Binding of orthosteric ligands to the allosteric site of the M2 muscarinic cholinergic receptor

Molecular Pharmacology

Volumn 74, Issue 3, 2008, Pages 834-843

  Redka, Dar'ya S ^a   Pisterzi, Luca F ^a   Wells, James W ^a  

^a UNIVERSITY OF TORONTO   (Canada)

Author keywords

[No Author keywords available]

Indexed keywords

GALLAMINE; HEMAGGLUTININ; METHYLSCOPOLAMINE; MUSCARINIC M2 RECEPTOR; OBIDOXIME; OLIGOMER; OXOTREMORINE M;

ANIMAL CELL; ARTICLE; BINDING SITE; CONTROLLED STUDY; CROSS LINKING; IMMUNOPRECIPITATION; LIGAND BINDING; NONHUMAN; PRIORITY JOURNAL; RECEPTOR AFFINITY; RECEPTOR BINDING;

ALLOSTERIC REGULATION; ALLOSTERIC SITE; ANIMALS; BINDING, COMPETITIVE; CELL LINE; GALLAMINE TRIETHIODIDE; HUMANS; INSECTS; KINETICS; LIGANDS; N-METHYLSCOPOLAMINE; OBIDOXIME CHLORIDE; PROTEIN STRUCTURE, QUATERNARY; RECEPTOR, MUSCARINIC M2; SOLUBILITY;

EID: 50449091828     PISSN: 0026895X     EISSN: 15210111     Source Type: Journal    
DOI: 10.1124/mol.108.048074     Document Type: Article

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