SCOPUS 정보 검색 플랫폼

Volumn 4, Issue 5, 2009, Pages 780-791

Highly potent naphthofuran-based retinoic acid receptor agonists

(7) Santín, Efrén Pérez b Khanwalkar, Harshal a Voegel, Johannes c Collette, Pascal c Mauvais, Pascale c Gronemeyer, Hinrich a De Lera, Ángel R b

a CNRS (France)

b UNIVERSITY OF VIGO (Spain)

c Galderma R and D (France)

Author keywords

Agonists; Antagonists; Arotinoids; Retinoid receptor subtypes; Transactivation

Indexed keywords

4 (3 BROMO 5,5,8,8 TETRAMETHYL 5,6,7,8 TETRAHYDRONAPHTHO[2,3 B]FURAN 2 YL)BENZOIC ACID; 4 (3 CHLORO 5,5,8,8 TETRAMETHYL 5,6,7,8 TETRAHYDRONAPHTHO[2,3 B]FURAN 2 YL)BENZOIC ACID; 4 (3 IODO 5,5,8,8 TETRAMETHYL 5,6,7,8 TETRAHYDRONAPHTHO[2,3 B]FURAN 2 YL)BENZOIC ACID; 4 (5,5,8,8 TETRAMETHYL 3 4 TOLYL 5,6,7,8 TETRAHYDRONAPHTHO[2,3 B]FURAN 2 YL)BENZOIC ACID; 4 (5,5,8,8 TETRAMETHYL 3 PHENYL 5,6,7,8 TETRAHYDRONAPHTHO[2,3 B]FURAN 2 YL)BENZOIC ACID; 4 (5,5,8,8 TETRAMETHYL 5,6,7,8 TETRAHYDRONAPHTHO[2,3 B]FURAN 2 YL)BENZOIC ACID; 4 [3 (3,3 DIMETHYLBUT 1 YNYL) 5,5,8,8 TETRAMETHYL 5,6,7,8 TETRAHYDRONAPHTHO[2,3 B]FURAN 2 YL]BENZOIC ACID; 4 [3 (4 FORMYLPHENYL) 5,5,8,8 TETRAMETHYL 5,6,7,8 TETRAHYDRONAPHTHO[2,3 B]FURAN 2 YL]BENZOIC ACID; 4 [3 (4 METHOXYPHENYL) 5,5,8,8 TETRAMETHYL 5,6,7,8 TETRAHYDRONAPHTHO[2,3 B]FURAN 2 YL]BENZOIC ACID; 4 [3 (BIPHENYL 4 YL) 5,5,8,8 TETRAMETHYL 5,6,7,8 TETRAHYDRONAPHTHO[2,3 B]FURAN 2 YL]BENZOIC ACID; 4 [5,5,8,8 TETRAMETHYL 3 (2 PHENYLETHEN 1 YL) 5,6,7,8 TETRAHYDRONAPHTHO[2,3 B]FURAN 2 YL]BENZOIC ACID; ANTINEOPLASTIC AGENT; AROTINOID; ETHYL 4 (3 IODO 5,5,8,8 TETRAMETHYL 5,6,7,8 TETRAHYDRONAPHTHO[2,3 B]FURAN 2 YL)BENZOIC ACID; ETHYL 4 (5,5,8,8 TETRAMETHYL 3 4 TOLYL 5,6,7,8 TETRAHYDRONAPHTHO[2,3 B]FURAN 2 YL)BENZOIC ACID; ETHYL 4 (5,5,8,8 TETRAMETHYL 3 PHENYL 5,6,7,8 TETRAHYDRONAPHTHO[2,3 B]FURAN 2 YL)BENZOIC ACID; ETHYL 4 [(3 METHOXY 5,5,8,8 TETRAMETHYL 5,6,7,8 TETRAHYDRONAPHTHALEN 2 YL)ETHYNYL]BENZOIC ACID; ETHYL 4 [3 (3,3 DIMETHYLBUT 1 YNYL) 5,5,8,8 TETRAMETHYL 5,6,7,8 TETRAHYDRONAPHTHO[2,3 B]FURAN 2 YL]BENZOIC ACID; ETHYL 4 [3 (4 FORMYLPHENYL) 5,5,8,8 TETRAMETHYL 5,6,7,8 TETRAHYDRONAPHTHO[2,3 B]FURAN 2 YL]BENZOIC ACID; ETHYL 4 [3 (4 METHOXYPHENYL) 5,5,8,8 TETRAMETHYL 5,6,7,8 TETRAHYDRONAPHTHO[2,3 B]FURAN 2 YL]BENZOIC ACID; ETHYL 4 [3 (BIPHENYL 4 YL) 5,5,8,8 TETRAMETHYL 5,6,7,8 TETRAHYDRONAPHTHO[2,3 B]FURAN 2 YL]BENZOIC ACID; ETHYL 4 [5,5,8,8 TETRAMETHYL 3 (2 PHENYLETHEN 1 YL) 5,6,7,8 TETRAHYDRONAPHTHO[2,3 B]FURAN 2 YL]BENZOIC ACID; RETINOIC ACID DERIVATIVE; UNCLASSIFIED DRUG; BENZOFURAN; BENZOFURAN DERIVATIVE; ISOPROTEIN; RETINOIC ACID RECEPTOR;

ARTICLE; CONTROLLED STUDY; CYCLIZATION; DRUG POTENCY; DRUG STRUCTURE; DRUG SYNTHESIS; HUMAN; HUMAN CELL; PRIORITY JOURNAL; SONOGASHIRA REACTION; SUBSTITUTION REACTION; SUZUKI REACTION; CHEMISTRY; DRUG EFFECT; DRUG POTENTIATION; GENETIC TRANSCRIPTION; HELA CELL; METABOLISM; SYNTHESIS; TUMOR CELL LINE;

BENZOFURANS; CELL LINE, TUMOR; HELA CELLS; HUMANS; PROTEIN ISOFORMS; RECEPTORS, RETINOIC ACID; TRANSCRIPTION, GENETIC;

EID: 67651109038 PISSN: 18607179 EISSN: 18607187 Source Type: Journal
DOI: 10.1002/cmdc.200900015 Document Type: Article

Times cited : (17)

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