SCOPUS 정보 검색 플랫폼

Volumn 7, Issue 17, 2009, Pages 3421-3429

Synthesis of 3-(1,2,3-triazol-1-yl)- and 3-(1,2,3-triazol-4-yl)-substituted pyrazolo[3,4-d]pyrimidin-4-amines via click chemistry: Potential inhibitors of the Plasmodium falciparum PfPK7 protein kinase

(5) Klein, Michael a Dinér, Peter a Dorin Semblat, Dominique b Doerig, Christian b Grøtli, Morten a

a UNIVERSITY OF GOTHENBURG (Sweden)

b EPFL (Switzerland)

Author keywords

[No Author keywords available]

Indexed keywords

CLICK CHEMISTRY; FURTHER DEVELOPMENT; ONE POT; ORGANIC AZIDES; PLASMODIUM FALCIPARUM; POTENTIAL INHIBITORS; POTENTIALLY UNSTABLE; PROTEIN KINASE; TARGET COMPOUND; TWO-STEP REACTIONS;

AMINATION; AMINES; ISOMERS;

LEAD COMPOUNDS;

AMINE; MITOGEN ACTIVATED PROTEIN KINASE KINASE; PK7 PROTEIN, PLASMODIUM FALCIPARUM; PROTEIN KINASE; PROTEIN KINASE INHIBITOR; PROTOZOAL PROTEIN; PYRIMIDINE DERIVATIVE; TRIAZOLE DERIVATIVE;

ARTICLE; DRUG ANTAGONISM; DRUG EFFECT; ENZYMOLOGY; IC 50; PLASMODIUM FALCIPARUM; STRUCTURE ACTIVITY RELATION; SYNTHESIS;

AMINES; INHIBITORY CONCENTRATION 50; MITOGEN-ACTIVATED PROTEIN KINASE KINASES; PLASMODIUM FALCIPARUM; PROTEIN KINASE INHIBITORS; PROTEIN KINASES; PROTOZOAN PROTEINS; PYRIMIDINES; STRUCTURE-ACTIVITY RELATIONSHIP; TRIAZOLES;

PLASMODIUM FALCIPARUM;

EID: 70349278432 PISSN: 14770520 EISSN: None Source Type: Journal
DOI: 10.1039/b906482f Document Type: Article

Times cited : (50)

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