. Am. Chem. Soc.
, vol.130
, pp. 5530-5541
-
-
Fu, P.1
Snapper, M.L.2
Hoveyda, A.H.3
-
42
-
-
8744273289
-
-
W.-H. Lin, H.-Z. Fu, J. Li, G. Cheng, R. A. Barnes, J. Chin. Pharm. Sci. 2003, 12, 117 - 122
-
(2003)
J. Chin. Pharm. Sci.
, vol.12
, pp. 117-122
-
-
Lin, W.-H.1
Fu, H.-Z.2
Li, J.3
Cheng, G.4
Barnes, R.A.5
-
43
-
-
0023101265
-
-
I. Kitagawa, N. Yoshioka, C. Kamba, M. Yoshikawa, Y. Hamamoto, Chem. Pharm. Bull. 1987, 35, 928 - 931
-
(1987)
Chem. Pharm. Bull.
, vol.35
, pp. 928-931
-
-
Kitagawa, I.1
Yoshioka, N.2
Kamba, C.3
Yoshikawa, M.4
Hamamoto, Y.5
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