7-Substituted 2-phenyl-benzofurans as ERβ selective ligands

Bioorganic and Medicinal Chemistry Letters

Volumn 14, Issue 19, 2004, Pages 4925-4929

  Collini, Michael D ^a   Kaufman, David H ^a   Manas, Eric S ^a   Harris, Heather A ^a   Henderson, Ruth A ^a   Xu, Zhang B ^b   Unwalla, Rayomand J ^a   Miller, Chris P ^a  

^a PFIZER INC   (United States)

^b Wyeth Research   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

BENZOFURAN DERIVATIVE; ESTRADIOL; ESTROGEN RECEPTOR BETA; GENISTEIN; HORMONE RECEPTOR AFFECTING AGENT; LIGAND;

ARTICLE; BINDING AFFINITY; CHEMICAL MODIFICATION; DRUG SYNTHESIS; LIPOPHILICITY; RECEPTOR AFFINITY; STRUCTURE ACTIVITY RELATION; SUBSTITUTION REACTION;

BENZOFURANS; CELL LINE, TUMOR; ESTROGEN RECEPTOR BETA; HUMANS; INSULIN-LIKE GROWTH FACTOR BINDING PROTEIN 4; LIGANDS; RNA, MESSENGER; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 4444249445     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2004.07.029     Document Type: Article

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