Interaction of Mg2+ with the allosteric site of muscarinic M2 receptors

Naunyn-Schmiedeberg's Archives of Pharmacology

Volumn 357, Issue 4, 1998, Pages 363-370

  Burgmer, Ulrike ^a   Schulz, Uwe ^a   Tränkle, Christian ^a   Mohr, Klaus ^a  

^a UNIVERSITY OF BONN   (Germany)

Author keywords

Allosteric interactions; Chin3 6; Mg2+ effects; Porcine M2 receptors; W84

Indexed keywords

1,6 HEXAMETHYLENEBIS[DIMETHYL(3 PHTHALIMIDOPROPYL)AMMONIUM BROMIDE]; CHIN 3/6; CHOLINERGIC RECEPTOR; DIVALENT CATION; LIGAND; MAGNESIUM ION; MUSCARINIC M2 RECEPTOR; UNCLASSIFIED DRUG; CHIN 3 6; CHIN 3-6; HEXAMETHONIUM; HEXAMETHYLENEBIS(DIMETHYL (3 PHTHALIMIDOPROPYL)AMMONIUM BROMIDE); HEXAMETHYLENEBIS(DIMETHYL-(3-PHTHALIMIDOPROPYL)AMMONIUM BROMIDE); MAGNESIUM; METHYLSCOPOLAMINE; MUSCARINIC RECEPTOR; PHTHALIMIDE DERIVATIVE; QUINAZOLINE DERIVATIVE;

ALLOSTERISM; ANIMAL CELL; ANIMAL TISSUE; ARTICLE; BINDING SITE; CONTROLLED STUDY; DRUG BINDING SITE; DRUG RECEPTOR BINDING; HEART; IONIC STRENGTH; LIGAND BINDING; MOLECULAR MODEL; NONHUMAN; RECEPTOR BINDING; ANIMAL; COMPARATIVE STUDY; HEART MUSCLE; METABOLISM; SWINE;

ALLOSTERIC SITE; ANIMALS; HEXAMETHONIUM COMPOUNDS; MAGNESIUM; MYOCARDIUM; N-METHYLSCOPOLAMINE; PHTHALIMIDES; QUINAZOLINES; RECEPTOR, MUSCARINIC M2; RECEPTORS, MUSCARINIC; SWINE;

EID: 0031596859     PISSN: 00281298     EISSN: None     Source Type: Journal    
DOI: 10.1007/PL00005180     Document Type: Article

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