Synthesis and biological evaluation of indolyl glyoxylamides as a new class of antileishmanial agents

Bioorganic and Medicinal Chemistry Letters

Volumn 20, Issue 21, 2010, Pages 6191-6194

  Chauhan, Shikha S ^a   Gupta, Leena ^a   Mittal, Monika ^a   Vishwakarma, Preeti ^a   Gupta, Suman ^a   Chauhan, Prem M S ^a  

^a CENTRAL DRUG RESEARCH INSTITUTE   (India)

Author keywords

Antileishmanial; Indolylglyoxylamides; Tetrahydro carboline

Indexed keywords

AMIDE; ANTILEISHMANIAL AGENT; INDOLYL GLYOXYLAMIDE DERIVATIVE; PENTAMIDINE; STIBOGLUCONATE SODIUM; UNCLASSIFIED DRUG;

ANIMAL CELL; ANTIPROTOZOAL ACTIVITY; ARTICLE; BIOLOGICAL ACTIVITY; CONTROLLED STUDY; DRUG CYTOTOXICITY; DRUG IDENTIFICATION; DRUG SCREENING; DRUG STRUCTURE; DRUG SYNTHESIS; IC 50; LEISHMANIA DONOVANI; MACROPHAGE; MOUSE; NONHUMAN; STRUCTURE ACTIVITY RELATION;

ANIMALS; ANTIMONY SODIUM GLUCONATE; ANTIPROTOZOAL AGENTS; CARBOLINES; INDICATORS AND REAGENTS; LEISHMANIA DONOVANI; MACROPHAGES; MAGNETIC RESONANCE SPECTROSCOPY; MASS SPECTROMETRY; MICE; PENTAMIDINE; SPECTROPHOTOMETRY, INFRARED; STRUCTURE-ACTIVITY RELATIONSHIP;

LEISHMANIA DONOVANI;

EID: 77957881130     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2010.08.119     Document Type: Article

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