SCOPUS 정보 검색 플랫폼

Volumn 3, Issue 3, 2008, Pages 454-460

Reduction of lipophilicity at the lipophilic domain of RXR agonists enables production of subtype preference: RXRα-preferential agonist possessing a sulfonamide moiety

(11) Takamatsu, Kayo a Takano, Atsushi a Yakushiji, Nobumasa a Morishita, Ken Ichi a Matsuura, Nobuyasu b Makishima, Makoto c Ali, Hamed Ismail d Akaho, Eiichi d Tai, Akihiro a Sasaki, Kenji a Kakuta, Hiroki a

a OKAYAMA UNIVERSITY (Japan)

b OKAYAMA UNIVERSITY OF SCIENCE (Japan)

c NIHON UNIVERSITY SCHOOL OF MEDICINE (Japan)

d KOBE GAKUIN UNIVERSITY (Japan)

Author keywords

Docking simulations; RXR agonists; Subtype preference; Subtype selectivity; Sulfonamides; Synergistic effects

Indexed keywords

ANTINEOPLASTIC AGENT; ANTIOBESITY AGENT; NITROBLUE TETRAZOLIUM; RETINOID X RECEPTOR; RETINOID X RECEPTOR ALPHA; RETINOID X RECEPTOR BETA; RETINOID X RECEPTOR GAMMA; SULFONAMIDE;

ANIMAL; ARTICLE; CELL DIFFERENTIATION; CELL STRAIN COS1; CERCOPITHECUS; CHEMICAL MODEL; DRUG EFFECT; DRUG POTENTIATION; HYDROPHOBICITY; METABOLISM; OXIDATION REDUCTION REACTION; PHYSIOLOGY; SYNTHESIS;

ANIMALS; ANTI-OBESITY AGENTS; ANTINEOPLASTIC AGENTS; CELL DIFFERENTIATION; CERCOPITHECUS AETHIOPS; COS CELLS; DRUG SYNERGISM; HYDROPHOBICITY; MODELS, CHEMICAL; NITROBLUE TETRAZOLIUM; OXIDATION-REDUCTION; RETINOID X RECEPTOR ALPHA; RETINOID X RECEPTOR BETA; RETINOID X RECEPTOR GAMMA; RETINOID X RECEPTORS; SULFONAMIDES;

EID: 48049114021 PISSN: 18607179 EISSN: 18607187 Source Type: Journal
DOI: 10.1002/cmdc.200700265 Document Type: Article

Times cited : (24)

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