Second Annual GPCRs: From Orphan to Blockbuster

Expert Opinion on Therapeutic Targets

Volumn 8, Issue 5, 2004, Pages 495-498

  Gilchrist, Annette ^a  

^a Cue BIOtech   (United States)

Author keywords

Agonist; Antagonist; Conformational change; G protein coupled receptor (GPCR); Inverse agonist; Signal transduction

Indexed keywords

G PROTEIN COUPLED RECEPTOR; LIGAND; NICOTINIC ACID;

CONFERENCE PAPER; CONFORMATIONAL TRANSITION; DRUG INDUSTRY; DRUG TARGETING; HIGH THROUGHPUT SCREENING; METHODOLOGY; NONHUMAN; PROTEIN EXPRESSION; PROTEIN FUNCTION; PROTEIN STRUCTURE; UNITED STATES;

ALLOSTERIC REGULATION; ANIMALS; CLONING, MOLECULAR; DRUG DESIGN; DRUG EVALUATION, PRECLINICAL; FEMALE; HUMANS; LIGANDS; MALE; MICE; MULTIGENE FAMILY; PROTEIN BINDING; PROTEIN CONFORMATION; RECEPTORS, G-PROTEIN-COUPLED; SIGNAL TRANSDUCTION; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 5444258762     PISSN: 14728222     EISSN: None     Source Type: Journal    
DOI: 10.1517/14728222.8.5.495     Document Type: Conference Paper

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