On the bioactive conformation of NAN-190 (1) and MP3022 (2), 5-HT(1A) receptor antagonists

Journal of Medicinal Chemistry

Volumn 42, Issue 24, 1999, Pages 4952-4960

  Paluchowska, Maria H ^a   Mokrosz, Maria J ^a   Bojarski, Andrzej ^a   Wesołowska, Anna ^a   Borycz, Jolanta ^a   Charakchieva Minol, Sijka ^a   Chojnacka Wójcik, Ewa ^a  

^a INSTITUTE OF PHARMACOLOGY   (Poland)

Author keywords

[No Author keywords available]

Indexed keywords

1 (2 METHOXYPHENYL) 4 (4 PHTHALIMIDOBUTYL)PIPERAZINE; 2 DIPROPYLAMINO 8 HYDROXYTETRALIN; RESERPINE; SEROTONIN 1A ANTAGONIST;

ANIMAL BEHAVIOR; ANIMAL EXPERIMENT; ARTICLE; BEHAVIOR MODIFICATION; CONTROLLED STUDY; DRUG ACTIVITY; DRUG CONFORMATION; DRUG RECEPTOR BINDING; DRUG STRUCTURE; DRUG SYNTHESIS; NONHUMAN; POSTSYNAPTIC INHIBITION; RAT;

ANIMALS; BEHAVIOR, ANIMAL; LIP; MALE; MODELS, MOLECULAR; MOLECULAR CONFORMATION; MOLECULAR STRUCTURE; MOTOR ACTIVITY; PHTHALIMIDES; PIPERAZINES; POSTURE; RATS; RATS, WISTAR; RECEPTORS, SEROTONIN; RECEPTORS, SEROTONIN, 5-HT1; SEROTONIN ANTAGONISTS; STRUCTURE-ACTIVITY RELATIONSHIP; TRIAZOLES;

EID: 0033518263     PISSN: 00222623     EISSN: None     Source Type: Journal    
DOI: 10.1021/jm991045h     Document Type: Article

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