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Volumn 4, Issue 7, 2009, Pages 1189-1195

Discovery of selective luteinizing hormone receptor agonists using the bivalent ligand method

(8) Bonger, Kimberly M a Van Den Berg, Richard J B H N a Knijnenburg, Annemiek D a Heitman, Laura H b Van Koppen, Chris J c Timmers, Cornelis M c Overkleeft, Herman S a Van Der Marel, Gijsbert A a

a LEIDEN UNIVERSITY (Netherlands)

b LEIDEN UNIVERSITY (Netherlands)

c MERCK RESEARCH LABORATORIES (United States)

Author keywords

Medicinal chemistry; Membrane proteins; Receptors; Signal transduction; Structure activity relationships

Indexed keywords

CARBOXYLIC ACID; FOLLICLE STIMULATING HORMONE RECEPTOR; G PROTEIN COUPLED RECEPTOR; GLYCOPROTEIN HORMONE RECEPTOR; HORMONE RECEPTOR; LIGAND; LUTEINIZING HORMONE RECEPTOR; LUTEINIZING HORMONE RECEPTOR AGONIST; MONOMER; UNCLASSIFIED DRUG;

ARTICLE; CHEMICAL STRUCTURE; CONTROLLED STUDY; DIMERIZATION; EVALUATION RESEARCH; MEMBRANE POTENTIAL; MOLECULAR WEIGHT; PRIORITY JOURNAL; STRUCTURE ANALYSIS; SYNTHESIS;

BENZENE; DRUG DISCOVERY; ETHYLENE GLYCOL; FOLLICLE STIMULATING HORMONE; LIGANDS; RECEPTORS, LH; RECOMBINANT PROTEINS; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 67749127694 PISSN: 18607179 EISSN: 18607187 Source Type: Journal
DOI: 10.1002/cmdc.200900058 Document Type: Article

Times cited : (14)

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