-
1
-
-
0031916896
-
The role of central melanocortin receptors in the activation of the hypothalamus-pituitary-adrenal-axis and the induction of excessive grooming
-
Von Frijtag, J. C., Croiset, G., Gispen, W. H., Adan, R. A., and Wiegant, V. M., The role of central melanocortin receptors in the activation of the hypothalamus-pituitary-adrenal-axis and the induction of excessive grooming. Br. J. Pharmacol., 123, 1503-1508 (1998).
-
(1998)
Br. J. Pharmacol.
, vol.123
, pp. 1503-1508
-
-
Von Frijtag, J.C.1
Croiset, G.2
Gispen, W.H.3
Adan, R.A.4
Wiegant, V.M.5
-
2
-
-
0029670663
-
Behavioral effects of alpha-MSH and MCH after central administration in the female rat
-
Gonzalez, M. I., Vaziri, S., and Wilson, C. A., Behavioral effects of alpha-MSH and MCH after central administration in the female rat. Peptides, 17, 171-177 (1996).
-
(1996)
Peptides
, vol.17
, pp. 171-177
-
-
Gonzalez, M.I.1
Vaziri, S.2
Wilson, C.A.3
-
3
-
-
0025193432
-
Proconflict effect of ACTH1-24: Interaction with benzodiazepines
-
Corda, M. G., Orlandi, M., and Fratta, W., Proconflict effect of ACTH1-24: interaction with benzodiazepines. Pharmacol. Biochem. Behav., 36, 631-634 (1990).
-
(1990)
Pharmacol. Biochem. Behav.
, vol.36
, pp. 631-634
-
-
Corda, M.G.1
Orlandi, M.2
Fratta, W.3
-
4
-
-
0029839328
-
Morphine down-regulates melanocortin-4 receptor expression in brain regions that mediate opiate addiction
-
Alvaro, J. D., Tatro, J. B., Quillan, J. M., Fogliano, M., Eisenhard, M., Lerner, M. R., Nestler, E. J., and Duman, R. S., Morphine down-regulates melanocortin-4 receptor expression in brain regions that mediate opiate addiction. Mol. Pharmacol., 50, 583-591 (1996).
-
(1996)
Mol. Pharmacol.
, vol.50
, pp. 583-591
-
-
Alvaro, J.D.1
Tatro, J.B.2
Quillan, J.M.3
Fogliano, M.4
Eisenhard, M.5
Lerner, M.R.6
Nestler, E.J.7
Duman, R.S.8
-
5
-
-
0032809011
-
Characterization of melanocortin receptor ligands on cloned brain melanocortin receptors and on grooming behavior in the rat
-
Adan, R. A., Szklarczyk, A. W., Oosterom, J., Brakkee, J. H., Nijenhuis, W. A., Schaaper, W. M., Meloen, R. H., and Gispen, W. H., Characterization of melanocortin receptor ligands on cloned brain melanocortin receptors and on grooming behavior in the rat. Eur. J. Pharmacol., 378, 249-258 (1999).
-
(1999)
Eur. J. Pharmacol.
, vol.378
, pp. 249-258
-
-
Adan, R.A.1
Szklarczyk, A.W.2
Oosterom, J.3
Brakkee, J.H.4
Nijenhuis, W.A.5
Schaaper, W.M.6
Meloen, R.H.7
Gispen, W.H.8
-
6
-
-
0028134706
-
Localization of the melanocortin-4 receptor (MC4-R) in neuroendocrine and autonomic control circuits in the brain
-
Mountjoy, K. G., Mortrud, M. T., Low, M. J., Simerly, R. B., and Cone, R. D., Localization of the melanocortin-4 receptor (MC4-R) in neuroendocrine and autonomic control circuits in the brain. Mol. Endocrinol., 8, 1298-1308 (1994).
-
(1994)
Mol. Endocrinol.
, vol.8
, pp. 1298-1308
-
-
Mountjoy, K.G.1
Mortrud, M.T.2
Low, M.J.3
Simerly, R.B.4
Cone, R.D.5
-
7
-
-
0038051141
-
Molecular genetics of human obesity-associated MC4R mutations
-
Lubrano-Berthelier, C., Cavazos, M., Dubern, B., Shapiro, A., Stunff, C. L., Zhang, S., Picart, F., Govaerts, C., Froguel, P., Bougneres, P., Clement, K., and Vaisse, C., Molecular genetics of human obesity-associated MC4R mutations. Ann. N.Y. Acad. Sci., 994, 49-57 (2003).
-
(2003)
Ann. N.Y. Acad. Sci.
, vol.994
, pp. 49-57
-
-
Lubrano-Berthelier, C.1
Cavazos, M.2
Dubern, B.3
Shapiro, A.4
Stunff, C.L.5
Zhang, S.6
Picart, F.7
Govaerts, C.8
Froguel, P.9
Bougneres, P.10
Clement, K.11
Vaisse, C.12
-
8
-
-
0037310741
-
Anxiolytic-like and antidepressant-like activities of MCL0129 (1-[(S)-2-(4-fluorophenyl)-2-(4-isopropylpiperadin-1-yl)ethyl] -4-[4-(2-methoxynaphthalen-1-yl)butyl]piperazine), a novel and potent nonpeptide antagonist of the melanocortin-4 receptor
-
Chaki, S., Hirota, S., Funakoshi, T., Suzuki, Y., Suetake, S., Okubo, T., Ishii, T., Nakazato, A., and Okuyama, S., Anxiolytic-like and antidepressant-like activities of MCL0129 (1-[(S)-2-(4-fluorophenyl)-2-(4- isopropylpiperadin-1-yl)ethyl]-4-[4-(2-methoxynaphthalen-1-yl)butyl]piperazine), a novel and potent nonpeptide antagonist of the melanocortin-4 receptor. J. Pharmacol. Exp. Ther., 304, 818-826 (2003).
-
(2003)
J. Pharmacol. Exp. Ther.
, vol.304
, pp. 818-826
-
-
Chaki, S.1
Hirota, S.2
Funakoshi, T.3
Suzuki, Y.4
Suetake, S.5
Okubo, T.6
Ishii, T.7
Nakazato, A.8
Okuyama, S.9
-
9
-
-
0141811657
-
1 angiotensin receptor activation and signaling
-
1 angiotensin receptor activation and signaling. Endocrinology, 144, 2220-2228 (2003).
-
(2003)
Endocrinology
, vol.144
, pp. 2220-2228
-
-
Gaborik, Z.1
Jagadeesh, G.2
Zhang, M.3
Spat, A.4
Catt, K.J.5
Hunyady, L.6
-
10
-
-
0034817072
-
Constitutive activation of A(3) adenosine receptors by site-directed mutagenesis to create constitutively active mutant human A(3) adenosine receptors (ARs)
-
Chen, A., Gao, Z. G., Barak, D., Liang, B. T., and Jacobson, K. A., Constitutive activation of A(3) adenosine receptors by site-directed mutagenesis to create constitutively active mutant human A(3) adenosine receptors (ARs). Biochem. Biophys. Res. Commun., 284, 596-601 (2001).
-
(2001)
Biochem. Biophys. Res. Commun.
, vol.284
, pp. 596-601
-
-
Chen, A.1
Gao, Z.G.2
Barak, D.3
Liang, B.T.4
Jacobson, K.A.5
-
11
-
-
0033974265
-
Mutational analysis of the highly conserved arginine within the Glu/Asp-Arg-Tyr motif of the alpha(1b)-adrenergic receptor: Effects on receptor isomerization and activation
-
Scheer, A., Costa, T., Fanelli, F., De Benedetti, P. G., Mhaouty-Kodja, S., Abuin, L., Nenniger-Tosato, M., and Cotecchia, S., Mutational analysis of the highly conserved arginine within the Glu/Asp-Arg-Tyr motif of the alpha(1b)-adrenergic receptor: effects on receptor isomerization and activation. Mol. Pharmacol., 57, 219-231 (2000).
-
(2000)
Mol. Pharmacol.
, vol.57
, pp. 219-231
-
-
Scheer, A.1
Costa, T.2
Fanelli, F.3
De Benedetti, P.G.4
Mhaouty-Kodja, S.5
Abuin, L.6
Nenniger-Tosato, M.7
Cotecchia, S.8
-
12
-
-
0029897495
-
Constitutively active mutants of the alpha 1B-adrenergic receptor: Role of highly conserved polar amino acids in receptor activation
-
Scheer, A., Fanelli, F., Costa, T., De Benedetti, P. G., and Cotecchia, S., Constitutively active mutants of the alpha 1B-adrenergic receptor: role of highly conserved polar amino acids in receptor activation. EMBO J., 15, 3566-3578 (1996).
-
(1996)
EMBO J.
, vol.15
, pp. 3566-3578
-
-
Scheer, A.1
Fanelli, F.2
Costa, T.3
De Benedetti, P.G.4
Cotecchia, S.5
-
13
-
-
0032217226
-
The D136A mutation of the V2 vasopressin receptor induces a constitutive activity which permits discrimination between antagonists with partial agonist and inverse agonist activities
-
Morin, D., Cotte, N., Balestre, M. N., Mouillac, B., Manning, M., Breton, C., and Barberis, C., The D136A mutation of the V2 vasopressin receptor induces a constitutive activity which permits discrimination between antagonists with partial agonist and inverse agonist activities. FEBS Lett., 441, 470-475 (1998).
-
(1998)
FEBS Lett.
, vol.441
, pp. 470-475
-
-
Morin, D.1
Cotte, N.2
Balestre, M.N.3
Mouillac, B.4
Manning, M.5
Breton, C.6
Barberis, C.7
-
14
-
-
0034112037
-
The effect of mutations in the DRY motif on the constitutive activity and structural instability of the histamine H(2) receptor
-
Alewijnse, A. E., Timmerman, H., Jacobs, E. H., Smit, M. J., Roovers, E., Cotecchia, S., and Leurs, R., The effect of mutations in the DRY motif on the constitutive activity and structural instability of the histamine H(2) receptor. Mol. Pharmacol., 57, 890-898 (2000).
-
(2000)
Mol. Pharmacol.
, vol.57
, pp. 890-898
-
-
Alewijnse, A.E.1
Timmerman, H.2
Jacobs, E.H.3
Smit, M.J.4
Roovers, E.5
Cotecchia, S.6
Leurs, R.7
-
15
-
-
0035810771
-
Agouti-related protein functions as an inverse agonist at a constitutively active brain melanocortin-4 receptor
-
Haskell-Luevano, C., and Monck, E. K., Agouti-related protein functions as an inverse agonist at a constitutively active brain melanocortin-4 receptor. Regul. Pept., 99, 1-7 (2001).
-
(2001)
Regul. Pept.
, vol.99
, pp. 1-7
-
-
Haskell-Luevano, C.1
Monck, E.K.2
-
16
-
-
0035918601
-
Structure activity studies of the melanocortin-4 receptor by in vitro mutagenesis: Identification of agouti-related protein (AGRP), melanocortin agonist and synthetic peptide antagonist interaction determinants
-
Haskell-Luevano, C., Cone, R. D., Monck, E. K., and Wan, Y. P., Structure activity studies of the melanocortin-4 receptor by in vitro mutagenesis: identification of agouti-related protein (AGRP), melanocortin agonist and synthetic peptide antagonist interaction determinants. Biochem., 40, 6164-6179 (2001).
-
(2001)
Biochem.
, vol.40
, pp. 6164-6179
-
-
Haskell-Luevano, C.1
Cone, R.D.2
Monck, E.K.3
Wan, Y.P.4
-
17
-
-
0027227288
-
Molecular cloning, expression, and gene localization of a fourth melanocortin receptor
-
Gantz, I., Miwa, H., Konda, Y., Shimoto, Y., Tashiro, T., Watson, S. J., DelValle, J., and Yamada, T. J., Molecular cloning, expression, and gene localization of a fourth melanocortin receptor. J. Biol. Chem., 268, 15174-15179 (1993).
-
(1993)
J. Biol. Chem.
, vol.268
, pp. 15174-15179
-
-
Gantz, I.1
Miwa, H.2
Konda, Y.3
Shimoto, Y.4
Tashiro, T.5
Watson, S.J.6
Delvalle, J.7
Yamada, T.J.8
|