메뉴 건너뛰기




Volumn 11, Issue 1, 2010, Pages 2-8

Two-step solid lipid extrusion as a process to modify dissolution behavior

Author keywords

Dissolution; Polyethylene glycol; Process variations; Solid lipid extrusion; Triglyceride

Indexed keywords

CHLORAMPHENICOL; LIPID; MACROGOL; TRIACYLGLYCEROL; TRIPALMITIN;

EID: 77950918430     PISSN: None     EISSN: 15309932     Source Type: Journal    
DOI: 10.1208/s12249-010-9395-y     Document Type: Article
Times cited : (16)

References (36)
  • 1
    • 0024603368 scopus 로고
    • In vitro release of cytotoxic agents from ion exchange resins
    • DOI 10.1016/0168-3659(89)90046-1
    • C Jones MA Burtan BN Gray J Hodgkin 1989 In vitro release of cytotoxic agents from ion exchange resins J Control Release 8 251 257 10.1016/0168- 3659(89)90046-1 1:CAS:528:DyaL1MXitlOjtro%3D (Pubitemid 19099003)
    • (1989) Journal of Controlled Release , vol.8 , Issue.3 , pp. 251-257
    • Jones, C.1    Burton, M.A.2    Gray, B.N.3    Hodgkin, J.4
  • 2
    • 84891501536 scopus 로고    scopus 로고
    • Formulation development and in vitro evaluation of membrane-moderated transdermal systems of ampicillin sodium in ethanol: PH 4.7 buffer solvent system
    • 10.1208/pt0801007
    • J Bagyalakshmi RP Vamskrishna R Manavalan TK Ravi PK Manna 2007 Formulation development and in vitro evaluation of membrane-moderated transdermal systems of ampicillin sodium in ethanol: pH 4.7 buffer solvent system AAPS Pharm Sci Tech 8 E1 E6 10.1208/pt0801007
    • (2007) AAPS Pharm Sci Tech , vol.8
    • Bagyalakshmi, J.1    Vamskrishna, R.P.2    Manavalan, R.3    Ravi, T.K.4    Manna, P.K.5
  • 3
    • 68349131767 scopus 로고    scopus 로고
    • Development and characterization of extended release Kollidon® SR mini-matrices
    • 10.1016/j.ejpb.2009.04.006 19406237
    • I Ozguney D Shuwisitkul R Bodmeier 2009 Development and characterization of extended release Kollidon® SR mini-matrices Eur J Pharm Biopharm 73 140 145 10.1016/j.ejpb.2009.04.006 19406237
    • (2009) Eur J Pharm Biopharm , vol.73 , pp. 140-145
    • Ozguney, I.1    Shuwisitkul, D.2    Bodmeier, R.3
  • 4
    • 0016830071 scopus 로고
    • Elementary osmotic pump
    • 10.1002/jps.2600641218 1:CAS:528:DyaE28XmsFahtw%3D%3D 1510
    • F Theeuwes 1975 Elementary osmotic pump J Pharm Sci 64 1987 1999 10.1002/jps.2600641218 1:CAS:528:DyaE28XmsFahtw%3D%3D 1510
    • (1975) J Pharm Sci , vol.64 , pp. 1987-1999
    • Theeuwes, F.1
  • 5
    • 51949107727 scopus 로고    scopus 로고
    • Controlled release solid dosage forms using combinations of (meth)acrylate copolymers
    • 10.1080/10837450802202098 1:CAS:528:DC%2BD1cXhtFaisr3J 18720248
    • D Gallardo D Skalsky P Kleinebudde 2008 Controlled release solid dosage forms using combinations of (meth)acrylate copolymers Pharm Dev Technol 13 413 423 10.1080/10837450802202098 1:CAS:528:DC%2BD1cXhtFaisr3J 18720248
    • (2008) Pharm Dev Technol , vol.13 , pp. 413-423
    • Gallardo, D.1    Skalsky, D.2    Kleinebudde, P.3
  • 7
    • 0019518548 scopus 로고
    • Solid colloidal drug delivery systems: Nanoparticles
    • DOI 10.1016/0378-5173(81)90100-9
    • RC Oppenheim 1981 Solid colloidal drug delivery systems: nanoparticles Int J Pharm 8 217 234 10.1016/0378-5173(81)90100-9 1:CAS:528:DyaL3MXks1Orsbg%3D (Pubitemid 11043798)
    • (1981) International Journal of Pharmaceutics , vol.8 , Issue.3 , pp. 217-234
    • Oppenheim, R.C.1
  • 8
    • 0014789067 scopus 로고
    • Controlled drug release through polymeric films
    • 10.1002/jps.2600590507 1:CAS:528:DyaE3cXkt1yrtLY%3D 5446414
    • AL Fites GS Banker VF Smolen 1970 Controlled drug release through polymeric films J Pharm Sci 59 610 613 10.1002/jps.2600590507 1:CAS:528:DyaE3cXkt1yrtLY%3D 5446414
    • (1970) J Pharm Sci , vol.59 , pp. 610-613
    • Fites, A.L.1    Banker, G.S.2    Smolen, V.F.3
  • 9
    • 0018772747 scopus 로고
    • Sustained release of drugs from ethylcellulose-polyethylene glycol films and kinetics of drug release
    • 10.1002/jps.2600680318 1:CAS:528:DyaE1MXhslClsL4%3D 34023
    • Y Samuelov M Donbrow M Friedman 1979 Sustained release of drugs from ethylcellulose-polyethylene glycol films and kinetics of drug release J Pharm Sci 68 325 329 10.1002/jps.2600680318 1:CAS:528:DyaE1MXhslClsL4%3D 34023
    • (1979) J Pharm Sci , vol.68 , pp. 325-329
    • Samuelov, Y.1    Donbrow, M.2    Friedman, M.3
  • 10
    • 0022408524 scopus 로고
    • Osmotic flow through controlled porosity films: An approach to delivery of water soluble compounds
    • 10.1016/0168-3659(85)90047-1 1:CAS:528:DyaL28Xls1egtw%3D%3D
    • GM Zentner GS Rork KJ Himmelstein 1985 Osmotic flow through controlled porosity films: an approach to delivery of water soluble compounds J Control Release 2 217 229 10.1016/0168-3659(85)90047-1 1:CAS:528:DyaL28Xls1egtw%3D%3D
    • (1985) J Control Release , vol.2 , pp. 217-229
    • Zentner, G.M.1    Rork, G.S.2    Himmelstein, K.J.3
  • 11
    • 0026346882 scopus 로고
    • Modifying the release properties of Eudragit L30D
    • 10.3109/03639049109048089
    • NA Muhammed W Boisvert MR Harris J Weiss 1991 Modifying the release properties of Eudragit L30D Drug Dev Ind Pharm 17 2497 2509 10.3109/ 03639049109048089
    • (1991) Drug Dev Ind Pharm , vol.17 , pp. 2497-2509
    • Muhammed, N.A.1    Boisvert, W.2    Harris, M.R.3    Weiss, J.4
  • 12
    • 33645865531 scopus 로고    scopus 로고
    • Use of k-carrageenan as alternative pelletisation aid to microcrystalline cellulose in extrusion/spheronisation. II. Influence of drug and filler type
    • 10.1016/j.ejpb.2005.10.003 1:CAS:528:DC%2BD28XjtFGhurY%3D 16325384
    • M Thommes P Kleinebudde 2006 Use of k-carrageenan as alternative pelletisation aid to microcrystalline cellulose in extrusion/spheronisation. II. Influence of drug and filler type Eur J Pharm Biopharm 63 68 75 10.1016/j.ejpb.2005.10.003 1:CAS:528:DC%2BD28XjtFGhurY%3D 16325384
    • (2006) Eur J Pharm Biopharm , vol.63 , pp. 68-75
    • Thommes, M.1    Kleinebudde, P.2
  • 13
    • 0032870844 scopus 로고    scopus 로고
    • Influence of the process parameters on the characteristics of starch based hot stage extrudates
    • DOI 10.1016/S0378-5173(99)00229-X, PII S037851739900229X
    • D Henrist JP Remon 1999 Influence of the process parameters on the characteristics of starch based hot stage extrudates Int J Pharm 189 7 17 10.1016/S0378-5173(99)00229-X 1:CAS:528:DyaK1MXmsV2qsbw%3D 10518681 (Pubitemid 29460761)
    • (1999) International Journal of Pharmaceutics , vol.189 , Issue.1 , pp. 7-17
    • Henrist, D.1    Remon, J.P.2
  • 14
    • 38749090965 scopus 로고    scopus 로고
    • The significance of variation in extrusion speeds and temperatures on a PEO/PCL blend based matrix for oral drug delivery
    • DOI 10.1016/j.ijpharm.2007.09.041, PII S0378517307008253
    • JG Lyons P Blackie CL Higginbotham 2008 The significance of variation in extrusion speeds and temperatures on a PEO/PCL blend based matrix for oral drug delivery Int J Pharm 351 201 208 10.1016/j.ijpharm.2007.09.041 1:CAS:528:DC%2BD1cXhs1Ohurc%3D 18036753 (Pubitemid 351186863)
    • (2008) International Journal of Pharmaceutics , vol.351 , Issue.1-2 , pp. 201-208
    • Lyons, J.G.1    Blackie, P.2    Higginbotham, C.L.3
  • 15
    • 0023847840 scopus 로고    scopus 로고
    • Polymeric microspheres as drug carriers
    • 10.1016/0142-9612(88)90081-6
    • SS Davis L Illum 1999 Polymeric microspheres as drug carriers Biomaterials 9 111 115 10.1016/0142-9612(88)90081-6
    • (1999) Biomaterials , vol.9 , pp. 111-115
    • Davis, S.S.1    Illum, L.2
  • 16
    • 0036805133 scopus 로고    scopus 로고
    • Development and evaluation of prolonged release pellets obtained by the melt pelletization process
    • DOI 10.1016/S0378-5173(02)00348-4, PII S0378517302003484
    • J Hamdani AJ Moes K Amighi 2002 Development and evaluation of prolonged release pellets obtained by the melt pelletization process Int J Pharm 245 167 177 10.1016/S0378-5173(02)00348-4 1:CAS:528:DC%2BD38XntFygs74%3D 12270253 (Pubitemid 35299902)
    • (2002) International Journal of Pharmaceutics , vol.245 , Issue.1-2 , pp. 167-177
    • Hamdani, J.1    Moes, A.J.2    Amighi, K.3
  • 17
    • 23944483499 scopus 로고    scopus 로고
    • Novel lipid-based formulations enhancing the in vitro dissolution and permeability characteristics of a poorly water-soluble model drug, piroxicam
    • DOI 10.1016/j.ijpharm.2005.05.032, PII S0378517305003467
    • S Prabhu M Ortega C Ma 2005 Novel lipid based formulations enhancing the in vitro dissolution and permeability characteristics of a poorly water-soluble model drug, piroxicam Int J Pharm 301 209 216 10.1016/j.ijpharm.2005.05.032 1:CAS:528:DC%2BD2MXptVWhtro%3D 16046087 (Pubitemid 41206605)
    • (2005) International Journal of Pharmaceutics , vol.301 , Issue.1-2 , pp. 209-216
    • Prabhu, S.1    Ortega, M.2    Ma, C.3
  • 18
    • 53549102484 scopus 로고    scopus 로고
    • An investigation into the mechanism of drug release from taste-masking fatty acid microspheres
    • 10.1002/jps.21243 1:CAS:528:DC%2BD1cXhtVyltL%2FP 18200505
    • S Qi D Deutsch DQ Craig 2008 An investigation into the mechanism of drug release from taste-masking fatty acid microspheres J Pharm Sci. 97 3842 3854 10.1002/jps.21243 1:CAS:528:DC%2BD1cXhtVyltL%2FP 18200505
    • (2008) J Pharm Sci. , vol.97 , pp. 3842-3854
    • Qi, S.1    Deutsch, D.2    Craig, D.Q.3
  • 19
    • 0038683266 scopus 로고    scopus 로고
    • Physical and thermal characterisation of Precirol® and Compritol® as lipophilic glycerides used for the preparation of controlled-release matrix pellets
    • DOI 10.1016/S0378-5173(03)00229-1
    • J Hamdani AJ Moes K Amighi 2003 Physical and thermal characterization of Precirol® and Compritol® as lipophilic glycerides used for the preparation of controlled release matrix pellets Int J Pharm 260 47 57 10.1016/S0378-5173(03)00229-1 1:CAS:528:DC%2BD3sXksFKrt70%3D 12818809 (Pubitemid 36724860)
    • (2003) International Journal of Pharmaceutics , vol.260 , Issue.1 , pp. 47-57
    • Hamdani, J.1    Moes, A.J.2    Amighi, K.3
  • 20
    • 0342617694 scopus 로고    scopus 로고
    • Lipid based vehicles for the oral delivery of poorly water soluble drugs
    • 10.1016/S0169-409X(96)00494-2 1:CAS:528:DyaK2sXhtlOqs70%3D
    • AJ Humberstone WN Charman 1997 Lipid based vehicles for the oral delivery of poorly water soluble drugs Adv Drug Deliv Rev 25 103 128 10.1016/S0169-409X(96)00494-2 1:CAS:528:DyaK2sXhtlOqs70%3D
    • (1997) Adv Drug Deliv Rev , vol.25 , pp. 103-128
    • Humberstone, A.J.1    Charman, W.N.2
  • 21
    • 38949117575 scopus 로고    scopus 로고
    • Approaches for the development of solid and semi-solid lipid-based formulations
    • DOI 10.1016/j.addr.2007.09.006, PII S0169409X0700316X
    • V Jannin J Musakhanian D Marchaud 2008 Approaches for the development of solid and semi-solid lipid-based formulations Adv Drug Del Rev 60 734 746 10.1016/j.addr.2007.09.006 1:CAS:528:DC%2BD1cXitVOmsro%3D (Pubitemid 351215578)
    • (2008) Advanced Drug Delivery Reviews , vol.60 , Issue.6 , pp. 734-746
    • Jannin, V.1    Musakhanian, J.2    Marchaud, D.3
  • 22
    • 54849425743 scopus 로고    scopus 로고
    • Controlled release of active as a consequence of the die diameter in solid lipid extrusion
    • 10.1016/j.jconrel.2008.07.033 1:CAS:528:DC%2BD1cXhtlWhtrzO 18725256
    • A Michalk VR Kanikanti HJ Hamann P Kleinebudde 2008 Controlled release of active as a consequence of the die diameter in solid lipid extrusion J Control Release 132 35 41 10.1016/j.jconrel.2008.07.033 1:CAS:528:DC%2BD1cXhtlWhtrzO 18725256
    • (2008) J Control Release , vol.132 , pp. 35-41
    • Michalk, A.1    Kanikanti, V.R.2    Hamann, H.J.3    Kleinebudde, P.4
  • 23
    • 57349104188 scopus 로고    scopus 로고
    • Understanding the solid-state behavior of triglyceride solid lipid extrudates and its influence on dissolution
    • 10.1016/j.ejpb.2008.05.015 1:CAS:528:DC%2BD1cXhsV2lurfJ 18588976
    • M Windbergs CJ Strachan P Kleinebudde 2009 Understanding the solid-state behavior of triglyceride solid lipid extrudates and its influence on dissolution Eur J Pharm Biopharm 71 80 87 10.1016/j.ejpb.2008.05.015 1:CAS:528: DC%2BD1cXhsV2lurfJ 18588976
    • (2009) Eur J Pharm Biopharm , vol.71 , pp. 80-87
    • Windbergs, M.1    Strachan, C.J.2    Kleinebudde, P.3
  • 25
    • 0035127104 scopus 로고    scopus 로고
    • Assessment of the extrudability of three different mixtures of saturated polyglycolysed glycerides by determination of the "specific work of extrusion" and by capillary rheometry
    • DOI 10.1081/PDT-100000045
    • J Pinto NP Silverio 2001 Assesment of the extrudability of three different mixtures of saturated polyglycolysed glycerides by determination of the "specific work of extrusion" and cappillar rheometry Pharm Dev Technol 6 117 128 10.1081/PDT-100000045 1:CAS:528:DC%2BD3MXhslGnurg%3D 11247271 (Pubitemid 32183149)
    • (2001) Pharmaceutical Development and Technology , vol.6 , Issue.1 , pp. 117-128
    • Pinto, J.F.1    Silverio, N.R.2
  • 26
    • 53849111543 scopus 로고    scopus 로고
    • Solid lipid extrudates as sustained-release matrices: The effect of surface structure on drug release properties
    • 10.1016/j.ejps.2008.08.002 1:CAS:528:DC%2BD1cXht1Klt7jM 18765281
    • C Reitz C Strachan P Kleinebudde 2008 Solid lipid extrudates as sustained-release matrices: the effect of surface structure on drug release properties Eur J Pharm Sci 35 335 343 10.1016/j.ejps.2008.08.002 1:CAS:528:DC%2BD1cXht1Klt7jM 18765281
    • (2008) Eur J Pharm Sci , vol.35 , pp. 335-343
    • Reitz, C.1    Strachan, C.2    Kleinebudde, P.3
  • 27
    • 67349085469 scopus 로고    scopus 로고
    • Influence of polyethylene glycol/polyethylene oxide on the release characteristics of sustained-release ethylcellulose mini-matrices produced by hot-melt extrusion: In vitro and in vivo evaluations
    • 10.1016/j.ejpb.2009.01.006 1:CAS:528:DC%2BD1MXmtVOisrs%3D 19462482
    • E Verhoeven TRM De Beer E Schacht G Van den Mooter JP Remon C Vervaet 2009 Influence of polyethylene glycol/polyethylene oxide on the release characteristics of sustained-release ethylcellulose mini-matrices produced by hot-melt extrusion: in vitro and in vivo evaluations Eur J Pharm Biopharm 72 463 470 10.1016/j.ejpb.2009.01.006 1:CAS:528:DC%2BD1MXmtVOisrs%3D 19462482
    • (2009) Eur J Pharm Biopharm , vol.72 , pp. 463-470
    • Verhoeven, E.1    De Beer, T.R.M.2    Schacht, E.3    Van Den Mooter, G.4    Remon, J.P.5    Vervaet, C.6
  • 28
    • 34250867420 scopus 로고    scopus 로고
    • New insight into the role of polyethylene glycol acting as protein release modifier in lipidic implants
    • DOI 10.1007/s11095-007-9271-y
    • S Herrmann S Mohl F Siepmann J Siepmann G Winter 2007 New insights into the role of polyethylene glycol acting as protein release modifier in lipidic implants Pharm Res 8 1527 1537 10.1007/s11095-007-9271-y (Pubitemid 46988219)
    • (2007) Pharmaceutical Research , vol.24 , Issue.8 , pp. 1527-1537
    • Herrmann, S.1    Mohl, S.2    Siepmann, F.3    Siepmann, J.4    Winter, G.5
  • 29
    • 67649132600 scopus 로고    scopus 로고
    • Tailor-made dissolution profiles by extruded matrices based on lipid polyethylene glycol mixtures
    • 10.1016/j.jconrel.2009.04.002 1:CAS:528:DC%2BD1MXnslKis7g%3D 19358867
    • M Windbergs CJ Strachan P Kleinebudde 2009 Tailor-made dissolution profiles by extruded matrices based on lipid polyethylene glycol mixtures J Control Release 137 211 216 10.1016/j.jconrel.2009.04.002 1:CAS:528: DC%2BD1MXnslKis7g%3D 19358867
    • (2009) J Control Release , vol.137 , pp. 211-216
    • Windbergs, M.1    Strachan, C.J.2    Kleinebudde, P.3
  • 30
    • 67349228462 scopus 로고    scopus 로고
    • Influence of structural variations on drug release from lipid/polyethylene glycol matrices
    • 10.1016/j.ejps.2009.04.010 1:CAS:528:DC%2BD1MXnsFKrtb0%3D 19406229
    • M Windbergs CJ Strachan P Kleinebudde 2009 Influence of structural variations on drug release from lipid/polyethylene glycol matrices Eur J Pharm Sci 37 555 562 10.1016/j.ejps.2009.04.010 1:CAS:528:DC%2BD1MXnsFKrtb0%3D 19406229
    • (2009) Eur J Pharm Sci , vol.37 , pp. 555-562
    • Windbergs, M.1    Strachan, C.J.2    Kleinebudde, P.3
  • 31
    • 0242665684 scopus 로고    scopus 로고
    • Influence of melt drawing on the morphology of one- and two-step processed LDPE/Thermoplastic starch blends
    • 10.1002/adv.10057 1:CAS:528:DC%2BD3sXovVagtbo%3D
    • FJ Rodriguez-Gonzalez N Virgilio BA Ramsay BD Favis 2003 Influence of melt drawing on the morphology of one- and two-step processed LDPE/Thermoplastic starch blends Adv Polym Tech 22 297 305 10.1002/adv.10057 1:CAS:528: DC%2BD3sXovVagtbo%3D
    • (2003) Adv Polym Tech , vol.22 , pp. 297-305
    • Rodriguez-Gonzalez, F.J.1    Virgilio, N.2    Ramsay, B.A.3    Favis, B.D.4
  • 32
    • 0001774713 scopus 로고
    • Thermal behaviour and polymorphism of acylglycerides
    • N. Garti K. Sato (eds). Marcel Dekker New York
    • Hagemann JW. Thermal behaviour and polymorphism of acylglycerides. In: Garti N, Sato K, editors. Crystallization and polymorphism of fats and fatty acids. New York: Marcel Dekker; 1988. p. 9-95.
    • (1988) Crystallization and Polymorphism of Fats and Fatty Acids , pp. 9-95
    • Hagemann, J.W.1
  • 33
    • 0025778655 scopus 로고
    • Characterisation of polyethylene glycols using differential scanning calorimetry
    • 10.1016/0378-5173(91)90405-D 1:CAS:528:DyaK3MXls1Kms74%3D
    • DQM Craig JM Newton 1991 Characterisation of polyethylene glycols using differential scanning calorimetry Int J Pharm 74 33 41 10.1016/0378-5173(91) 90405-D 1:CAS:528:DyaK3MXls1Kms74%3D
    • (1991) Int J Pharm , vol.74 , pp. 33-41
    • Craig, D.Q.M.1    Newton, J.M.2
  • 35
    • 34648818909 scopus 로고    scopus 로고
    • Drug solubility in phospholipid carrier as a predictive parameter for drug recovery in microparticles produced by the aerosol solvent extraction system (ASES) process
    • DOI 10.1080/03639040601128670, PII 782313400
    • N Sarisuta S Kunstitchai L Pichert BW Mueller 2007 Drug solubility in phospholipid carrier as a predictive parameter for drug recovery in microparticles produced by the aerosol solvent extraction system (ASES) process Drug Dev Ind Pharm 33 932 944 10.1080/03639040601128670 1:CAS:528: DC%2BD2sXhtVKqsL7P 17891579 (Pubitemid 47463798)
    • (2007) Drug Development and Industrial Pharmacy , vol.33 , Issue.9 , pp. 932-944
    • Sarisuta, N.1    Kunastitchai, S.2    Pichert, L.3    Muller, B.W.4
  • 36
    • 64649103561 scopus 로고    scopus 로고
    • Chemical imaging of oral solid dosage forms and changes upon dissolution using coherent anti-Stokes Raman scattering
    • 10.1021/ac8020856 1:CAS:528:DC%2BD1MXhslCisrc%3D
    • M Windbergs M Jurna HL Offerhaus JL Herek P Kleinebudde CJ Strachan 2009 Chemical imaging of oral solid dosage forms and changes upon dissolution using coherent anti-Stokes Raman scattering Anal Chem 81 2085 2091 10.1021/ac8020856 1:CAS:528:DC%2BD1MXhslCisrc%3D
    • (2009) Anal Chem , vol.81 , pp. 2085-2091
    • Windbergs, M.1    Jurna, M.2    Offerhaus, H.L.3    Herek, J.L.4    Kleinebudde, P.5    Strachan, C.J.6


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.