Polymer-based open-channel blockers for the acetylcholine receptor: The effect of spacer length on blockade kinetics

Biochemistry

Volumn 47, Issue 35, 2008, Pages 9163-9173

  Lin, Wan Chen ^a   Licht, Stuart ^a  

^a MASSACHUSETTS INSTITUTE OF TECHNOLOGY   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ABS RESINS; ASSOCIATION REACTIONS; CHLORINE COMPOUNDS; COMPUTER NETWORKS; ETHYLENE; ETHYLENE GLYCOL; GLYCOLS; OPEN CHANNEL FLOW; POLYETHYLENE GLYCOLS; POLYMERS;

ACETYLCHOLINE RECEPTORS; CHANNEL BLOCKERS; SPACER LENGTHS;

RATE CONSTANTS;

BIS(TRIMETHYLAMMONIUM); BLOCKING AGENT; CHOLINERGIC RECEPTOR; DECAMETHONIUM; ION CHANNEL; MACROGOL DERIVATIVE; POLYMER; TETRYLAMMONIUM; TRIMETHYLAMMONIUM SALT DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; CHEMICAL STRUCTURE; ELECTROPHYSIOLOGY; PRIORITY JOURNAL; SYMPATHETIC BLOCKING;

ANIMALS; CHOLINERGIC ANTAGONISTS; HUMANS; KINETICS; MICE; POLYETHYLENE GLYCOLS; RECEPTORS, CHOLINERGIC; TRIMETHYL AMMONIUM COMPOUNDS;

EID: 50849135894     PISSN: 00062960     EISSN: None     Source Type: Journal    
DOI: 10.1021/bi800737j     Document Type: Article

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