Identification and functional separation of retinoic acid receptor neutral antagonists and inverse agonists

Journal of Biological Chemistry

Volumn 271, Issue 37, 1996, Pages 22692-22696

  Klein, Elliott S ^a,c   Pino, Mary E ^a   Johnson, Alan T ^a   Davies, Peter J A ^b   Nagpal, Sunil ^a   Thacher, Scott M ^a   Krasinski, Glenn ^a   Chandraratna, Roshantha A S ^a,c  

^a ALLERGAN INC   (United States)

^b UNIVERSITY OF TEXAS   (United States)

^c Mail Code RD 3D ^*  (United States)

Author keywords

[No Author keywords available]

Indexed keywords

4 [2 [5,6 DIHYDRO 5,5 DIMETHYL 8 (4 METHYLPHENYL) 2 NAPHTHYL]ETHYNYL]BENZOIC ACID; AGN 192870; AGN 193385; AGN 193389; AGN 193840; RECEPTOR BLOCKING AGENT; RETINOIC ACID RECEPTOR; RETINOID; UNCLASSIFIED DRUG;

ARTICLE; CONTROLLED STUDY; DISSOCIATION CONSTANT; DOSE RESPONSE; DRUG RECEPTOR BINDING; GENE EXPRESSION REGULATION; HUMAN; HUMAN CELL; KERATINOCYTE; LIGAND BINDING; PRIORITY JOURNAL; SKIN; TRANSACTIVATION; TRANSCRIPTION REGULATION;

ANTIGENS, DIFFERENTIATION; BINDING, COMPETITIVE; CALCIUM-BINDING PROTEINS; CALGRANULIN A; CELLS, CULTURED; HUMANS; KERATINOCYTES; NAPHTHALENES; RECEPTORS, ADRENERGIC, BETA; RECEPTORS, RETINOIC ACID; RETINOIDS; TRANSCRIPTION, GENETIC;

EID: 0029811878     PISSN: 00219258     EISSN: None     Source Type: Journal    
DOI: 10.1074/jbc.271.37.22692     Document Type: Article

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